HRP20050157B1 - 8-[3-amino-piperidin-1-yl]-xanthines,the production thereof and the use of the same as medicaments - Google Patents

8-[3-amino-piperidin-1-yl]-xanthines,the production thereof and the use of the same as medicaments

Info

Publication number
HRP20050157B1
HRP20050157B1 HRP20050157A HRP20050157B1 HR P20050157 B1 HRP20050157 B1 HR P20050157B1 HR P20050157 A HRP20050157 A HR P20050157A HR P20050157 B1 HRP20050157 B1 HR P20050157B1
Authority
HR
Croatia
Prior art keywords
xanthines
piperidin
medicaments
amino
production
Prior art date
Application number
Inventor
Frank Himmelsbach
Elke Langkopf
Matthias Eckhardt
Michael Mark
Roland Maier
Ralf Richard Hermann Lotz
Mohammed Tadayyon
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31947613&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20050157(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE10238243A external-priority patent/DE10238243A1/en
Priority claimed from DE10312353A external-priority patent/DE10312353A1/en
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of HRP20050157A2 publication Critical patent/HRP20050157A2/en
Publication of HRP20050157B1 publication Critical patent/HRP20050157B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
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    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
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HR20050157 2002-08-21 2005-02-18 8-[3-amino-piperidin-1-yl]-xanthines,the production thereof and the use of the same as medicaments HRP20050157B1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10238243A DE10238243A1 (en) 2002-08-21 2002-08-21 New 8-(3-amino-piperidin-1-yl)-xanthine derivatives are dipeptidylpeptidase-IV inhibitors useful for, e.g. treating diabetes mellitus, arthritis or obesity
DE10312353A DE10312353A1 (en) 2003-03-20 2003-03-20 New 8-(3-amino-piperidin-1-yl)-xanthine derivatives are dipeptidylpeptidase-IV inhibitors useful for, e.g. treating diabetes mellitus, arthritis or obesity
PCT/EP2003/009127 WO2004018468A2 (en) 2002-08-21 2003-08-18 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments

Publications (2)

Publication Number Publication Date
HRP20050157A2 HRP20050157A2 (en) 2006-05-31
HRP20050157B1 true HRP20050157B1 (en) 2013-01-31

Family

ID=31947613

Family Applications (2)

Application Number Title Priority Date Filing Date
HR20050157 HRP20050157B1 (en) 2002-08-21 2005-02-18 8-[3-amino-piperidin-1-yl]-xanthines,the production thereof and the use of the same as medicaments
HR20090665A HRP20090665A2 (en) 2002-08-21 2009-12-14 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments

Family Applications After (1)

Application Number Title Priority Date Filing Date
HR20090665A HRP20090665A2 (en) 2002-08-21 2009-12-14 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments

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EP (6) EP1532149B9 (en)
JP (6) JP4233524B2 (en)
KR (2) KR101111101B1 (en)
CN (4) CN107674077A (en)
AR (3) AR041025A1 (en)
AT (1) ATE453644T1 (en)
AU (2) AU2003253418B2 (en)
BE (1) BE2011C038I2 (en)
BR (2) BRPI0313648B8 (en)
CA (1) CA2496249C (en)
CY (3) CY1109928T1 (en)
DE (2) DE50312295D1 (en)
DK (1) DK1532149T3 (en)
EA (3) EA010303B1 (en)
EC (2) ECSP055617A (en)
EG (1) EG25011A (en)
ES (1) ES2339112T3 (en)
FR (1) FR11C0052I2 (en)
HK (6) HK1081552A1 (en)
HR (2) HRP20050157B1 (en)
HU (1) HUS1100028I1 (en)
IL (1) IL166964A (en)
IN (2) IN2015DN01133A (en)
LU (2) LU91889I2 (en)
ME (1) ME00396B (en)
MX (1) MXPA05001684A (en)
MY (2) MY137619A (en)
NO (4) NO333970B1 (en)
PE (1) PE20040897A1 (en)
PL (2) PL403104A1 (en)
PT (1) PT1532149E (en)
RS (2) RS52142B (en)
SA (1) SA03240448B1 (en)
SI (1) SI1532149T1 (en)
TW (3) TWI319320B (en)
UA (1) UA84275C2 (en)
UY (1) UY27946A1 (en)
WO (1) WO2004018468A2 (en)

Families Citing this family (174)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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