AR077642A1 - Modulators of metabolism and treatment of disorders related thereto - Google Patents

Modulators of metabolism and treatment of disorders related thereto

Info

Publication number
AR077642A1
AR077642A1 ARP100102446A AR077642A1 AR 077642 A1 AR077642 A1 AR 077642A1 AR P100102446 A ARP100102446 A AR P100102446A AR 077642 A1 AR077642 A1 AR 077642A1
Authority
AR
Argentina
Prior art keywords
treatment
metabolism
modulators
disorders related
disorders
Prior art date
Application number
Other languages
Spanish (es)
Original Assignee
Arena Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to US27050209P priority Critical
Application filed by Arena Pharm Inc filed Critical Arena Pharm Inc
Publication of AR077642A1 publication Critical patent/AR077642A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

Abstract

Composicion farmacéutica de N-(2-fluoro-4-(metilsulfonil)fenil)-5-metil-6-(1-(5-metilpirazin-2-il)piperidin-4-iloxi)pirimidin-4-amina, utiles en el tratamiento de trastornos relacionados con GPR119, tales como trastornos relacionados con el metabolismo y complicaciones de los mismos, tales como la diabetes y la obesidad. pharmaceutical composition of N- (2-fluoro-4- (methylsulfonyl) phenyl) -5-methyl-6- (1- (5methyl-2-yl) piperidin-4-yloxy) pyrimidin-4-amine, useful in the treatment of disorders associated with GPR119, such as related metabolism and complications thereof such as diabetes and obesity disorders. Reivindicacion 1: Un compuesto seleccionado del compuesto de formula (1) y sales, solvatos e hidratos farmacéuticamente aceptables del mismo. CLAIMS 1. A compound selected from compound of formula (1) and salts, solvates and hydrates thereof.
ARP100102446 2009-07-09 2010-07-07 Modulators of metabolism and treatment of disorders related thereto AR077642A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
US27050209P true 2009-07-09 2009-07-09

Publications (1)

Publication Number Publication Date
AR077642A1 true AR077642A1 (en) 2011-09-14

Family

ID=42751753

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP100102446 AR077642A1 (en) 2009-07-09 2010-07-07 Modulators of metabolism and treatment of disorders related thereto

Country Status (3)

Country Link
AR (1) AR077642A1 (en)
TW (1) TW201105327A (en)
WO (1) WO2011005929A1 (en)

Families Citing this family (7)

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AU2013290100A1 (en) 2012-07-11 2015-01-29 Elcelyx Therapeutics, Inc. Compositions comprising statins, biguanides and further agents for reducing cardiometabolic risk
US20130310396A1 (en) * 2011-01-19 2013-11-21 Hongwen Zhu Thiazolidine derivatives and their therapeutic use
JP6463631B2 (en) 2011-06-09 2019-02-06 ライゼン・ファーマシューティカルズ・エスアー Novel compounds as modulators of gpr-119
WO2013187646A1 (en) 2012-06-12 2013-12-19 Chong Kun Dang Pharmaceutical Corp. Piperidine derivatives for gpr119 agonist
US9096641B2 (en) 2013-06-05 2015-08-04 Evestra, Inc. Imidazolyl progesterone antagonists
NZ720304A (en) 2013-11-26 2017-08-25 Chong Kun Dang Pharmaceutical Corp Amide derivatives for gpr119 agonist

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