MY165643A - 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions - Google Patents

8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

Info

Publication number
MY165643A
MY165643A MYPI20083230A MYPI20083230A MY165643A MY 165643 A MY165643 A MY 165643A MY PI20083230 A MYPI20083230 A MY PI20083230A MY PI20083230 A MYPI20083230 A MY PI20083230A MY 165643 A MY165643 A MY 165643A
Authority
MY
Malaysia
Prior art keywords
xanthines
piperidin
amino
preparation
pharmaceutical compositions
Prior art date
Application number
MYPI20083230A
Inventor
Frank Himmelsbach Dr
Matthias Eckhardt Dr
Elke Langkopf Dr
Michael Mark Dr
Roland Maier Dr
Ralf R H Lotz Dr
Mohammad Tadayyon Dr
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31947613&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MY165643(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE10238243A external-priority patent/DE10238243A1/en
Priority claimed from DE10312353A external-priority patent/DE10312353A1/en
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of MY165643A publication Critical patent/MY165643A/en

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    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
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    • A61K9/2013Organic compounds, e.g. phospholipids, fats
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Abstract

THE INVENTION RELATES TO A CLASS OF SOFT OR SEMI-SOFT CPG IMMUNOSTIMULATORY OLIGONUCLEOTIDES THAT ARE USEFUL FOR STIMULATING AN IMMUNE RESPONSE.
MYPI20083230A 2002-08-21 2003-08-19 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions MY165643A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10238243A DE10238243A1 (en) 2002-08-21 2002-08-21 New 8-(3-amino-piperidin-1-yl)-xanthine derivatives are dipeptidylpeptidase-IV inhibitors useful for, e.g. treating diabetes mellitus, arthritis or obesity
DE10312353A DE10312353A1 (en) 2003-03-20 2003-03-20 New 8-(3-amino-piperidin-1-yl)-xanthine derivatives are dipeptidylpeptidase-IV inhibitors useful for, e.g. treating diabetes mellitus, arthritis or obesity

Publications (1)

Publication Number Publication Date
MY165643A true MY165643A (en) 2018-04-18

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ID=31947613

Family Applications (2)

Application Number Title Priority Date Filing Date
MYPI20083230A MY165643A (en) 2002-08-21 2003-08-19 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
MYPI20033150A MY137619A (en) 2002-08-21 2003-08-19 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

Family Applications After (1)

Application Number Title Priority Date Filing Date
MYPI20033150A MY137619A (en) 2002-08-21 2003-08-19 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

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EP (6) EP3424926A1 (en)
JP (6) JP4233524B2 (en)
KR (2) KR101150449B1 (en)
CN (4) CN102964347B (en)
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BE (1) BE2011C038I2 (en)
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LT (1) LTC1532149I2 (en)
LU (2) LU91889I2 (en)
ME (1) MEP59708A (en)
MX (1) MXPA05001684A (en)
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NO (4) NO333970B1 (en)
PE (1) PE20040897A1 (en)
PL (2) PL403104A1 (en)
PT (1) PT1532149E (en)
RS (2) RS52142B (en)
SA (1) SA03240448B1 (en)
SI (1) SI1532149T1 (en)
TW (3) TWI469783B (en)
UA (1) UA84275C2 (en)
UY (1) UY27946A1 (en)
WO (1) WO2004018468A2 (en)

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