HK1134077A1 - 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments 8-[3---1-]- - Google Patents

8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments 8-[3---1-]-

Info

Publication number
HK1134077A1
HK1134077A1 HK10100904.3A HK10100904A HK1134077A1 HK 1134077 A1 HK1134077 A1 HK 1134077A1 HK 10100904 A HK10100904 A HK 10100904A HK 1134077 A1 HK1134077 A1 HK 1134077A1
Authority
HK
Hong Kong
Prior art keywords
xanthines
piperidin
medicaments
amino
production
Prior art date
Application number
HK10100904.3A
Other languages
Chinese (zh)
Inventor
弗蘭克‧希梅爾斯巴赫
埃爾克‧蘭格科普夫
馬賽厄斯‧埃克哈特
邁克爾‧馬克
羅蘭‧梅爾
拉爾夫‧
‧洛茨
莫哈邁德‧塔達約恩
Original Assignee
勃林格殷格翰製藥兩合公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31947613&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1134077(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE10238243A external-priority patent/DE10238243A1/en
Priority claimed from DE10312353A external-priority patent/DE10312353A1/en
Application filed by 勃林格殷格翰製藥兩合公司 filed Critical 勃林格殷格翰製藥兩合公司
Publication of HK1134077A1 publication Critical patent/HK1134077A1/en

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    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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HK10100904.3A 2002-08-21 2010-01-28 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments 8-[3---1-]- HK1134077A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10238243A DE10238243A1 (en) 2002-08-21 2002-08-21 New 8-(3-amino-piperidin-1-yl)-xanthine derivatives are dipeptidylpeptidase-IV inhibitors useful for, e.g. treating diabetes mellitus, arthritis or obesity
DE10312353A DE10312353A1 (en) 2003-03-20 2003-03-20 New 8-(3-amino-piperidin-1-yl)-xanthine derivatives are dipeptidylpeptidase-IV inhibitors useful for, e.g. treating diabetes mellitus, arthritis or obesity

Publications (1)

Publication Number Publication Date
HK1134077A1 true HK1134077A1 (en) 2010-04-16

Family

ID=31947613

Family Applications (6)

Application Number Title Priority Date Filing Date
HK06101985.9A HK1081552A1 (en) 2002-08-21 2006-02-16 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments
HK10100903.4A HK1134076A1 (en) 2002-08-21 2010-01-28
HK10100904.3A HK1134077A1 (en) 2002-08-21 2010-01-28 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments 8-[3---1-]-
HK13110418.8A HK1183028A1 (en) 2002-08-21 2013-09-09 Compound of 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments 8-[3---1-]-
HK16103474.1A HK1215439A1 (en) 2002-08-21 2016-03-24 Compound of 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments 8-[3---1-]-
HK18109982.1A HK1250708A1 (en) 2002-08-21 2018-08-02 Compound of 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments

Family Applications Before (2)

Application Number Title Priority Date Filing Date
HK06101985.9A HK1081552A1 (en) 2002-08-21 2006-02-16 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments
HK10100903.4A HK1134076A1 (en) 2002-08-21 2010-01-28

Family Applications After (3)

Application Number Title Priority Date Filing Date
HK13110418.8A HK1183028A1 (en) 2002-08-21 2013-09-09 Compound of 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments 8-[3---1-]-
HK16103474.1A HK1215439A1 (en) 2002-08-21 2016-03-24 Compound of 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments 8-[3---1-]-
HK18109982.1A HK1250708A1 (en) 2002-08-21 2018-08-02 Compound of 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments

Country Status (38)

Country Link
EP (6) EP3424926A1 (en)
JP (6) JP4233524B2 (en)
KR (2) KR101150449B1 (en)
CN (4) CN105001222B (en)
AR (3) AR041025A1 (en)
AT (1) ATE453644T1 (en)
AU (2) AU2003253418B2 (en)
BE (1) BE2011C038I2 (en)
BR (2) BR122012026540B8 (en)
CA (1) CA2496249C (en)
CY (3) CY1109928T1 (en)
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