RS52142B - 8-[3-amino-piperidin-1-il]-ksantini, njihovo dobijanje i njihova primena kao farmaceutskih kompozicija - Google Patents

8-[3-amino-piperidin-1-il]-ksantini, njihovo dobijanje i njihova primena kao farmaceutskih kompozicija

Info

Publication number
RS52142B
RS52142B YU20050137A YUP13705A RS52142B RS 52142 B RS52142 B RS 52142B YU 20050137 A YU20050137 A YU 20050137A YU P13705 A YUP13705 A YU P13705A RS 52142 B RS52142 B RS 52142B
Authority
RS
Serbia
Prior art keywords
group
methyl
xanthines
piperidin
medicaments
Prior art date
Application number
YU20050137A
Other languages
English (en)
Inventor
Elke Langkopf
Matthias Eckhardt
Mohammad Tadayyon
Michael Mark
Roland Maier
Ralf Richard Hermann Lotz
Frank Himmelsbach
Original Assignee
Boehringer Ingelheim Pharma Gmbh & Co. Kg.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31947613&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RS52142(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE10238243A external-priority patent/DE10238243A1/de
Priority claimed from DE10312353A external-priority patent/DE10312353A1/de
Application filed by Boehringer Ingelheim Pharma Gmbh & Co. Kg. filed Critical Boehringer Ingelheim Pharma Gmbh & Co. Kg.
Publication of RS20050137A publication Critical patent/RS20050137A/sr
Publication of RS52142B publication Critical patent/RS52142B/sr

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    • C—CHEMISTRY; METALLURGY
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    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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Abstract

Jedinjenja opšte formulepri čemuR1 označava 4-metoksi-1-naftilmetil grupu, 2-hinolinilmetil, 4-hinolinilmetil ili 6-hinolinilmetil grupu, 1-izohinolinilmetil, 3-metil-1-izohinolinilmetil, 4-metil-1-izohinolinilmetil ili 3-izohinolinilmetil grupu ili2-hinazolinilmetil, 4-metil-2-hinazolinilmetil ili 4-hinazolinilmetil grupu,R2 označava metil grupu iR3 označava 2-buten-1-il ili 2-butin-1-il grupu,njihovi tautomeri, enantiomeri, dijastereomeri, njihove smeše i njihove soli.Prijava sadrži još 19 patentnih zahteva.
YU20050137A 2002-08-21 2003-08-18 8-[3-amino-piperidin-1-il]-ksantini, njihovo dobijanje i njihova primena kao farmaceutskih kompozicija RS52142B (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10238243A DE10238243A1 (de) 2002-08-21 2002-08-21 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
DE10312353A DE10312353A1 (de) 2003-03-20 2003-03-20 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
PCT/EP2003/009127 WO2004018468A2 (de) 2002-08-21 2003-08-18 8-[3-amino-piperidin-1-yl]-xanthine, deren herstellung und deren verwendung als arzneimittel

Publications (2)

Publication Number Publication Date
RS20050137A RS20050137A (en) 2007-11-15
RS52142B true RS52142B (sr) 2012-08-31

Family

ID=31947613

Family Applications (2)

Application Number Title Priority Date Filing Date
YU20050137A RS52142B (sr) 2002-08-21 2003-08-18 8-[3-amino-piperidin-1-il]-ksantini, njihovo dobijanje i njihova primena kao farmaceutskih kompozicija
RS20120139 RS20120139A3 (en) 2002-08-21 2003-08-18 8- [3-AMINO-PYRIDIN-1-IL] -XANTINE, THEIR PREPARATION AND THEIR APPLICATION AS PHARMACEUTICAL COMPOSITIONS

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