RU2011138835A - Применение производного рапамицина - Google Patents

Применение производного рапамицина Download PDF

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RU2011138835A
RU2011138835A RU2011138835/15A RU2011138835A RU2011138835A RU 2011138835 A RU2011138835 A RU 2011138835A RU 2011138835/15 A RU2011138835/15 A RU 2011138835/15A RU 2011138835 A RU2011138835 A RU 2011138835A RU 2011138835 A RU2011138835 A RU 2011138835A
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Russia
Prior art keywords
ramapicin
derivative
application
rapamycin
hydroxyethyl
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RU2011138835/15A
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English (en)
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RU2483727C1 (ru
Inventor
Хейди ЛАНЕ
Теренс О'РЕЙЛЛИ
Джинетта Марджори ВУД
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Новартис Аг
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Priority claimed from GB0104072A external-priority patent/GB0104072D0/en
Priority claimed from GB0124957A external-priority patent/GB0124957D0/en
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Publication of RU2011138835A publication Critical patent/RU2011138835A/ru
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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Abstract

1. Применение 40-O-(2-гидроксиэтил)-рапамицина для получения фармацевтической композиции, предназначенной для лечения опухоли поджелудочной железы.2. Применение по п.1, где единичная доза 40-O-(2-гидроксиэтил)-рапамицина, составляющая от 0, 1 до 25 мг, вводится ежедневно.3. Применение по любому из пп.1 или 2, дополнительно включающее один или более фармацевтически приемлемый растворитель или носитель.

Claims (3)

1. Применение 40-O-(2-гидроксиэтил)-рапамицина для получения фармацевтической композиции, предназначенной для лечения опухоли поджелудочной железы.
2. Применение по п.1, где единичная доза 40-O-(2-гидроксиэтил)-рапамицина, составляющая от 0, 1 до 25 мг, вводится ежедневно.
3. Применение по любому из пп.1 или 2, дополнительно включающее один или более фармацевтически приемлемый растворитель или носитель.
RU2011138835/15A 2001-02-19 2011-09-22 Применение производного рапамицина RU2483727C1 (ru)

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