FI113152B - Menetelmä hallitusti vapautuvan oksikodoniformulaation valmistamiseksi - Google Patents
Menetelmä hallitusti vapautuvan oksikodoniformulaation valmistamiseksi Download PDFInfo
- Publication number
- FI113152B FI113152B FI933330A FI933330A FI113152B FI 113152 B FI113152 B FI 113152B FI 933330 A FI933330 A FI 933330A FI 933330 A FI933330 A FI 933330A FI 113152 B FI113152 B FI 113152B
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- Finland
- Prior art keywords
- oxycodone
- hours
- formulation
- mean
- controlled release
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- BRUQQQPBMZOVGD-XFKAJCMBSA-N Oxycodone Chemical compound O=C([C@@H]1O2)CC[C@@]3(O)[C@H]4CC5=CC=C(OC)C2=C5[C@@]13CCN4C BRUQQQPBMZOVGD-XFKAJCMBSA-N 0.000 title claims abstract description 115
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5015—Organic compounds, e.g. fats, sugars
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Emergency Medicine (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
- Measuring Fluid Pressure (AREA)
- Polyethers (AREA)
- Saccharide Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Plant Substances (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Polysaccharides And Polysaccharide Derivatives (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/800,549 US5266331A (en) | 1991-11-27 | 1991-11-27 | Controlled release oxycodone compositions |
| US80054991 | 1991-11-27 | ||
| US9210146 | 1992-11-25 | ||
| PCT/US1992/010146 WO1993010765A1 (en) | 1991-11-27 | 1992-11-25 | Controlled release oxycodone compositions |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI933330A0 FI933330A0 (fi) | 1993-07-23 |
| FI933330A FI933330A (fi) | 1993-07-23 |
| FI113152B true FI113152B (fi) | 2004-03-15 |
Family
ID=25178688
Family Applications (5)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI933330A FI113152B (fi) | 1991-11-27 | 1993-07-23 | Menetelmä hallitusti vapautuvan oksikodoniformulaation valmistamiseksi |
| FI20031891A FI118252B (fi) | 1991-11-27 | 2003-12-22 | Menetelmä hallitusti vapautuvan formulaation valmistamiseksi |
| FI20031890A FI118251B (fi) | 1991-11-27 | 2003-12-22 | Menetelmä hallitusti vapautuvan, selluloosaeetteriä sisältävän oksikodonisuolaformulaation valmistamiseksi |
| FI20031889A FI116658B (fi) | 1991-11-27 | 2003-12-22 | Menetelmä hallitusti vapautuvan formulaation valmistamiseksi |
| FI20031888A FI118250B (fi) | 1991-11-27 | 2003-12-22 | Menetelmä hallitusti vapautuvan oksikodoniannosmuodon valmistamiseksi |
Family Applications After (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI20031891A FI118252B (fi) | 1991-11-27 | 2003-12-22 | Menetelmä hallitusti vapautuvan formulaation valmistamiseksi |
| FI20031890A FI118251B (fi) | 1991-11-27 | 2003-12-22 | Menetelmä hallitusti vapautuvan, selluloosaeetteriä sisältävän oksikodonisuolaformulaation valmistamiseksi |
| FI20031889A FI116658B (fi) | 1991-11-27 | 2003-12-22 | Menetelmä hallitusti vapautuvan formulaation valmistamiseksi |
| FI20031888A FI118250B (fi) | 1991-11-27 | 2003-12-22 | Menetelmä hallitusti vapautuvan oksikodoniannosmuodon valmistamiseksi |
Country Status (31)
| Country | Link |
|---|---|
| US (13) | US5266331A (no) |
| EP (15) | EP1327446B2 (no) |
| JP (2) | JP3375960B2 (no) |
| KR (1) | KR100280973B1 (no) |
| CN (2) | CN1165307C (no) |
| AT (9) | ATE226822T1 (no) |
| AU (1) | AU657027B2 (no) |
| BG (1) | BG61753B1 (no) |
| BR (1) | BR9205498A (no) |
| CA (1) | CA2098738C (no) |
| CZ (4) | CZ286913B6 (no) |
| DE (10) | DE69214802T2 (no) |
| DK (10) | DK1438959T3 (no) |
| ES (9) | ES2096781T3 (no) |
| FI (5) | FI113152B (no) |
| GR (1) | GR3022273T3 (no) |
| HK (6) | HK1059209A1 (no) |
| HU (10) | HU227815B1 (no) |
| IL (1) | IL103909A (no) |
| MX (1) | MX9302968A (no) |
| NO (6) | NO307028B3 (no) |
| PH (1) | PH31679A (no) |
| PL (2) | PL173574B1 (no) |
| PT (8) | PT1327446E (no) |
| RO (1) | RO115112B1 (no) |
| RS (3) | RS50056B (no) |
| RU (1) | RU2122411C1 (no) |
| SK (1) | SK280295B6 (no) |
| WO (1) | WO1993010765A1 (no) |
| YU (1) | YU49495B (no) |
| ZA (1) | ZA929227B (no) |
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1992
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- 1992-11-25 EP EP03006022A patent/EP1327446B2/en not_active Expired - Lifetime
- 1992-11-25 US US08/081,302 patent/US5549912A/en not_active Expired - Lifetime
- 1992-11-25 DE DE69214802T patent/DE69214802T2/de not_active Expired - Lifetime
- 1992-11-25 DK DK04005576T patent/DK1438959T3/da active
- 1992-11-25 CZ CZ19931764A patent/CZ286913B6/cs not_active IP Right Cessation
- 1992-11-25 EP EP10165398A patent/EP2243484A3/en not_active Withdrawn
- 1992-11-25 RU RU93051780A patent/RU2122411C1/ru active
- 1992-11-25 ES ES92925406T patent/ES2096781T3/es not_active Expired - Lifetime
- 1992-11-25 EP EP02008249A patent/EP1258246B1/en not_active Expired - Lifetime
- 1992-11-25 AT AT96102992T patent/ATE226822T1/de active
- 1992-11-25 AU AU31476/93A patent/AU657027B2/en not_active Expired
- 1992-11-25 DE DE69233699T patent/DE69233699T2/de not_active Expired - Lifetime
- 1992-11-25 KR KR1019930702201A patent/KR100280973B1/ko not_active IP Right Cessation
- 1992-11-25 PT PT02008249T patent/PT1258246E/pt unknown
- 1992-11-25 PT PT07100188T patent/PT1810679E/pt unknown
- 1992-11-25 ES ES02008249T patent/ES2213720T3/es not_active Expired - Lifetime
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- 1992-11-25 CZ CS20041129A patent/CZ300183B6/cs not_active IP Right Cessation
- 1992-11-25 EP EP04005576A patent/EP1438959B1/en not_active Expired - Lifetime
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- 1992-11-25 DE DE69233691T patent/DE69233691T2/de not_active Expired - Lifetime
- 1992-11-25 DE DE69232837.8T patent/DE69232837T3/de not_active Expired - Lifetime
- 1992-11-25 PT PT03006020T patent/PT1325746E/pt unknown
- 1992-11-25 PT PT04026291T patent/PT1502592E/pt unknown
- 1992-11-25 EP EP03006020A patent/EP1325746B1/en not_active Expired - Lifetime
- 1992-11-25 EP EP09164377A patent/EP2106797A3/en not_active Withdrawn
- 1992-11-25 DK DK04026291T patent/DK1502592T3/da active
- 1992-11-25 EP EP07100188A patent/EP1810679B1/en not_active Revoked
- 1992-11-25 AT AT92925406T patent/ATE144418T1/de active
- 1992-11-25 AT AT04005576T patent/ATE360421T1/de active
- 1992-11-25 CZ CS20032327A patent/CZ298499B6/cs not_active IP Right Cessation
- 1992-11-25 RO RO93-00878A patent/RO115112B1/ro unknown
- 1992-11-25 HU HU0401532A patent/HU227815B1/hu unknown
- 1992-11-25 DK DK07100188.7T patent/DK1810679T3/da active
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