ES2222514T3 - Conjugados de dha y agentes farmaceuticos. - Google Patents

Conjugados de dha y agentes farmaceuticos.

Info

Publication number
ES2222514T3
ES2222514T3 ES97926723T ES97926723T ES2222514T3 ES 2222514 T3 ES2222514 T3 ES 2222514T3 ES 97926723 T ES97926723 T ES 97926723T ES 97926723 T ES97926723 T ES 97926723T ES 2222514 T3 ES2222514 T3 ES 2222514T3
Authority
ES
Spain
Prior art keywords
taxol
conjugate
conjugates
dha
tissue
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES97926723T
Other languages
English (en)
Spanish (es)
Inventor
Matthews O. Bradley
Victor E. Shashoua
Nigel L. Webb
Charles S. Swindell
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
American Regent Inc
Original Assignee
Luitpold Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Luitpold Pharmaceuticals Inc filed Critical Luitpold Pharmaceuticals Inc
Application granted granted Critical
Publication of ES2222514T3 publication Critical patent/ES2222514T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/542—Carboxylic acids, e.g. a fatty acid or an amino acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Epoxy Compounds (AREA)
  • Medicinal Preparation (AREA)
ES97926723T 1996-05-22 1997-05-22 Conjugados de dha y agentes farmaceuticos. Expired - Lifetime ES2222514T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US651312 1996-05-22
US08/651,312 US5795909A (en) 1996-05-22 1996-05-22 DHA-pharmaceutical agent conjugates of taxanes

Publications (1)

Publication Number Publication Date
ES2222514T3 true ES2222514T3 (es) 2005-02-01

Family

ID=24612392

Family Applications (1)

Application Number Title Priority Date Filing Date
ES97926723T Expired - Lifetime ES2222514T3 (es) 1996-05-22 1997-05-22 Conjugados de dha y agentes farmaceuticos.

Country Status (10)

Country Link
US (3) US5795909A (enExample)
EP (2) EP0909183B1 (enExample)
JP (1) JP4402173B2 (enExample)
AT (1) ATE273025T1 (enExample)
AU (1) AU725759B2 (enExample)
CA (1) CA2255614C (enExample)
DE (1) DE69730217T2 (enExample)
DK (1) DK0909183T3 (enExample)
ES (1) ES2222514T3 (enExample)
WO (1) WO1997044063A2 (enExample)

Families Citing this family (257)

* Cited by examiner, † Cited by third party
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US5795909A (en) 1998-08-18
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WO1997044063A2 (en) 1997-11-27
US6602902B2 (en) 2003-08-05
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