EE05190B1 - Dispergeeruvad fosfolipiididega stabiliseeritud mikroosakesed - Google Patents

Dispergeeruvad fosfolipiididega stabiliseeritud mikroosakesed

Info

Publication number
EE05190B1
EE05190B1 EEP200100269A EEP200100269A EE05190B1 EE 05190 B1 EE05190 B1 EE 05190B1 EE P200100269 A EEP200100269 A EE P200100269A EE P200100269 A EEP200100269 A EE P200100269A EE 05190 B1 EE05190 B1 EE 05190B1
Authority
EE
Estonia
Prior art keywords
phospholipids
microparticles stabilized
dispersible microparticles
dispersible
stabilized
Prior art date
Application number
EEP200100269A
Other languages
English (en)
Estonian (et)
Inventor
Parikh Indu
K. Mishra Awadhesh
Donga Robert
G. Vachon Michael
Original Assignee
Rtp Pharma Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rtp Pharma Inc. filed Critical Rtp Pharma Inc.
Publication of EE200100269A publication Critical patent/EE200100269A/xx
Publication of EE05190B1 publication Critical patent/EE05190B1/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
EEP200100269A 1998-11-20 1999-11-19 Dispergeeruvad fosfolipiididega stabiliseeritud mikroosakesed EE05190B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10920298P 1998-11-20 1998-11-20
PCT/US1999/027436 WO2000030616A1 (en) 1998-11-20 1999-11-19 Dispersible phospholipid stabilized microparticles

Publications (2)

Publication Number Publication Date
EE200100269A EE200100269A (et) 2002-08-15
EE05190B1 true EE05190B1 (et) 2009-08-17

Family

ID=22326353

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200100269A EE05190B1 (et) 1998-11-20 1999-11-19 Dispergeeruvad fosfolipiididega stabiliseeritud mikroosakesed

Country Status (24)

Country Link
US (3) US7939105B2 (no)
EP (1) EP1133281A1 (no)
JP (2) JP4809533B2 (no)
KR (1) KR20010073232A (no)
CN (1) CN1287769C (no)
AU (1) AU767154B2 (no)
BG (1) BG65254B1 (no)
BR (1) BR9915738A (no)
CA (1) CA2349203C (no)
CZ (1) CZ20011739A3 (no)
EE (1) EE05190B1 (no)
HK (1) HK1042856B (no)
HU (1) HUP0105089A3 (no)
ID (1) ID29270A (no)
IL (2) IL143197A0 (no)
IS (1) IS5945A (no)
NO (1) NO331819B1 (no)
NZ (1) NZ511792A (no)
PL (1) PL201578B1 (no)
RU (1) RU2233654C2 (no)
SK (1) SK288117B6 (no)
UA (1) UA80652C2 (no)
WO (1) WO2000030616A1 (no)
ZA (1) ZA200104069B (no)

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NO20012467D0 (no) 2001-05-18
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CA2349203A1 (en) 2000-06-02
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ID29270A (id) 2001-08-16
BG105573A (en) 2002-01-31
EE200100269A (et) 2002-08-15
HK1042856A1 (en) 2002-08-30
JP2002530321A (ja) 2002-09-17
JP4809533B2 (ja) 2011-11-09
KR20010073232A (ko) 2001-07-31
US20020106403A1 (en) 2002-08-08
NZ511792A (en) 2003-08-29
US7939106B2 (en) 2011-05-10
CN1287769C (zh) 2006-12-06
PL201578B1 (pl) 2009-04-30
HUP0105089A3 (en) 2002-09-30
HK1042856B (zh) 2007-07-27
NO20012467L (no) 2001-07-18
JP2011137031A (ja) 2011-07-14
SK6852001A3 (en) 2001-12-03
NO331819B1 (no) 2012-04-10
IL143197A0 (en) 2002-04-21
AU1737500A (en) 2000-06-13
AU767154B2 (en) 2003-10-30
US20110244032A1 (en) 2011-10-06
IS5945A (is) 2001-05-18
CA2349203C (en) 2013-05-21
RU2233654C2 (ru) 2004-08-10
HUP0105089A2 (hu) 2002-05-29
US7939105B2 (en) 2011-05-10
WO2000030616A1 (en) 2000-06-02
BR9915738A (pt) 2001-10-02
UA80652C2 (uk) 2007-10-10
IL143197A (en) 2009-09-01
SK288117B6 (sk) 2013-09-03
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US20030206949A1 (en) 2003-11-06

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