DK1088555T3 - Præparat med vedholdende frigivelse - Google Patents

Præparat med vedholdende frigivelse

Info

Publication number
DK1088555T3
DK1088555T3 DK00203850T DK00203850T DK1088555T3 DK 1088555 T3 DK1088555 T3 DK 1088555T3 DK 00203850 T DK00203850 T DK 00203850T DK 00203850 T DK00203850 T DK 00203850T DK 1088555 T3 DK1088555 T3 DK 1088555T3
Authority
DK
Denmark
Prior art keywords
group
formula
release preparation
sustained
amino
Prior art date
Application number
DK00203850T
Other languages
Danish (da)
English (en)
Inventor
Yasuaki Ogawa
Shigeru Kamei
Yasutaka Igari
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Application granted granted Critical
Publication of DK1088555T3 publication Critical patent/DK1088555T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08—Peptides having 5 to 11 amino acids
    • A61K38/09—Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
DK00203850T 1992-12-07 1993-12-03 Præparat med vedholdende frigivelse DK1088555T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP32707092 1992-12-07
JP1897893 1993-02-05
JP14513493 1993-06-16
EP93309681A EP0601799B1 (fr) 1992-12-07 1993-12-03 Préparation du type à libération prolongée

Publications (1)

Publication Number Publication Date
DK1088555T3 true DK1088555T3 (da) 2005-07-04

Family

ID=27282444

Family Applications (2)

Application Number Title Priority Date Filing Date
DK93309681T DK0601799T3 (da) 1992-12-07 1993-12-03 Præparat med langvarig frigivelse
DK00203850T DK1088555T3 (da) 1992-12-07 1993-12-03 Præparat med vedholdende frigivelse

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK93309681T DK0601799T3 (da) 1992-12-07 1993-12-03 Præparat med langvarig frigivelse

Country Status (24)

Country Link
US (7) US5480868A (fr)
EP (2) EP0601799B1 (fr)
JP (1) JP3725906B2 (fr)
KR (2) KR100305951B1 (fr)
CN (2) CN1099893C (fr)
AT (2) ATE203910T1 (fr)
AU (1) AU669939B2 (fr)
CA (1) CA2110730C (fr)
DE (2) DE69333817T2 (fr)
DK (2) DK0601799T3 (fr)
EE (1) EE03117B1 (fr)
ES (2) ES2158856T3 (fr)
FI (2) FI935471A (fr)
GE (1) GEP19991600B (fr)
GR (1) GR3037085T3 (fr)
HK (1) HK1037519A1 (fr)
LV (1) LV10927B (fr)
MX (1) MX9307686A (fr)
NO (1) NO310704B1 (fr)
NZ (1) NZ250349A (fr)
PT (2) PT1088555E (fr)
SG (1) SG46283A1 (fr)
TW (1) TW333456B (fr)
WO (1) WO1994013317A1 (fr)

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EP0601799A1 (fr) 1994-06-15
US5480868A (en) 1996-01-02
DK0601799T3 (da) 2001-10-01
US20030039698A1 (en) 2003-02-27
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