HK1037519A1 - Sustained-release leuprorelin preparation. - Google Patents

Sustained-release leuprorelin preparation.

Info

Publication number
HK1037519A1
HK1037519A1 HK01106799A HK01106799A HK1037519A1 HK 1037519 A1 HK1037519 A1 HK 1037519A1 HK 01106799 A HK01106799 A HK 01106799A HK 01106799 A HK01106799 A HK 01106799A HK 1037519 A1 HK1037519 A1 HK 1037519A1
Authority
HK
Hong Kong
Prior art keywords
group
sustained
formula
release
amino
Prior art date
Application number
HK01106799A
Other languages
English (en)
Inventor
Shigeru Kamei
Yasutaka Igari
Yasuaki Ogawa
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of HK1037519A1 publication Critical patent/HK1037519A1/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08—Peptides having 5 to 11 amino acids
    • A61K38/09—Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
HK01106799A 1992-12-07 2001-09-26 Sustained-release leuprorelin preparation. HK1037519A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP32707092 1992-12-07
JP1897893 1993-02-05
JP14513493 1993-06-16

Publications (1)

Publication Number Publication Date
HK1037519A1 true HK1037519A1 (en) 2002-02-15

Family

ID=27282444

Family Applications (1)

Application Number Title Priority Date Filing Date
HK01106799A HK1037519A1 (en) 1992-12-07 2001-09-26 Sustained-release leuprorelin preparation.

Country Status (24)

Country Link
US (7) US5480868A (xx)
EP (2) EP0601799B1 (xx)
JP (1) JP3725906B2 (xx)
KR (2) KR100305951B1 (xx)
CN (2) CN1099893C (xx)
AT (2) ATE295733T1 (xx)
AU (1) AU669939B2 (xx)
CA (1) CA2110730C (xx)
DE (2) DE69333817T2 (xx)
DK (2) DK0601799T3 (xx)
EE (1) EE03117B1 (xx)
ES (2) ES2158856T3 (xx)
FI (2) FI935471A (xx)
GE (1) GEP19991600B (xx)
GR (1) GR3037085T3 (xx)
HK (1) HK1037519A1 (xx)
LV (1) LV10927B (xx)
MX (1) MX9307686A (xx)
NO (1) NO310704B1 (xx)
NZ (1) NZ250349A (xx)
PT (2) PT601799E (xx)
SG (1) SG46283A1 (xx)
TW (1) TW333456B (xx)
WO (1) WO1994013317A1 (xx)

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US20020173467A1 (en) 2002-11-21
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EP1088555B1 (en) 2005-05-18
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CA2110730C (en) 2008-09-16
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