CA2905409C - Stabilized modified release vitamin d formulation and method of administering same - Google Patents

Stabilized modified release vitamin d formulation and method of administering same Download PDF

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Publication number
CA2905409C
CA2905409C CA2905409A CA2905409A CA2905409C CA 2905409 C CA2905409 C CA 2905409C CA 2905409 A CA2905409 A CA 2905409A CA 2905409 A CA2905409 A CA 2905409A CA 2905409 C CA2905409 C CA 2905409C
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CA
Canada
Prior art keywords
formulation
hydroxyvitamin
vitamin
compound
dosage form
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Application number
CA2905409A
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English (en)
French (fr)
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CA2905409A1 (en
Inventor
Jay A. White
Joel Z. Melnick
Sammy A. Agudoawu
Samir P. Tabash
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eirgen Pharma Ltd
Original Assignee
Opko Ireland Global Holdings Ltd
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Application filed by Opko Ireland Global Holdings Ltd filed Critical Opko Ireland Global Holdings Ltd
Publication of CA2905409A1 publication Critical patent/CA2905409A1/en
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds
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    • A61K31/59—Compounds containing 9, 10- seco- cyclopenta[a]hydrophenanthrene ring systems
    • A61K31/593—9,10-Secocholestane derivatives, e.g. cholecalciferol, i.e. vitamin D3
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    • A61K31/592—9,10-Secoergostane derivatives, e.g. ergocalciferol, i.e. vitamin D2
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
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CA2905409A 2013-03-15 2014-03-14 Stabilized modified release vitamin d formulation and method of administering same Active CA2905409C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361801896P 2013-03-15 2013-03-15
US61/801,896 2013-03-15
PCT/US2014/028132 WO2014143941A1 (en) 2013-03-15 2014-03-14 Stabilized modified release vitamin d formulation and method of administring same

Publications (2)

Publication Number Publication Date
CA2905409A1 CA2905409A1 (en) 2014-09-18
CA2905409C true CA2905409C (en) 2023-01-03

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CA2905409A Active CA2905409C (en) 2013-03-15 2014-03-14 Stabilized modified release vitamin d formulation and method of administering same

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US (7) US9861644B2 (https=)
EP (4) EP3332773B8 (https=)
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HRP20201284T1 (hr) 2020-12-11
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CY1123167T1 (el) 2021-10-29
HK1220362A1 (zh) 2017-05-05
KR20140140004A (ko) 2014-12-08
KR20190095216A (ko) 2019-08-14
US11253528B2 (en) 2022-02-22
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US20260034148A1 (en) 2026-02-05
CN105246464A (zh) 2016-01-13
JP7282832B2 (ja) 2023-05-29
BR112015023658A2 (pt) 2017-07-18
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SI2968172T1 (sl) 2020-12-31
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DE202014011525U1 (de) 2021-11-11
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PL3650016T3 (pl) 2021-12-27
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US20180271884A1 (en) 2018-09-27
LT3332773T (lt) 2020-12-10
MY194092A (en) 2022-11-11
KR20140113374A (ko) 2014-09-24
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DK2968172T3 (da) 2020-09-14
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US10350224B2 (en) 2019-07-16

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