BR112019019101A2 - compostos macrocíclicos como inibidores de ros1 cinase - Google Patents
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762472185P | 2017-03-16 | 2017-03-16 | |
| PCT/US2018/022833 WO2018170381A1 (en) | 2017-03-16 | 2018-03-16 | Macrocyclic compounds as ros1 kinase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR112019019101A2 true BR112019019101A2 (pt) | 2020-04-22 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112019019101A BR112019019101A2 (pt) | 2017-03-16 | 2018-03-16 | compostos macrocíclicos como inibidores de ros1 cinase |
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| US (3) | US20190076436A1 (OSRAM) |
| EP (1) | EP3595651A1 (OSRAM) |
| JP (1) | JP2020514356A (OSRAM) |
| KR (1) | KR20190126003A (OSRAM) |
| CN (1) | CN110769820A (OSRAM) |
| AU (1) | AU2018234726A1 (OSRAM) |
| BR (1) | BR112019019101A2 (OSRAM) |
| CA (1) | CA3056754A1 (OSRAM) |
| CL (1) | CL2019002612A1 (OSRAM) |
| IL (1) | IL269216A (OSRAM) |
| JO (1) | JOP20190213A1 (OSRAM) |
| MA (1) | MA49888A (OSRAM) |
| MX (1) | MX2019010988A (OSRAM) |
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| CN109475545A (zh) | 2016-04-19 | 2019-03-15 | 埃克塞里艾克西斯公司 | 三阴性乳腺癌治疗方法 |
| CN109790143A (zh) | 2016-05-10 | 2019-05-21 | C4医药公司 | 用于靶蛋白降解的胺连接的c3-戊二酰亚胺降解决定子体 |
| SI3458456T1 (sl) | 2016-05-18 | 2021-04-30 | Loxo Oncology, Inc. | Priprava (S)-N-(5-((R)-2-(2,5-difluorofenil) pirolidin-1-il) pirazolo (1,5-A) pirimidin-3-il)-3-hidroksipirolidin-1-karboksamida |
| WO2017201156A1 (en) | 2016-05-18 | 2017-11-23 | Duke University | Method of treating kras wild-type metastatic colorectal cell carcinoma using cabozantinib plus panitumumab |
| JP2019519540A (ja) | 2016-06-01 | 2019-07-11 | エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft | 肺癌患者におけるalk阻害薬療法に対する応答を予測する未分化リンパ腫キナーゼにおける新規な変異 |
| US10227329B2 (en) | 2016-07-22 | 2019-03-12 | Blueprint Medicines Corporation | Compounds useful for treating disorders related to RET |
| TWI704148B (zh) | 2016-10-10 | 2020-09-11 | 美商亞雷生物製藥股份有限公司 | 作為ret激酶抑制劑之經取代吡唑并[1,5-a]吡啶化合物 |
| JOP20190092A1 (ar) | 2016-10-26 | 2019-04-25 | Array Biopharma Inc | عملية لتحضير مركبات بيرازولو[1، 5-a]بيريميدين وأملاح منها |
| CA3049452A1 (en) | 2017-01-20 | 2018-07-26 | Gisela Schwab | Combinations of cabozantinib and atezolizumab to treat cancer |
| CN108456163A (zh) | 2017-02-20 | 2018-08-28 | 中国科学院上海药物研究所 | 含邻氨基杂芳环炔基的化合物及其制备方法和用途 |
| JOP20190213A1 (ar) | 2017-03-16 | 2019-09-16 | Array Biopharma Inc | مركبات حلقية ضخمة كمثبطات لكيناز ros1 |
| EP3700576A1 (en) | 2017-10-26 | 2020-09-02 | Array Biopharma Inc. | Formulations of a macrocyclic trk kinase inhibitor |
-
2017
- 2017-06-16 JO JOP/2019/0213A patent/JOP20190213A1/ar unknown
-
2018
- 2018-03-16 SG SG11201908532U patent/SG11201908532UA/en unknown
- 2018-03-16 EP EP18716714.3A patent/EP3595651A1/en not_active Withdrawn
- 2018-03-16 TN TNP/2019/000263A patent/TN2019000263A1/en unknown
- 2018-03-16 AU AU2018234726A patent/AU2018234726A1/en not_active Abandoned
- 2018-03-16 MX MX2019010988A patent/MX2019010988A/es unknown
- 2018-03-16 KR KR1020197029924A patent/KR20190126003A/ko not_active Withdrawn
- 2018-03-16 JP JP2019550588A patent/JP2020514356A/ja active Pending
- 2018-03-16 CN CN201880032348.5A patent/CN110769820A/zh active Pending
- 2018-03-16 MA MA049888A patent/MA49888A/fr unknown
- 2018-03-16 CA CA3056754A patent/CA3056754A1/en active Pending
- 2018-03-16 WO PCT/US2018/022833 patent/WO2018170381A1/en not_active Ceased
- 2018-03-16 BR BR112019019101A patent/BR112019019101A2/pt not_active Application Discontinuation
- 2018-03-16 RU RU2019132666A patent/RU2019132666A/ru not_active Application Discontinuation
- 2018-03-16 TW TW107109131A patent/TW201838631A/zh unknown
- 2018-11-26 US US16/199,867 patent/US20190076436A1/en not_active Abandoned
- 2018-11-26 US US16/199,818 patent/US10966985B2/en not_active Expired - Fee Related
- 2018-11-26 US US16/199,875 patent/US10688100B2/en not_active Expired - Fee Related
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2019
- 2019-09-09 IL IL26921619A patent/IL269216A/en unknown
- 2019-09-12 CL CL2019002612A patent/CL2019002612A1/es unknown
- 2019-09-12 PH PH12019502069A patent/PH12019502069A1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| TW201838631A (zh) | 2018-11-01 |
| MA49888A (fr) | 2020-06-24 |
| US20190076436A1 (en) | 2019-03-14 |
| US20190151322A1 (en) | 2019-05-23 |
| SG11201908532UA (en) | 2019-10-30 |
| CN110769820A (zh) | 2020-02-07 |
| AU2018234726A1 (en) | 2019-09-26 |
| CL2019002612A1 (es) | 2020-05-29 |
| JOP20190213A1 (ar) | 2019-09-16 |
| US20190076437A1 (en) | 2019-03-14 |
| PH12019502069A1 (en) | 2020-09-14 |
| TN2019000263A1 (en) | 2021-01-07 |
| JP2020514356A (ja) | 2020-05-21 |
| WO2018170381A1 (en) | 2018-09-20 |
| KR20190126003A (ko) | 2019-11-07 |
| CA3056754A1 (en) | 2018-09-20 |
| US10966985B2 (en) | 2021-04-06 |
| RU2019132666A (ru) | 2021-04-16 |
| US10688100B2 (en) | 2020-06-23 |
| EP3595651A1 (en) | 2020-01-22 |
| MX2019010988A (es) | 2020-02-05 |
| IL269216A (en) | 2019-11-28 |
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