AU777701B2 - Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use - Google Patents

Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use Download PDF

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Publication number
AU777701B2
AU777701B2 AU57852/00A AU5785200A AU777701B2 AU 777701 B2 AU777701 B2 AU 777701B2 AU 57852/00 A AU57852/00 A AU 57852/00A AU 5785200 A AU5785200 A AU 5785200A AU 777701 B2 AU777701 B2 AU 777701B2
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AU
Australia
Prior art keywords
found
calc
indazole
nmr
mmol
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Expired, expires
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AU57852/00A
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English (en)
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AU5785200A (en
Inventor
Steven Lee Bender
Allen J. Borchardt
John F. Braganza
Michael Raymond Collins
Stephan James Cripps
Ye Hua
Michael David Johnson
Theodore Otto Johnson Jr.
Robert Steven Kania
Hiep The Luu
Cynthia Louise Palmer
Siegfried Heinz Reich
Anna Maria Tempczyk-Russell
Min Teng
Christine Thomas
Michael David Varney
Michael Brennan Wallace
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Agouron Pharmaceuticals LLC
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Agouron Pharmaceuticals LLC
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Application filed by Agouron Pharmaceuticals LLC filed Critical Agouron Pharmaceuticals LLC
Publication of AU5785200A publication Critical patent/AU5785200A/en
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Assigned to AGOURON PHARMACEUTICALS, LLC reassignment AGOURON PHARMACEUTICALS, LLC Request to Amend Deed and Register Assignors: AGOURON PHARMACEUTICALS, INC.
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Diabetes (AREA)
  • Ophthalmology & Optometry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU57852/00A 1999-07-02 2000-06-30 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use Expired AU777701B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US14213099P 1999-07-02 1999-07-02
US60/142130 1999-07-02
PCT/US2000/018263 WO2001002369A2 (en) 1999-07-02 2000-06-30 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use

Publications (2)

Publication Number Publication Date
AU5785200A AU5785200A (en) 2001-01-22
AU777701B2 true AU777701B2 (en) 2004-10-28

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EP (2) EP1218348B1 (forum.php)
JP (2) JP3878849B2 (forum.php)
KR (1) KR100529639B1 (forum.php)
CN (2) CN1137884C (forum.php)
AP (1) AP1486A (forum.php)
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AT (1) ATE376543T1 (forum.php)
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HU230000B1 (en) 1999-02-10 2015-04-28 Astrazeneca Ab Intermediates for the preparation of angiogenesis inhibitory quinazoline derivatives
PE20010306A1 (es) * 1999-07-02 2001-03-29 Agouron Pharma Compuestos de indazol y composiciones farmaceuticas que los contienen utiles para la inhibicion de proteina kinasa
KR100755622B1 (ko) 1999-12-24 2007-09-04 아벤티스 파마 리미티드 아자인돌
AU2001229727B2 (en) 2000-02-07 2004-10-14 Bristol-Myers Squibb Co. 3-aminopyrazole inhibitors of cyclin dependent kinases
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EP1278749B1 (en) 2000-04-25 2005-01-26 Bristol-Myers Squibb Company USE OF 5-THIO-, SULFINYL- AND SULFONYLPYRAZOLO 3,4-b]-PYRIDINES AS CYCLIN DEPENDENT KINASE INHIBITORS
BR0113056A (pt) 2000-08-09 2003-07-08 Astrazeneca Ab Composto, processo papa a preparação do mesmo, composição farmacêutica, e, método para produzir um efeito antiangiogênico e/ou redutor da permeabilidade vascular em um animal de sangue quente, e, uso de um composto
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ES2334641T3 (es) 2000-09-01 2010-03-15 Novartis Vaccines And Diagnostics, Inc. Derivados aza heterociclicos y su uso terapeutico.
PL211125B1 (pl) 2000-09-11 2012-04-30 Novartis Vaccines & Diagnostic Pochodne chinolinonu jako inhibitory kinazy tyrozynowej, kompozycje je zawierające i ich zastosowanie
CN101024627A (zh) 2000-10-20 2007-08-29 卫材R&D管理有限公司 含氮芳环衍生物
TWI243164B (en) 2001-02-13 2005-11-11 Aventis Pharma Gmbh Acylated indanyl amines and their use as pharmaceuticals
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