SG11201400666PA - Indazole-3-carboxamides and their use as wnt/b-catenin signaling pathway inhibitors - Google Patents
Indazole-3-carboxamides and their use as wnt/b-catenin signaling pathway inhibitorsInfo
- Publication number
- SG11201400666PA SG11201400666PA SG11201400666PA SG11201400666PA SG11201400666PA SG 11201400666P A SG11201400666P A SG 11201400666PA SG 11201400666P A SG11201400666P A SG 11201400666PA SG 11201400666P A SG11201400666P A SG 11201400666PA SG 11201400666P A SG11201400666P A SG 11201400666PA
- Authority
- SG
- Singapore
- Prior art keywords
- wnt
- carboxamides
- indazole
- signaling pathway
- pathway inhibitors
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C07—ORGANIC CHEMISTRY
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- C07—ORGANIC CHEMISTRY
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Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
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US201161534601P | 2011-09-14 | 2011-09-14 | |
US201261624646P | 2012-04-16 | 2012-04-16 | |
PCT/US2012/055172 WO2013040215A1 (en) | 2011-09-14 | 2012-09-13 | Indazole-3-carboxamides and their use as wnt/b-catenin signaling pathway inhibitors |
Publications (1)
Publication Number | Publication Date |
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SG11201400666PA true SG11201400666PA (en) | 2014-09-26 |
Family
ID=47883736
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG11201400666PA SG11201400666PA (en) | 2011-09-14 | 2012-09-13 | Indazole-3-carboxamides and their use as wnt/b-catenin signaling pathway inhibitors |
SG10202002005SA SG10202002005SA (en) | 2011-09-14 | 2012-09-13 | Indazole-3-carboxamides and their use as wnt/b-catenin signaling pathway inhibitors |
SG10201914121YA SG10201914121YA (en) | 2011-09-14 | 2012-09-13 | Indazole-3-carboxamides and their use as wnt/b-catenin signaling pathway inhibitors |
Family Applications After (2)
Application Number | Title | Priority Date | Filing Date |
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SG10202002005SA SG10202002005SA (en) | 2011-09-14 | 2012-09-13 | Indazole-3-carboxamides and their use as wnt/b-catenin signaling pathway inhibitors |
SG10201914121YA SG10201914121YA (en) | 2011-09-14 | 2012-09-13 | Indazole-3-carboxamides and their use as wnt/b-catenin signaling pathway inhibitors |
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EP (2) | EP3473099A1 (en) |
JP (2) | JP2014526510A (en) |
KR (1) | KR102010611B1 (en) |
CN (2) | CN103929963A (en) |
AU (2) | AU2012308570B2 (en) |
BR (1) | BR112014006127A2 (en) |
CA (1) | CA2848659C (en) |
CL (1) | CL2014000642A1 (en) |
CO (1) | CO6940416A2 (en) |
CY (1) | CY1122795T1 (en) |
DK (1) | DK2755483T3 (en) |
ES (1) | ES2711777T3 (en) |
HR (1) | HRP20190281T1 (en) |
HU (1) | HUE041576T2 (en) |
IL (1) | IL231536A (en) |
IN (1) | IN2014CN02646A (en) |
LT (1) | LT2755483T (en) |
ME (1) | ME03332B (en) |
MX (2) | MX341504B (en) |
MY (1) | MY184882A (en) |
PE (1) | PE20141678A1 (en) |
PL (1) | PL2755483T3 (en) |
PT (1) | PT2755483T (en) |
RS (1) | RS58462B1 (en) |
RU (1) | RU2627693C2 (en) |
SG (3) | SG11201400666PA (en) |
SI (1) | SI2755483T1 (en) |
WO (1) | WO2013040215A1 (en) |
ZA (1) | ZA201402623B (en) |
Families Citing this family (77)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8252812B2 (en) | 2009-08-10 | 2012-08-28 | Samumed, Llc | Indazole inhibitors of the WNT signal pathway and therapeutic uses thereof |
RS56669B1 (en) | 2009-12-21 | 2018-03-30 | Samumed Llc | 1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof |
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