GT200400136A - 3.5-DISPOSED INDAZOL COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS TO INTERVENE IN OR INHIBIT CELLULAR APPROVALIFERATION. - Google Patents

3.5-DISPOSED INDAZOL COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS TO INTERVENE IN OR INHIBIT CELLULAR APPROVALIFERATION.

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Publication number
GT200400136A
GT200400136A GT200400136A GT200400136A GT200400136A GT 200400136 A GT200400136 A GT 200400136A GT 200400136 A GT200400136 A GT 200400136A GT 200400136 A GT200400136 A GT 200400136A GT 200400136 A GT200400136 A GT 200400136A
Authority
GT
Guatemala
Prior art keywords
compounds
intervene
disposed
methods
pharmaceutical compositions
Prior art date
Application number
GT200400136A
Other languages
Spanish (es)
Inventor
Susan Elizabeth Kephart
Indrawan James Mcalpine
Seigfried Heins Reich
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Filing date
Publication date
Application filed filed Critical
Publication of GT200400136A publication Critical patent/GT200400136A/en

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Abstract

SE DESCRIBEN COMPUESTOS DE INDAZOL 3,5DISUSTITUIDOS QUE MODULAN Y/O INHIBEN LA PROLIFERACION CELULAR TAL COMO LA ACTIVIDAD DE LAS PROTEINAS QUINASAS. ESTOS COMPUESTOS Y COMPOSICIONES FARMACEUTICAS QUE LOS CONTIENEN SON CAPACES DE INTERVENIR EN ENFERMEDADES DEPENDIENTES DE LA CDK PARA MODULAR Y/O INHIBIR LA PROLIFERACION CELULARA NO DESEADA. LA INVENCION TAMBIEN SE DIRIGE AL USO TERAPEUTICO O PROFILACTICO DE COMPOSICIONES FARMACEUTICAS QUE CONTIENEN TALES COMPUESTOS Y A METODOS PARA TRATAR EL CANCER ASI COMO OTRAS CONDICIONES PATOLOGICAS ASOCIADAS CON ANGIOGENESIS Y/O PROLIFERACION CELULAR, NO DESEADA, TALES COMO: RETINOPATIA DIABETICA, GLAUCOMA NEOVASCULAR, ARTRITIS REUMATOIDE Y SORIASIS, POR ADMINISTRACION DE CANTIDADES EFICACES DE TALES COMPUESTOS.INDAZOL COMPOUNDS 3.5 DISPOSED THAT MODULATE AND / OR INHIBIT CELLULAR PROLIFERATION SUCH AS THE ACTIVITY OF KINASE PROTEINS. THESE PHARMACEUTICAL COMPOUNDS AND COMPOSITIONS CONTAINING THEM ARE ABLE TO INTERVENE IN DEPENDENT DISEASES OF THE CDK TO MODULATE AND / OR INHIBIT THE UNWANTED CELLULAR PROLIFERATION. THE INVENTION IS ALSO ADDRESSED TO THE THERAPEUTIC OR PROFILACTIC USE OF PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS TO TREAT CANCER AS WELL AS OTHER PATHOLOGICAL CONDITIONS ASSOCIATED WITH ANGIOGENESIS AND / OR PROLIFTIATIMED ROLLAR, DISTRIBUTED CELEBRATION, ASSOCIATED BY NUMBER REUMATOID AND SORIASIS, BY ADMINISTRATION OF EFFECTIVE AMOUNTS OF SUCH COMPOUNDS.

GT200400136A 2003-07-30 2004-07-19 3.5-DISPOSED INDAZOL COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS TO INTERVENE IN OR INHIBIT CELLULAR APPROVALIFERATION. GT200400136A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US49147403P 2003-07-30 2003-07-30

Publications (1)

Publication Number Publication Date
GT200400136A true GT200400136A (en) 2005-05-02

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Family Applications (1)

Application Number Title Priority Date Filing Date
GT200400136A GT200400136A (en) 2003-07-30 2004-07-19 3.5-DISPOSED INDAZOL COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS TO INTERVENE IN OR INHIBIT CELLULAR APPROVALIFERATION.

Country Status (3)

Country Link
CN (1) CN1829713A (en)
GT (1) GT200400136A (en)
ZA (1) ZA200600821B (en)

Families Citing this family (38)

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CN102675286B (en) * 2011-03-07 2015-08-19 中国科学院上海药物研究所 One class indazole compounds and preparation method thereof, purposes and pharmaceutical composition
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WO2017024015A1 (en) 2015-08-03 2017-02-09 Samumed, Llc. 3-(3h-imidazo[4,5-b]pyridin-2-yl)-1h-pyrazolo[4,3-b]pyridines and therapeutic uses thereof
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US10463651B2 (en) 2015-08-03 2019-11-05 Samumed, Llc 3-(1H-pyrrolo[3,2-C]pyridin-2-YL)-1H-indazoles and therapeutic uses thereof
US10519169B2 (en) 2015-08-03 2019-12-31 Samumed, Llc 3-(1H-pyrrolo[2,3-C]pyridin-2-yl)-1 H-pyrazolo[4,3-B]pyridines and therapeutic uses thereof
WO2017024021A1 (en) 2015-08-03 2017-02-09 Samumed, Llc 3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-indazoles and therapeutic uses thereof
WO2017023988A1 (en) 2015-08-03 2017-02-09 Samumed, Llc. 3-(3h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[4,3-b]pyridines and therapeutic uses thereof
US10392383B2 (en) 2015-08-03 2019-08-27 Samumed, Llc 3-(1H-benzo[d]imidazol-2-yl)-1H-pyrazolo[4,3-b]pyridines and therapeutic uses thereof
WO2017023996A1 (en) 2015-08-03 2017-02-09 Samumed, Llc. 3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof
WO2017023984A1 (en) 2015-08-03 2017-02-09 Samumed, Llc. 3-(1h-pyrrolo[3,2-c]pyridin-2-yl)-1h-pyrazolo[3,4-c]pyridines and therapeutic uses thereof
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AU2017345699A1 (en) 2016-10-21 2019-05-16 Samumed, Llc Methods of using indazole-3-carboxamides and their use as Wnt/B-catenin signaling pathway inhibitors
WO2018085865A1 (en) 2016-11-07 2018-05-11 Samumed, Llc Single-dose, ready-to-use injectable formulations

Also Published As

Publication number Publication date
CN1829713A (en) 2006-09-06
ZA200600821B (en) 2007-04-25

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