ATE212993T1 - Pyrolopyrimidine und verfahren zu ihrer herstellung - Google Patents

Pyrolopyrimidine und verfahren zu ihrer herstellung

Info

Publication number
ATE212993T1
ATE212993T1 AT96923893T AT96923893T ATE212993T1 AT E212993 T1 ATE212993 T1 AT E212993T1 AT 96923893 T AT96923893 T AT 96923893T AT 96923893 T AT96923893 T AT 96923893T AT E212993 T1 ATE212993 T1 AT E212993T1
Authority
AT
Austria
Prior art keywords
pct
date jan
sec
pyrolopyrimidines
production
Prior art date
Application number
AT96923893T
Other languages
English (en)
Inventor
Peter Traxler
Guido Bold
Wolfgang Karl-Diether Brill
Joerg Frei
Original Assignee
Novartis Erfind Verwalt Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27508793&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE212993(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Erfind Verwalt Gmbh filed Critical Novartis Erfind Verwalt Gmbh
Application granted granted Critical
Publication of ATE212993T1 publication Critical patent/ATE212993T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
AT96923893T 1995-07-06 1996-06-24 Pyrolopyrimidine und verfahren zu ihrer herstellung ATE212993T1 (de)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
CH197695 1995-07-06
CH249895 1995-09-01
CH319895 1995-11-10
CH25596 1996-02-01
CH122496 1996-05-13
PCT/EP1996/002728 WO1997002266A1 (en) 1995-07-06 1996-06-24 Pyrrolopyrimidines and processes for the preparation thereof

Publications (1)

Publication Number Publication Date
ATE212993T1 true ATE212993T1 (de) 2002-02-15

Family

ID=27508793

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96923893T ATE212993T1 (de) 1995-07-06 1996-06-24 Pyrolopyrimidine und verfahren zu ihrer herstellung

Country Status (25)

Country Link
US (1) US6140332A (de)
EP (1) EP0836605B1 (de)
JP (1) JP4146514B2 (de)
KR (1) KR100437582B1 (de)
CN (1) CN1100778C (de)
AT (1) ATE212993T1 (de)
BR (1) BR9609617B1 (de)
CA (1) CA2224435C (de)
CY (1) CY2365B1 (de)
CZ (1) CZ1598A3 (de)
DE (1) DE69619114T2 (de)
DK (1) DK0836605T3 (de)
EA (1) EA001428B1 (de)
ES (1) ES2172670T3 (de)
HU (1) HUP9900330A3 (de)
IL (1) IL122855A (de)
MX (1) MX9800215A (de)
NO (1) NO310359B1 (de)
NZ (1) NZ312665A (de)
PL (1) PL188959B1 (de)
PT (1) PT836605E (de)
SI (1) SI9620103A (de)
SK (1) SK398A3 (de)
TR (1) TR199800012T1 (de)
WO (1) WO1997002266A1 (de)

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