AP2011005745A0 - Modulators of toll-like receptors. - Google Patents
Modulators of toll-like receptors.Info
- Publication number
- AP2011005745A0 AP2011005745A0 AP2011000745A AP2011000745A AP2011005745A0 AP 2011005745 A0 AP2011005745 A0 AP 2011005745A0 AP 2011000745 A AP2011000745 A AP 2011000745A AP 2011000745 A AP2011000745 A AP 2011000745A AP 2011005745 A0 AP2011005745 A0 AP 2011005745A0
- Authority
- AP
- ARIPO
- Prior art keywords
- toll
- modulators
- receptors
- Prior art date
Links
- 102000002689 Toll-like receptor Human genes 0.000 title 1
- 108020000411 Toll-like receptor Proteins 0.000 title 1
Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/527—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim spiro-condensed
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- A61K31/5375—1,4-Oxazines, e.g. morpholine
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- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
- A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
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- A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
- A61K31/708—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid having oxo groups directly attached to the purine ring system, e.g. guanosine, guanylic acid
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- C07D487/04—Ortho-condensed systems
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- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
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- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
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- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
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- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Molecular Biology (AREA)
- Virology (AREA)
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- Immunology (AREA)
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- Oncology (AREA)
- Communicable Diseases (AREA)
- Pulmonology (AREA)
- Zoology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Otolaryngology (AREA)
- Biotechnology (AREA)
- AIDS & HIV (AREA)
- Biochemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Electrochromic Elements, Electrophoresis, Or Variable Reflection Or Absorption Elements (AREA)
- Devices For Checking Fares Or Tickets At Control Points (AREA)
- Digital Transmission Methods That Use Modulated Carrier Waves (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US12106108P | 2008-12-09 | 2008-12-09 | |
US17040409P | 2009-04-17 | 2009-04-17 | |
US22438609P | 2009-07-09 | 2009-07-09 | |
US22737809P | 2009-07-21 | 2009-07-21 | |
US24263509P | 2009-09-15 | 2009-09-15 |
Publications (1)
Publication Number | Publication Date |
---|---|
AP2011005745A0 true AP2011005745A0 (en) | 2011-06-30 |
Family
ID=41621203
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AP2011000745A AP2011005745A0 (en) | 2008-12-09 | 2009-12-07 | Modulators of toll-like receptors. |
Country Status (33)
Country | Link |
---|---|
US (8) | US8367670B2 (fr) |
EP (3) | EP2818469B1 (fr) |
JP (3) | JP5600116B2 (fr) |
KR (2) | KR101787309B1 (fr) |
CN (2) | CN102272134B (fr) |
AP (1) | AP2011005745A0 (fr) |
AR (1) | AR074506A1 (fr) |
AU (1) | AU2009333559B2 (fr) |
BR (1) | BRPI0923305B1 (fr) |
CA (1) | CA2745295C (fr) |
CL (1) | CL2011001392A1 (fr) |
CO (1) | CO6362010A2 (fr) |
CY (1) | CY1115176T1 (fr) |
DK (1) | DK2364314T3 (fr) |
EA (3) | EA026557B1 (fr) |
EC (2) | ECSP11011189A (fr) |
ES (2) | ES2467108T3 (fr) |
HK (2) | HK1161880A1 (fr) |
HR (1) | HRP20140539T1 (fr) |
IL (2) | IL213101A (fr) |
MX (1) | MX2011006152A (fr) |
NZ (2) | NZ612380A (fr) |
PE (1) | PE20120106A1 (fr) |
PL (1) | PL2364314T3 (fr) |
PT (2) | PT2364314E (fr) |
RS (1) | RS53347B (fr) |
SG (1) | SG172060A1 (fr) |
SI (1) | SI2364314T1 (fr) |
SM (1) | SMT201400083B (fr) |
TW (5) | TWI534136B (fr) |
UY (1) | UY32306A (fr) |
WO (1) | WO2010077613A1 (fr) |
ZA (1) | ZA201104998B (fr) |
Families Citing this family (235)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102272134B (zh) | 2008-12-09 | 2013-10-16 | 吉里德科学公司 | Toll样受体调节剂 |
JP5988492B2 (ja) | 2009-09-02 | 2016-09-07 | ノバルティス アーゲー | Tlr活性モジュレーターを含む免疫原性組成物 |
PL2477987T3 (pl) * | 2009-09-14 | 2018-06-29 | Gilead Sciences, Inc. | Modulatory receptorów toll-podobnych |
EP2516441B1 (fr) * | 2009-12-23 | 2015-01-21 | Elan Pharmaceuticals Inc. | Pteridinones en tant qu' inhibiteurs de plk (polo-like kinase) |
EA201890869A3 (ru) | 2010-06-03 | 2019-03-29 | Фармасайкликс, Инк. | Применение ингибиторов тирозинкиназы брутона (btk) |
EP2719395A1 (fr) | 2010-09-01 | 2014-04-16 | Novartis AG | Adsorption d'immunopotentiateurs sur des sels métalliques insolubles |
CA2822037A1 (fr) | 2010-12-20 | 2012-06-28 | Gilead Sciences, Inc. | Combinations pour traiter le vhc |
EP3208263A1 (fr) * | 2011-01-12 | 2017-08-23 | VentiRx Pharmaceuticals, Inc. | Benzoazépines substituées en tant que modulateurs de récepteurs de type toll |
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WO2013132041A2 (fr) | 2012-03-08 | 2013-09-12 | Novartis Ag | Formulations à adjuvant de vaccins de rappel |
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