JP2012067131A5 - - Google Patents

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Publication number
JP2012067131A5
JP2012067131A5 JP2011289220A JP2011289220A JP2012067131A5 JP 2012067131 A5 JP2012067131 A5 JP 2012067131A5 JP 2011289220 A JP2011289220 A JP 2011289220A JP 2011289220 A JP2011289220 A JP 2011289220A JP 2012067131 A5 JP2012067131 A5 JP 2012067131A5
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pyridinylmethoxy
anilino
quinolinyl
dimethylamino
ethoxy
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JP2011289220A
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Japanese (ja)
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JP5965640B2 (ja
JP2012067131A (ja
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JP2011289220A 2007-10-17 2011-12-28 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態 Active JP5965640B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12479607P 2007-10-17 2007-10-17
US61/124,796 2007-10-17

Related Parent Applications (1)

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JP2010258729A Division JP2011063610A (ja) 2007-10-17 2010-11-19 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態

Related Child Applications (1)

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JP2012279650A Division JP2013053170A (ja) 2007-10-17 2012-12-21 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態

Publications (3)

Publication Number Publication Date
JP2012067131A JP2012067131A (ja) 2012-04-05
JP2012067131A5 true JP2012067131A5 (enExample) 2013-02-14
JP5965640B2 JP5965640B2 (ja) 2016-08-10

Family

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Family Applications (11)

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JP2010530105A Pending JP2011500712A (ja) 2007-10-17 2008-10-16 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2010258729A Withdrawn JP2011063610A (ja) 2007-10-17 2010-11-19 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2011289220A Active JP5965640B2 (ja) 2007-10-17 2011-12-28 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2012279650A Pending JP2013053170A (ja) 2007-10-17 2012-12-21 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2015080748A Pending JP2015127352A (ja) 2007-10-17 2015-04-10 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2016238151A Active JP6412090B2 (ja) 2007-10-17 2016-12-08 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2018079067A Withdrawn JP2018109071A (ja) 2007-10-17 2018-04-17 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2020070281A Withdrawn JP2020111606A (ja) 2007-10-17 2020-04-09 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2021146090A Pending JP2021185200A (ja) 2007-10-17 2021-09-08 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2023160192A Withdrawn JP2023164747A (ja) 2007-10-17 2023-09-25 (e)-n-{4-[3-クロロ-4-(2-ピリジニルメトキシ)アニリノ]-3-シアノ-7-エトキシ-6-キノリニル}-4-(ジメチルアミノ)-2-ブテンアミドのマレイン酸塩およびその結晶形態
JP2025124961A Pending JP2025137789A (ja) 2007-10-17 2025-07-25 (e)-n-{4-[3-クロロ-4-(2-ピリジニルメトキシ)アニリノ]-3-シアノ-7-エトキシ-6-キノリニル}-4-(ジメチルアミノ)-2-ブテンアミドのマレイン酸塩およびその結晶形態

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JP2010530105A Pending JP2011500712A (ja) 2007-10-17 2008-10-16 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2010258729A Withdrawn JP2011063610A (ja) 2007-10-17 2010-11-19 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態

Family Applications After (8)

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JP2012279650A Pending JP2013053170A (ja) 2007-10-17 2012-12-21 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2015080748A Pending JP2015127352A (ja) 2007-10-17 2015-04-10 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2016238151A Active JP6412090B2 (ja) 2007-10-17 2016-12-08 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2018079067A Withdrawn JP2018109071A (ja) 2007-10-17 2018-04-17 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2020070281A Withdrawn JP2020111606A (ja) 2007-10-17 2020-04-09 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2021146090A Pending JP2021185200A (ja) 2007-10-17 2021-09-08 (e)−n−{4−[3−クロロ−4−(2−ピリジニルメトキシ)アニリノ]−3−シアノ−7−エトキシ−6−キノリニル}−4−(ジメチルアミノ)−2−ブテンアミドのマレイン酸塩およびその結晶形態
JP2023160192A Withdrawn JP2023164747A (ja) 2007-10-17 2023-09-25 (e)-n-{4-[3-クロロ-4-(2-ピリジニルメトキシ)アニリノ]-3-シアノ-7-エトキシ-6-キノリニル}-4-(ジメチルアミノ)-2-ブテンアミドのマレイン酸塩およびその結晶形態
JP2025124961A Pending JP2025137789A (ja) 2007-10-17 2025-07-25 (e)-n-{4-[3-クロロ-4-(2-ピリジニルメトキシ)アニリノ]-3-シアノ-7-エトキシ-6-キノリニル}-4-(ジメチルアミノ)-2-ブテンアミドのマレイン酸塩およびその結晶形態

Country Status (20)

Country Link
US (6) US8022216B2 (enExample)
EP (6) EP2258698A3 (enExample)
JP (11) JP2011500712A (enExample)
KR (5) KR20180041753A (enExample)
CN (7) CN106822127B (enExample)
AR (2) AR068932A1 (enExample)
AU (1) AU2008312474B2 (enExample)
BR (2) BR122019023745B8 (enExample)
CA (2) CA2928071C (enExample)
CL (1) CL2008003088A1 (enExample)
ES (3) ES2602123T3 (enExample)
IL (3) IL308687A (enExample)
IN (1) IN2015DN01135A (enExample)
MX (5) MX2010004173A (enExample)
NZ (3) NZ616136A (enExample)
PA (1) PA8800701A1 (enExample)
RU (2) RU2463300C2 (enExample)
SG (2) SG10201900175TA (enExample)
TW (1) TW200934761A (enExample)
WO (1) WO2009052264A2 (enExample)

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CN104513200B (zh) * 2013-09-26 2017-05-03 江苏苏中药业集团股份有限公司 取代丁烯酰胺的马来酸盐及其晶型
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CN111344280B (zh) * 2017-11-20 2022-08-12 苏州韬略生物科技股份有限公司 (e)-n-(3-氰基-7-乙氧基-4-((4-苯氧基苯基)氨基)喹啉-6-基)-4-(二甲基氨基) 丁-2-烯酰胺马来酸盐及晶型
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CN109053702A (zh) * 2018-08-13 2018-12-21 扬子江药业集团有限公司 一种阿法替尼类似物及其制备方法和用途
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