JP2015516425A5 - - Google Patents

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Publication number
JP2015516425A5
JP2015516425A5 JP2015511606A JP2015511606A JP2015516425A5 JP 2015516425 A5 JP2015516425 A5 JP 2015516425A5 JP 2015511606 A JP2015511606 A JP 2015511606A JP 2015511606 A JP2015511606 A JP 2015511606A JP 2015516425 A5 JP2015516425 A5 JP 2015516425A5
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JP
Japan
Prior art keywords
crystalline form
solution
powder
diffraction pattern
dimethylaminoethoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2015511606A
Other languages
English (en)
Japanese (ja)
Other versions
JP2015516425A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2013/039877 external-priority patent/WO2013169727A1/en
Publication of JP2015516425A publication Critical patent/JP2015516425A/ja
Publication of JP2015516425A5 publication Critical patent/JP2015516425A5/ja
Withdrawn legal-status Critical Current

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JP2015511606A 2012-05-07 2013-05-07 ６−ｏ−（４−ジメチルアミノエトキシ）シンナモイルフマギロールのシュウ酸塩の多形塩ならびにその製造および使用方法 Withdrawn JP2015516425A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261643586P 2012-05-07 2012-05-07
US61/643,586 2012-05-07
PCT/US2013/039877 WO2013169727A1 (en) 2012-05-07 2013-05-07 Polymorphic salt of the oxalate salt of 6 - o - ( 4 - dimethylaminoethoxy) cinnarnoyl fumagillol and methods of making and using same

Publications (2)

Publication Number Publication Date
JP2015516425A JP2015516425A (ja) 2015-06-11
JP2015516425A5 true JP2015516425A5 (enExample) 2016-06-23

Family

ID=48446683

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015511606A Withdrawn JP2015516425A (ja) 2012-05-07 2013-05-07 ６−ｏ−（４−ジメチルアミノエトキシ）シンナモイルフマギロールのシュウ酸塩の多形塩ならびにその製造および使用方法

Country Status (10)

Country Link
US (1) US9260419B2 (enExample)
EP (1) EP2847176A1 (enExample)
JP (1) JP2015516425A (enExample)
KR (1) KR20150016303A (enExample)
AU (1) AU2013259760A1 (enExample)
BR (1) BR112014027808A2 (enExample)
CA (1) CA2872649A1 (enExample)
IL (1) IL235521A (enExample)
MX (1) MX2014013525A (enExample)
WO (1) WO2013169727A1 (enExample)

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WO2011085198A1 (en) 2010-01-08 2011-07-14 Zafgen Corporation Metap-2 inhibitor for use in treating benign prostatic hypertrophy (bph)
WO2011127304A2 (en) 2010-04-07 2011-10-13 Zafgen Corporation Methods of treating an overweight subject
EP2763671A2 (en) 2011-10-03 2014-08-13 Zafgen, Inc. Methods of treating age related disorders
BR112014028041A2 (pt) 2012-05-08 2017-06-27 Zafgen Inc tratamento de obesidade hipotalâmica com inibidores de metap2
CA2873574A1 (en) 2012-05-09 2013-11-14 Zafgen, Inc. Fumagillol type compounds and methods of making and using same
AU2014236528A1 (en) 2013-03-14 2015-09-24 Zafgen, Inc. Methods of treating renal disease and other disorders
AR105671A1 (es) 2015-08-11 2017-10-25 Zafgen Inc Compuestos heterocíclicos de fumagillol y sus métodos de elaboración y uso
CN106432255A (zh) 2015-08-11 2017-02-22 扎夫根公司 烟曲霉素醇螺环化合物和制备和使用其的方法

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