JP2018520205A5 - - Google Patents

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Publication number
JP2018520205A5
JP2018520205A5 JP2018511323A JP2018511323A JP2018520205A5 JP 2018520205 A5 JP2018520205 A5 JP 2018520205A5 JP 2018511323 A JP2018511323 A JP 2018511323A JP 2018511323 A JP2018511323 A JP 2018511323A JP 2018520205 A5 JP2018520205 A5 JP 2018520205A5
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JP
Japan
Prior art keywords
formula
compound represented
crystalline form
mesylate salt
powder
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2018511323A
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English (en)
Japanese (ja)
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JP2018520205A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/CN2016/085360 external-priority patent/WO2016184436A1/zh
Publication of JP2018520205A publication Critical patent/JP2018520205A/ja
Publication of JP2018520205A5 publication Critical patent/JP2018520205A5/ja
Pending legal-status Critical Current

Links

JP2018511323A 2015-05-21 2016-06-08 レンバチニブメシル酸塩の新規結晶形及びその製造方法 Pending JP2018520205A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN201510263300 2015-05-21
CN201510263300.3 2015-05-21
PCT/CN2016/085360 WO2016184436A1 (zh) 2015-05-21 2016-06-08 乐伐替尼甲磺酸盐的新晶型及其制备方法

Publications (2)

Publication Number Publication Date
JP2018520205A JP2018520205A (ja) 2018-07-26
JP2018520205A5 true JP2018520205A5 (enExample) 2018-09-06

Family

ID=57319484

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2018511323A Pending JP2018520205A (ja) 2015-05-21 2016-06-08 レンバチニブメシル酸塩の新規結晶形及びその製造方法

Country Status (7)

Country Link
US (1) US10246418B2 (enExample)
EP (1) EP3287444A4 (enExample)
JP (1) JP2018520205A (enExample)
CN (2) CN107848979A (enExample)
IL (1) IL255738A (enExample)
MX (1) MX2017014799A (enExample)
WO (1) WO2016184436A1 (enExample)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112012003592B8 (pt) 2009-08-19 2021-05-25 Eisai R&D Man Co Ltd composição farmacêutica contendo derivado de quinolina
US10633533B2 (en) 2014-09-30 2020-04-28 Lg Chem, Ltd. Block copolymer
US10562855B2 (en) * 2016-06-08 2020-02-18 Crystal Pharmatech Co., Ltd. Crystalline form of lenvantinib mesylate and process of preparation thereof
RU2019123542A (ru) * 2016-12-29 2021-02-01 Др. Редди'З Лабораториз Лимитед Формы твердой фазы мезилата ленватиниба
CN110494423B (zh) * 2017-04-25 2022-04-26 苏州科睿思制药有限公司 乐伐替尼甲磺酸盐的新晶型及其制备方法
US11236050B2 (en) 2017-12-09 2022-02-01 Msn Laboratories Private Limited, R&D Center Polymorphs of 4-[3-chloro-4-(n′-cyclopropyl ureido)phenoxy] -7-methoxyquinoline-6-carboxamide, its salts and process for the preparation thereof
CN109988112A (zh) * 2017-12-29 2019-07-09 四川科伦药物研究院有限公司 仑伐替尼甲磺酸盐的晶型及其制备方法
CN112204011A (zh) * 2018-06-01 2021-01-08 成都苑东生物制药股份有限公司 一种甲磺酸乐伐替尼新晶型及其制备方法
CN110818634B (zh) * 2018-08-13 2021-11-30 上海新礼泰药业有限公司 甲磺酸乐伐替尼的精制方法
EP3620453A1 (en) 2018-09-07 2020-03-11 Indena S.p.A. New crystal form of lenvatinib
CN111574359A (zh) * 2019-02-19 2020-08-25 愈磐生物科技（苏州）有限公司 乐伐替尼-没食子酸共晶晶型及其应用
CN111689897B (zh) * 2019-03-13 2024-02-06 齐鲁制药有限公司 一种高纯度甲磺酸乐伐替尼晶型c的制备方法
CN109867626A (zh) * 2019-04-18 2019-06-11 安礼特（上海）医药科技有限公司 一种甲磺酸仑伐替尼多晶型物及其制备方法
CN110229103A (zh) * 2019-06-27 2019-09-13 尚科生物医药（上海）有限公司 一种乐伐替尼甲磺酸盐晶型b的制备方法
CN112174886A (zh) * 2019-07-02 2021-01-05 成都苑东生物制药股份有限公司 一种甲磺酸乐伐替尼晶型x的制备方法
WO2021007189A1 (en) 2019-07-08 2021-01-14 Rezolute, Inc. Crystalline forms of plasma kallikrein inhibitors
CN110563644A (zh) * 2019-10-30 2019-12-13 北京赛思源生物医药技术有限公司 一种仑伐替尼甲磺酸盐的新晶型
US11059787B2 (en) 2019-11-12 2021-07-13 Shenzhen Bolan Pharmaceutical Co., Ltd Crystalline form of lenvatinib mesylate and methods thereof
CN117945999B (zh) * 2020-01-19 2025-08-22 重庆医药工业研究院有限责任公司 一种氟伐替尼或甲磺酸盐的晶型及其制备方法
CN114174264B (zh) * 2020-04-24 2024-02-27 成都苑东生物制药股份有限公司 一种甲磺酸仑伐替尼晶型xi及其制备方法
CN112939859B (zh) * 2021-02-03 2022-03-11 南京方生和医药科技有限公司 甲磺酸仑伐替尼m晶型的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6627646B2 (en) * 2001-07-17 2003-09-30 Sepracor Inc. Norastemizole polymorphs
KR100839554B1 (ko) * 2003-12-25 2008-06-20 에자이 알앤드디 매니지먼트 가부시키가이샤 4-(3-클로로-4-(시클로프로필아미노카르보닐)아미노페녹시)-7-메톡시-6-퀴놀린카르복사미드의 염 또는 그 용매화물의결정 및 이들의 제조 방법
ATE428421T1 (de) * 2004-09-17 2009-05-15 Eisai R&D Man Co Ltd Medizinische zusammensetzung mit verbesserter stabilität und reduzierten gelierungseigenschaften
AU2006260148B9 (en) * 2005-06-23 2009-09-17 Eisai R&D Managment Co., Ltd. Amorphous salt of 4-(3-chloro-4-(cyclopropylaminocarbonyl)aminophenoxy)- 7-methoxy-6-quinolinecarboxamide and process for producing the same
BR112012003592B8 (pt) * 2009-08-19 2021-05-25 Eisai R&D Man Co Ltd composição farmacêutica contendo derivado de quinolina

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