JP2013237682A5 - - Google Patents

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Publication number
JP2013237682A5
JP2013237682A5 JP2013147411A JP2013147411A JP2013237682A5 JP 2013237682 A5 JP2013237682 A5 JP 2013237682A5 JP 2013147411 A JP2013147411 A JP 2013147411A JP 2013147411 A JP2013147411 A JP 2013147411A JP 2013237682 A5 JP2013237682 A5 JP 2013237682A5
Authority
JP
Japan
Prior art keywords
crystalline form
aripiprazole crystalline
degrees
aripiprazole
pharmaceutical composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2013147411A
Other languages
English (en)
Japanese (ja)
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JP2013237682A (ja
Filing date
Publication date
Application filed filed Critical
Publication of JP2013237682A publication Critical patent/JP2013237682A/ja
Publication of JP2013237682A5 publication Critical patent/JP2013237682A5/ja
Pending legal-status Critical Current

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JP2013147411A 2003-12-16 2013-07-16 アリピプラゾール結晶質形態を調製する方法 Pending JP2013237682A (ja)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US53029703P 2003-12-16 2003-12-16
US60/530,297 2003-12-16
US53383103P 2003-12-30 2003-12-30
US60/533,831 2003-12-30
US61840404P 2004-10-13 2004-10-13
US60/618,404 2004-10-13
US61896004P 2004-10-14 2004-10-14
US60/618,960 2004-10-14

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2006545583A Division JP5546717B2 (ja) 2003-12-16 2004-12-16 アリピプラゾール結晶質形態を調製する方法

Publications (2)

Publication Number Publication Date
JP2013237682A JP2013237682A (ja) 2013-11-28
JP2013237682A5 true JP2013237682A5 (enExample) 2014-06-19

Family

ID=34705304

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2006545583A Expired - Lifetime JP5546717B2 (ja) 2003-12-16 2004-12-16 アリピプラゾール結晶質形態を調製する方法
JP2013147411A Pending JP2013237682A (ja) 2003-12-16 2013-07-16 アリピプラゾール結晶質形態を調製する方法

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2006545583A Expired - Lifetime JP5546717B2 (ja) 2003-12-16 2004-12-16 アリピプラゾール結晶質形態を調製する方法

Country Status (11)

Country Link
US (2) US7504504B2 (enExample)
EP (1) EP1613598B1 (enExample)
JP (2) JP5546717B2 (enExample)
AT (1) ATE529409T1 (enExample)
CA (1) CA2550726A1 (enExample)
ES (1) ES2374922T3 (enExample)
IL (1) IL175512A (enExample)
PL (1) PL1613598T3 (enExample)
PT (1) PT1613598E (enExample)
TW (1) TW200529850A (enExample)
WO (1) WO2005058835A2 (enExample)

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EP1919453A2 (en) * 2005-12-22 2008-05-14 Teva Pharmaceutical Industries Ltd Processes for reducing particle size of aripiprazole
PL1808164T3 (pl) 2006-01-05 2009-06-30 Teva Pharma Sposób z granulacją na mokro do wytwarzania kompozycji farmaceutycznych aripiprazolu
DE602006006536D1 (de) * 2006-01-05 2009-06-10 Teva Pharma Trockene Aripiprazolformulierungen
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EP1880714A1 (en) 2006-07-20 2008-01-23 Helm AG Amorphous Aripiprazole and Process for the Preparation thereof
US7799790B2 (en) 2006-07-20 2010-09-21 Helm Ag Amorphous aripiprazole and process for the preparation thereof
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WO2008051541A2 (en) * 2006-10-24 2008-05-02 Cambrex Charles City, Inc. Process for preparing anhydrous aripirazole type i
ES2353444T3 (es) 2008-01-23 2011-03-02 Helm Ag Aripiprazol amorfo y procedimiento para su preparación.
EP2238976B1 (en) 2009-04-03 2012-06-27 Hexal AG Oral films comprising 7-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]-3,4-dihydro- 1H-quinolin-2-one base or salts or hydrates thereof
CN101948426A (zh) * 2010-09-13 2011-01-19 浙江华海药业股份有限公司 一种制备阿立哌唑晶型b的新方法
US9757374B2 (en) 2010-10-28 2017-09-12 Aequus Pharmaceuticals Inc. Aripiprazole compositions and methods for its transdermal delivery
EP2632463B1 (en) 2010-10-28 2018-04-04 Aequus Pharmaceuticals Inc. Aripiprazole compositions and methods for their transdermal delivery
WO2012077134A1 (en) * 2010-12-07 2012-06-14 Ind-Swift Laboratories Limted Process for preparing aripiprazole polymorphs
KR101340214B1 (ko) * 2011-03-31 2013-12-10 주식회사 대웅제약 무수 아리피프라졸 ⅱ형 결정의 제조방법
CN102850268B (zh) * 2011-06-27 2015-07-15 上海中西制药有限公司 阿立哌唑ⅰ型微晶、阿立哌唑固体制剂及制备方法
KR101372840B1 (ko) * 2012-08-02 2014-03-12 주식회사 에스텍파마 무수 아리피프라졸 결정의 제조방법
WO2015067313A1 (en) 2013-11-07 2015-05-14 Synthon B.V. Orodispersible pharmaceutical compositions comprising aripiprazole
EP3578546A1 (en) 2013-11-15 2019-12-11 Akebia Therapeutics Inc. Solid forms of {[5-(3-chlorophenyl)-3-hydroxypyridine-2-carbonyl]amino}acetic acid, compositions, and uses thereof
CN106474058B (zh) 2015-08-31 2020-01-07 南京诺瑞特医药科技有限公司 具有延长的保质期的阿立哌唑可注射悬浮液制剂
TWI665194B (zh) * 2016-02-19 2019-07-11 諾瑞特國際藥業股份有限公司 阿立哌唑的新晶型

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EP1812397A1 (en) * 2004-11-18 2007-08-01 Synthon B.V. Process of making crystalline aripiprazole
WO2006053780A1 (en) * 2004-11-18 2006-05-26 Synthon B.V. Crystalline aripiprazole solvates
EP1686117A1 (en) * 2005-01-27 2006-08-02 Sandoz AG Polymorph and solvates of aripiprazole
US20070148100A1 (en) * 2005-09-15 2007-06-28 Elan Pharma International, Limited Nanoparticulate aripiprazole formulations
EP1919453A2 (en) * 2005-12-22 2008-05-14 Teva Pharmaceutical Industries Ltd Processes for reducing particle size of aripiprazole
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WO2007113846A1 (en) * 2006-04-03 2007-10-11 Alembic Limited A process for the preparation of aripiprazole
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EP1880714A1 (en) * 2006-07-20 2008-01-23 Helm AG Amorphous Aripiprazole and Process for the Preparation thereof

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