JP2011522827A5 - - Google Patents

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Publication number
JP2011522827A5
JP2011522827A5 JP2011512645A JP2011512645A JP2011522827A5 JP 2011522827 A5 JP2011522827 A5 JP 2011522827A5 JP 2011512645 A JP2011512645 A JP 2011512645A JP 2011512645 A JP2011512645 A JP 2011512645A JP 2011522827 A5 JP2011522827 A5 JP 2011522827A5
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JP
Japan
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medicament
mammals
mammals use
purity
pharmaceutical composition
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JP2011512645A
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English (en)
Japanese (ja)
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JP2011522827A (ja
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Priority claimed from PCT/US2009/046256 external-priority patent/WO2009149258A2/en
Publication of JP2011522827A publication Critical patent/JP2011522827A/ja
Publication of JP2011522827A5 publication Critical patent/JP2011522827A5/ja
Pending legal-status Critical Current

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JP2011512645A 2008-06-04 2009-06-04 ６−［（４ｓ）−２−メチル−４−（２−ナフチル）−１，２，３，４−テトラヒドロイソキノリン−７−イル］ピリダジン−３−アミンの結晶形 Pending JP2011522827A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5871708P 2008-06-04 2008-06-04
US61/058,717 2008-06-04
PCT/US2009/046256 WO2009149258A2 (en) 2008-06-04 2009-06-04 Crystalline form of 6-[(4s)-2-methyl-4-(2-naphthyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridazin-3-amine

Publications (2)

Publication Number Publication Date
JP2011522827A JP2011522827A (ja) 2011-08-04
JP2011522827A5 true JP2011522827A5 (enExample) 2012-08-09

Family

ID=41277466

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2011512646A Expired - Fee Related JP5567557B2 (ja) 2008-06-04 2009-06-04 テトラヒドロイソキノリンの製造方法
JP2011512645A Pending JP2011522827A (ja) 2008-06-04 2009-06-04 ６−［（４ｓ）−２−メチル−４−（２−ナフチル）−１，２，３，４−テトラヒドロイソキノリン−７−イル］ピリダジン−３−アミンの結晶形
JP2014100580A Pending JP2014169312A (ja) 2008-06-04 2014-05-14 テトラヒドロイソキノリンの製造方法

Family Applications Before (1)

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JP2011512646A Expired - Fee Related JP5567557B2 (ja) 2008-06-04 2009-06-04 テトラヒドロイソキノリンの製造方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2014100580A Pending JP2014169312A (ja) 2008-06-04 2014-05-14 テトラヒドロイソキノリンの製造方法

Country Status (9)

Country Link
US (4) US8445494B2 (enExample)
EP (2) EP2280955B8 (enExample)
JP (3) JP5567557B2 (enExample)
KR (1) KR20110011653A (enExample)
CN (2) CN102112465B (enExample)
AR (1) AR071997A1 (enExample)
ES (1) ES2652462T3 (enExample)
TW (1) TW201002682A (enExample)
WO (2) WO2009149259A2 (enExample)

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KR101389246B1 (ko) 2004-07-15 2014-04-24 브리스톨-마이어스스퀴브컴파니 아릴- 및 헤테로아릴-치환된 테트라히드로이소퀴놀린, 및 이것의 노르에피네프린, 도파민 및 세로토닌의 재흡수를 차단하기 위한 용도
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CN102638982B (zh) 2009-05-12 2015-07-08 百时美施贵宝公司 (S)-7-([1,2,4]三唑并[1,5-a]吡啶-6-基)-4-(3,4-二氯苯基)-1,2,3,4-四氢异喹啉的晶型及其用途
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US9045468B2 (en) 2010-08-17 2015-06-02 Albany Molecular Research, Inc. 2,5-methano- and 2,5-ethano-tetrahydrobenzazepine derivatives and use thereof to block reuptake of norepinephrine, dopamine, and serotonin
NO2686520T3 (enExample) 2011-06-06 2018-03-17
JP6440625B2 (ja) 2012-11-14 2018-12-19 ザ・ジョンズ・ホプキンス・ユニバーシティー 精神分裂病を処置するための方法および組成物
WO2014159501A2 (en) * 2013-03-14 2014-10-02 Bristol-Myers Squibb Company Processes for preparing tetrahydroisoquinolines
CN103601699A (zh) * 2013-11-04 2014-02-26 南京大学 一类1,3,4-噻二唑-2-酰胺衍生物及其制备方法
KR102495018B1 (ko) 2013-11-15 2023-02-06 아케비아 테라퓨틱스 인코포레이티드 ｛[5-(3-클로로페닐)-3-하이드록시피리딘-2-카보닐]아미노｝아세트산의 고체형, 이의 조성물 및 용도
TW202406895A (zh) 2018-05-09 2024-02-16 美商阿克比治療有限公司 用於製備2-[[5-(3-氯苯基)-3-羥基吡啶-2-羰基]胺基]乙酸之方法
US11524939B2 (en) 2019-11-13 2022-12-13 Akebia Therapeutics, Inc. Solid forms of {[5-(3-chlorophenyl)-3-hydroxypyridine-2-carbonyl]amino} acetic acid

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