IL143089A0 - N-[4-(3-chloro-4-fluoro-phenylamino)-7-(3-morpholin-4-yl-propoxy)-quinazolin-6-yl]-acrylamide, an irreversible inhibitor of tyrosine kinases - Google Patents

N-[4-(3-chloro-4-fluoro-phenylamino)-7-(3-morpholin-4-yl-propoxy)-quinazolin-6-yl]-acrylamide, an irreversible inhibitor of tyrosine kinases

Info

Publication number
IL143089A0
IL143089A0 IL14308999A IL14308999A IL143089A0 IL 143089 A0 IL143089 A0 IL 143089A0 IL 14308999 A IL14308999 A IL 14308999A IL 14308999 A IL14308999 A IL 14308999A IL 143089 A0 IL143089 A0 IL 143089A0
Authority
IL
Israel
Prior art keywords
quinazolin
morpholin
phenylamino
propoxy
acrylamide
Prior art date
Application number
IL14308999A
Other languages
English (en)
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of IL143089A0 publication Critical patent/IL143089A0/xx

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL14308999A 1998-11-19 1999-09-23 N-[4-(3-chloro-4-fluoro-phenylamino)-7-(3-morpholin-4-yl-propoxy)-quinazolin-6-yl]-acrylamide, an irreversible inhibitor of tyrosine kinases IL143089A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10906598P 1998-11-19 1998-11-19
PCT/US1999/022116 WO2000031048A1 (en) 1998-11-19 1999-09-23 N-[4-(3-chloro-4-fluoro-phenylamino)-7-(3-morpholin-4-yl-propoxy)-quinazolin-6-yl]-acrylamide, an irreversible inhibitor of tyrosine kinases

Publications (1)

Publication Number Publication Date
IL143089A0 true IL143089A0 (en) 2002-04-21

Family

ID=22325607

Family Applications (1)

Application Number Title Priority Date Filing Date
IL14308999A IL143089A0 (en) 1998-11-19 1999-09-23 N-[4-(3-chloro-4-fluoro-phenylamino)-7-(3-morpholin-4-yl-propoxy)-quinazolin-6-yl]-acrylamide, an irreversible inhibitor of tyrosine kinases

Country Status (31)

Country Link
US (1) US6344455B1 (US07585860-20090908-C00112.png)
EP (1) EP1131304B1 (US07585860-20090908-C00112.png)
JP (1) JP3687900B2 (US07585860-20090908-C00112.png)
KR (1) KR20010080491A (US07585860-20090908-C00112.png)
CN (1) CN1160338C (US07585860-20090908-C00112.png)
AR (1) AR023706A1 (US07585860-20090908-C00112.png)
AT (1) ATE229008T1 (US07585860-20090908-C00112.png)
AU (1) AU763626B2 (US07585860-20090908-C00112.png)
BG (1) BG105608A (US07585860-20090908-C00112.png)
BR (1) BR9915487A (US07585860-20090908-C00112.png)
CA (1) CA2349721A1 (US07585860-20090908-C00112.png)
CO (1) CO5150185A1 (US07585860-20090908-C00112.png)
CZ (1) CZ20011759A3 (US07585860-20090908-C00112.png)
DE (1) DE69904358T2 (US07585860-20090908-C00112.png)
DK (1) DK1131304T3 (US07585860-20090908-C00112.png)
EA (1) EA003786B1 (US07585860-20090908-C00112.png)
EE (1) EE200100271A (US07585860-20090908-C00112.png)
ES (1) ES2188254T3 (US07585860-20090908-C00112.png)
GE (1) GEP20032997B (US07585860-20090908-C00112.png)
HK (1) HK1041695A1 (US07585860-20090908-C00112.png)
HU (1) HUP0104211A3 (US07585860-20090908-C00112.png)
IL (1) IL143089A0 (US07585860-20090908-C00112.png)
NO (1) NO319357B1 (US07585860-20090908-C00112.png)
NZ (2) NZ512189A (US07585860-20090908-C00112.png)
PE (1) PE20001242A1 (US07585860-20090908-C00112.png)
PL (1) PL347717A1 (US07585860-20090908-C00112.png)
PT (1) PT1131304E (US07585860-20090908-C00112.png)
SK (1) SK283688B6 (US07585860-20090908-C00112.png)
UY (1) UY25809A1 (US07585860-20090908-C00112.png)
WO (1) WO2000031048A1 (US07585860-20090908-C00112.png)
ZA (1) ZA200103535B (US07585860-20090908-C00112.png)

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