CY1108101T1 - Ενωσεις πυριμιδινης και η χρηση τους στην παρασκευη ενος τριαζολο-πυριμιδιν καρβα νουκλεοζιτη - Google Patents
Ενωσεις πυριμιδινης και η χρηση τους στην παρασκευη ενος τριαζολο-πυριμιδιν καρβα νουκλεοζιτηInfo
- Publication number
- CY1108101T1 CY1108101T1 CY20081100388T CY081100388T CY1108101T1 CY 1108101 T1 CY1108101 T1 CY 1108101T1 CY 20081100388 T CY20081100388 T CY 20081100388T CY 081100388 T CY081100388 T CY 081100388T CY 1108101 T1 CY1108101 T1 CY 1108101T1
- Authority
- CY
- Cyprus
- Prior art keywords
- pyrimidine
- nucleozite
- trizolo
- preparing
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Η παρούσα εφεύρεση αναφέρεται σε μία ένωση πυριμιδίνης (I) χρήσιμη ως φαρμακευτικό ενδιάμεσο, σε μία διαδικασία για την παρασκευή της εν λόγω ένωσης πυριμιδίνης, σε ενδιάμεσα που χρησιμοποιούνται στην εν λόγω διαδικασία, και στη χρήση της εν λόγω ένωσης πυριμιδίνης στην παρασκευή των φαρμακευτικών.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0013488.2A GB0013488D0 (en) | 2000-06-02 | 2000-06-02 | Chemical compound |
SE0002102A SE0002102D0 (sv) | 2000-06-02 | 2000-06-06 | Chemical compound |
EP01937111A EP1299390B1 (en) | 2000-06-02 | 2001-05-31 | Pyrimidine compounds and their use in the preparation of a triazolo -pyrimidine carba nucleoside |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1108101T1 true CY1108101T1 (el) | 2014-02-12 |
Family
ID=26244413
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20081100388T CY1108101T1 (el) | 2000-06-02 | 2008-04-09 | Ενωσεις πυριμιδινης και η χρηση τους στην παρασκευη ενος τριαζολο-πυριμιδιν καρβα νουκλεοζιτη |
Country Status (36)
Country | Link |
---|---|
US (6) | US7067663B2 (el) |
EP (1) | EP1299390B1 (el) |
JP (1) | JP4947870B2 (el) |
KR (2) | KR100802884B1 (el) |
CN (3) | CN100354268C (el) |
AR (1) | AR028605A1 (el) |
AT (1) | ATE386039T1 (el) |
AU (4) | AU6287601A (el) |
BG (1) | BG65866B1 (el) |
BR (1) | BR0111319A (el) |
CA (1) | CA2408914C (el) |
CY (1) | CY1108101T1 (el) |
CZ (3) | CZ302644B6 (el) |
DE (1) | DE60132776T2 (el) |
DK (1) | DK1299390T3 (el) |
EE (1) | EE05223B1 (el) |
ES (1) | ES2299487T3 (el) |
GB (1) | GB0013488D0 (el) |
HK (1) | HK1053122A1 (el) |
HU (1) | HU229281B1 (el) |
IL (3) | IL152776A0 (el) |
IS (1) | IS2600B (el) |
MX (2) | MXPA02011793A (el) |
MY (1) | MY131942A (el) |
NO (1) | NO324266B1 (el) |
NZ (1) | NZ522637A (el) |
PL (3) | PL210375B1 (el) |
PT (1) | PT1299390E (el) |
RU (1) | RU2295526C2 (el) |
SE (1) | SE0002102D0 (el) |
SI (1) | SI1299390T1 (el) |
SK (1) | SK286845B6 (el) |
TW (1) | TWI285203B (el) |
UA (1) | UA73182C2 (el) |
WO (1) | WO2001092263A1 (el) |
ZA (1) | ZA200209068B (el) |
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SI2340252T1 (sl) | 2008-09-09 | 2016-02-29 | Astrazeneca Ab | Postopek priprave (1S-)1-alfa, 2-alfa, 3-beta(1S*,2R*)5-beta))-3-(7-(2-(3,4-difluorofenil)-ciklopropilamino)-5- (propiltio)-3H-1,2,3-triazolo(4,5-D)pirimidin-3-il)-5-(2-hidroksietoksi) ciklopentan-1,2-diola in njegovih vmesnih spojin |
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CA2859743A1 (en) | 2010-12-20 | 2012-06-28 | Actavis Group Ptc Ehf | Novel processes for preparing triazolo[4,5-d]pyrimidine derivatives and intermediates thereof |
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DE69621021T2 (de) | 1995-07-11 | 2002-10-31 | Astrazeneca Ab | Inhibitoren der plättchenaggregation |
WO1998028300A1 (en) * | 1996-12-20 | 1998-07-02 | Astra Pharmaceuticals Ltd. | Triazolo[4,5-d]pyrimidinyl derivatives and their use as medicaments |
TW530058B (en) | 1997-07-22 | 2003-05-01 | Astra Pharma Prod | Triazolo [4,5-d]pyrimidine compounos and their use and process for preparation |
SE9702773D0 (sv) * | 1997-07-22 | 1997-07-22 | Astra Pharma Prod | Novel compounds |
TR200002380T2 (tr) * | 1998-02-17 | 2001-03-21 | Astrazeneca Uk Limited | Yeni triazolo (4,5-d) pirimidin bileşikleri |
TWI229674B (en) * | 1998-12-04 | 2005-03-21 | Astra Pharma Prod | Novel triazolo[4,5-d]pyrimidine compounds, pharmaceutical composition containing the same, their process for preparation and uses |
CZ20002947A3 (cs) * | 1999-02-05 | 2000-11-15 | Astrazeneca Uk Limited | Nové triazolo(4,5-d)pyrimidiny, způsob jejich přípravy a farmaceutický prostředek, který je obsahuje |
SE9904129D0 (sv) * | 1999-11-15 | 1999-11-15 | Astra Pharma Prod | Novel compounds |
GB0013407D0 (en) * | 2000-06-02 | 2000-07-26 | Astrazeneca Ab | Forms of a chemical compound |
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2000
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2001
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