BR112015004205A2 - sulfamoil-arilamidas e o uso das mesmas como medicamentos para o tratamento da hepatite b - Google Patents

sulfamoil-arilamidas e o uso das mesmas como medicamentos para o tratamento da hepatite b

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Publication number
BR112015004205A2
BR112015004205A2 BR112015004205A BR112015004205A BR112015004205A2 BR 112015004205 A2 BR112015004205 A2 BR 112015004205A2 BR 112015004205 A BR112015004205 A BR 112015004205A BR 112015004205 A BR112015004205 A BR 112015004205A BR 112015004205 A2 BR112015004205 A2 BR 112015004205A2
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Prior art keywords
arylamides
sulfamoyl
hepatitis
treatment
medicines
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BR112015004205A
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English (en)
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BR112015004205B1 (pt
Inventor
Rombouts Geert
Vandyck Koen
Jean-Marie Bernard Raboisson Pierre
Julien Last Stefaan
Gaston Verschueren Wim
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Janssen Sciences Ireland Uc
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Application filed by Janssen Sciences Ireland Uc filed Critical Janssen Sciences Ireland Uc
Publication of BR112015004205A2 publication Critical patent/BR112015004205A2/pt
Publication of BR112015004205B1 publication Critical patent/BR112015004205B1/pt

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    • C07C311/15Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
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Abstract

resumo patente de invenção: "sulfamoil-arilamidas e o uso das mesmas como medicamentos para o tratamento da hepatite b". inibidores da replicação do hbv da fórmula (i) incluindo formas estereoquimicamente isoméricas, e sais, hidratos, solvatos dos mesmos, em que b, r1, r2 e r4 têm o significado como definido aqui. a presente invenção se relaciona também a processos para preparação dos referidos compostos, composições farmacêuticas contendo os mesmos e seu uso, sozinhos ou em combinação com outros inibidores do hbv, na terapia contra o hbv.
BR112015004205-8A 2012-08-28 2013-08-28 Sulfamoil-arilamidas, seu uso das mesmas como medicamentos para o tratamento da hepatite b, composição farmacêutica que as compreende e produto BR112015004205B1 (pt)

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EP12182076.5 2012-08-28
EP12182076 2012-08-28
EP12185055.6 2012-09-19
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EP12190837.0 2012-10-31
EP12190837 2012-10-31
EP13157230.7 2013-02-28
EP13157230 2013-02-28
EP13169574.4 2013-05-28
EP13169574 2013-05-28
PCT/EP2013/067829 WO2014033176A1 (en) 2012-08-28 2013-08-28 Sulfamoyl-arylamides and the use thereof as medicaments for the treatment of hepatitis b

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BR112015004192-2A BR112015004192B1 (pt) 2012-08-28 2013-08-28 sulfamoíl-arilamidas, composição farmacêutica que os compreende e uso das mesmas no tratamento da hepatite b

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