SG10201605291WA - Sulfamoyl-arylamides and the use thereof as medicaments for the treatment of hepatitis b - Google Patents

Sulfamoyl-arylamides and the use thereof as medicaments for the treatment of hepatitis b

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Publication number
SG10201605291WA
SG10201605291WA SG10201605291WA SG10201605291WA SG10201605291WA SG 10201605291W A SG10201605291W A SG 10201605291WA SG 10201605291W A SG10201605291W A SG 10201605291WA SG 10201605291W A SG10201605291W A SG 10201605291WA SG 10201605291W A SG10201605291W A SG 10201605291WA
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Singapore
Prior art keywords
arylamides
sulfamoyl
medicaments
hepatitis
treatment
Prior art date
Application number
SG10201605291WA
Inventor
Koen Vandyck
Stefaan Julien Last
Geert Rombouts
Wim Gaston Verschueren
Pierre Jean-Marie Bernard Raboisson
Original Assignee
Janssen Sciences Ireland Uc
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Publication date
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Application filed by Janssen Sciences Ireland Uc filed Critical Janssen Sciences Ireland Uc
Publication of SG10201605291WA publication Critical patent/SG10201605291WA/en

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    • C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/37—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
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    • C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
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    • A61K31/18—Sulfonamides
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4453—Non condensed piperidines, e.g. piperocaine only substituted in position 1, e.g. propipocaine, diperodon
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
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    • C07C311/20—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
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