SK285768B6 - Imidazopyridínové deriváty inhibujúce vylučovaniežalúdočnej kyseliny, spôsob ich prípravy, farmaceutický prostriedok a ich použitie - Google Patents

Imidazopyridínové deriváty inhibujúce vylučovaniežalúdočnej kyseliny, spôsob ich prípravy, farmaceutický prostriedok a ich použitie Download PDF

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Publication number
SK285768B6
SK285768B6 SK1492-2000A SK14922000A SK285768B6 SK 285768 B6 SK285768 B6 SK 285768B6 SK 14922000 A SK14922000 A SK 14922000A SK 285768 B6 SK285768 B6 SK 285768B6
Authority
SK
Slovakia
Prior art keywords
formula
pyridine
compound
carboxamide
dimethyl
Prior art date
Application number
SK1492-2000A
Other languages
English (en)
Slovak (sk)
Other versions
SK14922000A3 (sk
Inventor
Kosrat Amin
Mikael Dahlstrm
Peter Nordberg
Ingemar Starke
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of SK14922000A3 publication Critical patent/SK14922000A3/sk
Publication of SK285768B6 publication Critical patent/SK285768B6/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SK1492-2000A 1998-04-29 1999-04-23 Imidazopyridínové deriváty inhibujúce vylučovaniežalúdočnej kyseliny, spôsob ich prípravy, farmaceutický prostriedok a ich použitie SK285768B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9801526A SE9801526D0 (sv) 1998-04-29 1998-04-29 New compounds
PCT/SE1999/000663 WO1999055706A1 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion

Publications (2)

Publication Number Publication Date
SK14922000A3 SK14922000A3 (sk) 2001-06-11
SK285768B6 true SK285768B6 (sk) 2007-07-06

Family

ID=20411154

Family Applications (2)

Application Number Title Priority Date Filing Date
SK1492-2000A SK285768B6 (sk) 1998-04-29 1999-04-23 Imidazopyridínové deriváty inhibujúce vylučovaniežalúdočnej kyseliny, spôsob ich prípravy, farmaceutický prostriedok a ich použitie
SK1491-2000A SK14912000A3 (sk) 1998-04-29 1999-04-23 Imidazopyridínové deriváty, ktoré inhibujú vylučovanie žalúdočnej kyseliny, spôsob ich prípravy, medziprodukty tohto spôsobu a farmaceutická formulácia

Family Applications After (1)

Application Number Title Priority Date Filing Date
SK1491-2000A SK14912000A3 (sk) 1998-04-29 1999-04-23 Imidazopyridínové deriváty, ktoré inhibujú vylučovanie žalúdočnej kyseliny, spôsob ich prípravy, medziprodukty tohto spôsobu a farmaceutická formulácia

Country Status (34)

Country Link
US (2) US6313137B1 (ja)
EP (4) EP1491543B1 (ja)
JP (2) JP3883383B2 (ja)
KR (3) KR100650472B1 (ja)
CN (2) CN1174980C (ja)
AR (2) AR015769A1 (ja)
AT (4) ATE372340T1 (ja)
AU (2) AU769108B2 (ja)
BR (2) BR9909995B1 (ja)
CA (2) CA2329921A1 (ja)
CZ (2) CZ292567B6 (ja)
DE (4) DE69937077T2 (ja)
DK (2) DK1073657T3 (ja)
EE (2) EE04916B1 (ja)
ES (2) ES2249913T3 (ja)
HK (5) HK1033457A1 (ja)
HU (2) HUP0102313A3 (ja)
ID (2) ID26819A (ja)
IL (4) IL139297A0 (ja)
IS (2) IS5684A (ja)
MY (2) MY121389A (ja)
NO (2) NO318203B1 (ja)
NZ (2) NZ507638A (ja)
PL (2) PL195000B1 (ja)
RU (2) RU2235725C2 (ja)
SA (2) SA99200065B1 (ja)
SE (1) SE9801526D0 (ja)
SI (1) SI1073656T1 (ja)
SK (2) SK285768B6 (ja)
TR (4) TR200102612T2 (ja)
TW (2) TWI250159B (ja)
UA (2) UA66846C2 (ja)
WO (2) WO1999055706A1 (ja)
ZA (2) ZA200005797B (ja)

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SE9802794D0 (sv) * 1998-08-21 1998-08-21 Astra Ab New compounds
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SE0003186D0 (sv) * 2000-09-07 2000-09-07 Astrazeneca Ab New process
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
SE0100295D0 (sv) * 2001-02-01 2001-02-01 Astrazeneca Ab New compounds
SE0100297D0 (sv) * 2001-02-01 2001-02-01 Astrazeneca Ab New compounds
SE0100296D0 (sv) * 2001-02-01 2001-02-01 Astrazeneca Ab New compounds
WO2002064121A1 (en) * 2001-02-13 2002-08-22 Astrazeneca Ab Novel modified released formulation
WO2002069968A1 (en) * 2001-03-08 2002-09-12 Astrazeneca Ab New use
SE0102808D0 (sv) * 2001-08-22 2001-08-22 Astrazeneca Ab New compounds
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
SE0201939D0 (sv) * 2002-06-20 2002-06-20 Astrazeneca Ab New combination
SE0201940D0 (sv) * 2002-06-20 2002-06-20 Astrazeneca Ab New combination II
CN100549011C (zh) 2002-09-19 2009-10-14 先灵公司 用作细胞周期蛋白依赖性激酶抑制剂的新颖咪唑并吡啶
CA2506027A1 (en) 2002-11-19 2004-06-03 Altana Pharma Ag 8-substituted imidazopyridines
AR043002A1 (es) * 2003-02-18 2005-07-13 Altana Pharma Ag Imidazopirazinas 6-substituidos
PT2476667E (pt) * 2003-02-26 2014-09-18 Sugen Inc Compostos de aminoheteroarilo como inibidores da proteína quinase
KR101179012B1 (ko) 2003-03-10 2012-09-03 니코메드 게엠베하 로플루미라스트 신규한 제조 방법
SE525349C2 (sv) * 2003-06-23 2005-02-08 Volvo Penta Ab Utombordsdrev för båtar
SE0301904D0 (sv) * 2003-06-26 2003-06-26 Astrazeneca Ab Novel imidazopyridine compound II with therapeutic effect
SE0301903D0 (sv) * 2003-06-26 2003-06-26 Astrazeneca Ab Novel imidazopyridine compound III with therapeutic effect
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US8993599B2 (en) 2003-07-18 2015-03-31 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
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SE0303451D0 (sv) * 2003-12-18 2003-12-18 Astrazeneca Ab New compounds
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US8906940B2 (en) 2004-05-25 2014-12-09 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
US20090291977A1 (en) * 2004-12-17 2009-11-26 Madoka Jinno Chromane Derivatives Useful As Acid Pump Antagonists
AU2006224619B2 (en) 2005-03-16 2012-06-07 Takeda Gmbh Taste masked dosage form containing roflumilast
AR056187A1 (es) * 2005-03-21 2007-09-26 S Bio Pte Ltd Derivados de imidazo[1,2-a)piridina: preparacion, composiciones farmaceuticas y uso para preparar medicamentos
US7666880B2 (en) 2005-03-21 2010-02-23 S*Bio Pte Ltd. Imidazo[1,2-A]pyridine derivatives: preparation and pharmaceutical applications
JP2008536817A (ja) * 2005-03-24 2008-09-11 グラクソ グループ リミテッド 胃腸疾患の処置用医薬として有用なイミダゾ（１，２−ａ）ピリジン誘導体
GB0513423D0 (en) * 2005-06-30 2005-08-03 Glaxo Group Ltd Novel compounds
DK1959955T3 (da) 2005-12-05 2011-02-07 Pfizer Prod Inc Fremgangsmåde til behandling af abnorm cellevækst
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KR101777971B1 (ko) * 2016-07-05 2017-09-12 제일약품주식회사 이미다조[1,2-a]피리딘 유도체, 이의 제조방법 및 이의 용도
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Also Published As

Publication number Publication date
EP1073656A1 (en) 2001-02-07
SK14922000A3 (sk) 2001-06-11
CN1307577A (zh) 2001-08-08
DK1073656T3 (da) 2006-01-16
CA2329921A1 (en) 1999-11-04
SE9801526D0 (sv) 1998-04-29
PL343801A1 (en) 2001-09-10
SI1073656T1 (sl) 2006-02-28
WO1999055706A1 (en) 1999-11-04
DE69927803T2 (de) 2006-07-06
CA2329922C (en) 2006-04-11
IL139297A (en) 2007-06-03
NZ507638A (en) 2003-10-31
EP1073657B1 (en) 2005-12-07
KR20050121760A (ko) 2005-12-27
NO20005450L (no) 2000-12-22
WO1999055706A9 (en) 2000-03-16
US6313137B1 (en) 2001-11-06
EP1491542A2 (en) 2004-12-29
CZ292567B6 (cs) 2003-10-15
AU769190B2 (en) 2004-01-22
TW490466B (en) 2002-06-11
KR20010043133A (ko) 2001-05-25
KR20010043134A (ko) 2001-05-25
IS5683A (is) 2000-10-25
TR200003149T2 (tr) 2001-03-21
MY121379A (en) 2006-01-28
TR200102728T2 (tr) 2002-06-21
WO1999055705A1 (en) 1999-11-04
JP2002513025A (ja) 2002-05-08
HK1036981A1 (en) 2002-01-25
EP1491543B1 (en) 2007-09-05
MY121389A (en) 2006-01-28
DE69937077D1 (de) 2007-10-18
JP2002513024A (ja) 2002-05-08
UA66846C2 (uk) 2004-06-15
NO317262B1 (no) 2004-09-27
EE200000626A (et) 2002-04-15
IL139200A (en) 2010-04-29
JP3692034B2 (ja) 2005-09-07
HUP0102425A2 (hu) 2001-11-28
CN1174980C (zh) 2004-11-10
NZ507639A (en) 2004-01-30
ZA200005797B (en) 2002-01-18
US6313136B1 (en) 2001-11-06
ZA200005796B (en) 2002-01-18
IS5684A (is) 2000-10-25
EP1491542A3 (en) 2005-01-05
HK1036984A1 (en) 2002-01-25
KR100595805B1 (ko) 2006-07-03
NO20005450D0 (no) 2000-10-27
AU769108B2 (en) 2004-01-15
IL139200A0 (en) 2001-11-25
NO20005451D0 (no) 2000-10-27
DK1073657T3 (da) 2006-03-13
NO20005451L (no) 2000-12-27
HUP0102313A2 (hu) 2001-12-28
SK14912000A3 (sk) 2001-06-11
AR015769A1 (es) 2001-05-16
CZ293977B6 (cs) 2004-09-15
AU4300699A (en) 1999-11-16
JP3883383B2 (ja) 2007-02-21
ID26819A (id) 2001-02-15
BR9909995A (pt) 2000-12-26
CA2329922A1 (en) 1999-11-04
ES2249913T3 (es) 2006-04-01
KR100650472B1 (ko) 2006-11-28
CZ20003981A3 (cs) 2001-03-14
CN1306533A (zh) 2001-08-01
RU2235725C2 (ru) 2004-09-10
DE69928792T2 (de) 2006-07-20
SA99200064B1 (ar) 2006-10-11
EE04676B1 (et) 2006-08-15
ATE372339T1 (de) 2007-09-15
SA99200065B1 (ar) 2006-11-07
DE69937076T2 (de) 2008-05-29
HK1033457A1 (en) 2001-08-31
ES2252975T3 (es) 2006-05-16
DE69937077T2 (de) 2008-05-29
HUP0102425A3 (en) 2002-12-28
BR9909995B1 (pt) 2010-07-13
BR9909996B1 (pt) 2010-08-24
EE04916B1 (et) 2007-10-15
HK1033317A1 (en) 2001-08-24
EP1491543A1 (en) 2004-12-29
TR200003176T2 (tr) 2001-03-21
NO318203B1 (no) 2005-02-14
DE69937076D1 (de) 2007-10-18
AR015768A1 (es) 2001-05-16
KR100595806B1 (ko) 2006-07-03
UA67769C2 (uk) 2004-07-15
PL343797A1 (en) 2001-09-10
TR200102612T2 (tr) 2002-06-21
ATE307130T1 (de) 2005-11-15
CZ20003982A3 (cs) 2001-02-14
TWI250159B (en) 2006-03-01
HK1071139A1 (en) 2005-07-08
EE200000664A (et) 2002-04-15
EP1491542B1 (en) 2007-09-05
CN1165535C (zh) 2004-09-08
DE69928792D1 (de) 2006-01-12
BR9909996A (pt) 2000-12-26
ATE372340T1 (de) 2007-09-15
IL139297A0 (en) 2001-11-25
PL195000B1 (pl) 2007-07-31
ATE312101T1 (de) 2005-12-15
EP1073656B1 (en) 2005-10-19
ID27530A (id) 2001-04-12
RU2238271C2 (ru) 2004-10-20
EP1073657A1 (en) 2001-02-07
DE69927803D1 (de) 2006-03-02
SA99200065A (ar) 2005-12-03
HUP0102313A3 (en) 2002-10-28
AU4300799A (en) 1999-11-16

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Effective date: 20100423