UA66846C2 - Похідні імідазопіридину, які інгібують секрецію шлункової кислоти - Google Patents

Похідні імідазопіридину, які інгібують секрецію шлункової кислоти

Info

Publication number
UA66846C2
UA66846C2 UA2000106034A UA00106034A UA66846C2 UA 66846 C2 UA66846 C2 UA 66846C2 UA 2000106034 A UA2000106034 A UA 2000106034A UA 00106034 A UA00106034 A UA 00106034A UA 66846 C2 UA66846 C2 UA 66846C2
Authority
UA
Ukraine
Prior art keywords
gastric acid
acid secretion
derivatyives
inhibiting
imidazo pyridine
Prior art date
Application number
UA2000106034A
Other languages
English (en)
Russian (ru)
Inventor
Косрат Амін
Мікаель Дальстрем
Петер Норберґ
Інґемар Старке
Ингемар Старке
Original Assignee
Астразенека Аб
Астра АБ
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Астразенека Аб, Астра АБ filed Critical Астразенека Аб
Publication of UA66846C2 publication Critical patent/UA66846C2/uk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Винахід стосується похідних імідазопіридину формули I, в яких феніл є заміщеним, а імідазопіридинова група заміщена карбоксамідною в 6-ій позиції, що інгібують екзогенно чи ендогенно стимульовану секрецію шлункової кислоти і які можна використовувати при попередженні та лікуванні шлунково-кишкових запальних захворювань. (І)
UA2000106034A 1998-04-29 1999-04-23 Похідні імідазопіридину, які інгібують секрецію шлункової кислоти UA66846C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9801526A SE9801526D0 (sv) 1998-04-29 1998-04-29 New compounds
PCT/SE1999/000663 WO1999055706A1 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion

Publications (1)

Publication Number Publication Date
UA66846C2 true UA66846C2 (uk) 2004-06-15

Family

ID=20411154

Family Applications (2)

Application Number Title Priority Date Filing Date
UA2000106033A UA67769C2 (uk) 1998-04-29 1999-04-23 Похідні імідазопіридину, які інгібують секрецію шлункової кислоти
UA2000106034A UA66846C2 (uk) 1998-04-29 1999-04-23 Похідні імідазопіридину, які інгібують секрецію шлункової кислоти

Family Applications Before (1)

Application Number Title Priority Date Filing Date
UA2000106033A UA67769C2 (uk) 1998-04-29 1999-04-23 Похідні імідазопіридину, які інгібують секрецію шлункової кислоти

Country Status (34)

Country Link
US (2) US6313137B1 (uk)
EP (4) EP1491543B1 (uk)
JP (2) JP3692034B2 (uk)
KR (3) KR100595806B1 (uk)
CN (2) CN1165535C (uk)
AR (2) AR015768A1 (uk)
AT (4) ATE372340T1 (uk)
AU (2) AU769190B2 (uk)
BR (2) BR9909996B1 (uk)
CA (2) CA2329922C (uk)
CZ (2) CZ292567B6 (uk)
DE (4) DE69937077T2 (uk)
DK (2) DK1073656T3 (uk)
EE (2) EE04916B1 (uk)
ES (2) ES2252975T3 (uk)
HK (5) HK1033457A1 (uk)
HU (2) HUP0102313A3 (uk)
ID (2) ID27530A (uk)
IL (4) IL139200A0 (uk)
IS (2) IS5683A (uk)
MY (2) MY121379A (uk)
NO (2) NO318203B1 (uk)
NZ (2) NZ507639A (uk)
PL (2) PL343797A1 (uk)
RU (2) RU2235725C2 (uk)
SA (2) SA99200065B1 (uk)
SE (1) SE9801526D0 (uk)
SI (1) SI1073656T1 (uk)
SK (2) SK14912000A3 (uk)
TR (4) TR200003176T2 (uk)
TW (2) TWI250159B (uk)
UA (2) UA67769C2 (uk)
WO (2) WO1999055706A1 (uk)
ZA (2) ZA200005796B (uk)

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US6489346B1 (en) 1996-01-04 2002-12-03 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
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UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
SE0100297D0 (sv) * 2001-02-01 2001-02-01 Astrazeneca Ab New compounds
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ME00524B (me) 2003-03-10 2011-10-10 Astrazeneca Ab Novi postupak za dobijanje roflumilasta
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SE0301904D0 (sv) * 2003-06-26 2003-06-26 Astrazeneca Ab Novel imidazopyridine compound II with therapeutic effect
SE0301903D0 (sv) * 2003-06-26 2003-06-26 Astrazeneca Ab Novel imidazopyridine compound III with therapeutic effect
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US8993599B2 (en) 2003-07-18 2015-03-31 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
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SE0303451D0 (sv) * 2003-12-18 2003-12-18 Astrazeneca Ab New compounds
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KR20190057569A (ko) 2017-11-20 2019-05-29 제일약품주식회사 7-아미노-1h-인돌-5-카르복사미드 유도체 및 이의 용도
CN111683976B (zh) 2018-02-05 2022-11-18 生物辐射实验室股份有限公司 具有阴离子交换-疏水混合模式配体的色谱树脂
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RU2732297C2 (ru) * 2018-11-14 2020-09-15 Общество с ограниченной ответственностью "Гурус БиоФарм" Производные нестероидных противовоспалительных средств
MX2022005305A (es) 2019-11-04 2022-08-16 Cinclus Pharma Holding AB Formulacion oral de x842.
MX2024005292A (es) 2021-11-05 2024-05-17 Cinclus Pharma Holding Ab Publ Polimorfos de la sal de clorhidrato de glurato de linaprazan.
KR20240093547A (ko) 2021-11-05 2024-06-24 싱클루스 파마 홀딩 에이비 (피유비엘) 리나프라잔 글루레이트의 메실레이트 염의 다형체
KR102496869B1 (ko) * 2022-07-29 2023-02-07 제일약품주식회사 이미다조[1,2-a]피리딘 화합물의 신규 염, 이의 결정형 및 제조방법
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Also Published As

Publication number Publication date
KR20010043133A (ko) 2001-05-25
HK1036981A1 (en) 2002-01-25
EE04676B1 (et) 2006-08-15
AR015768A1 (es) 2001-05-16
ATE312101T1 (de) 2005-12-15
EP1491543A1 (en) 2004-12-29
DE69927803D1 (de) 2006-03-02
SK14912000A3 (sk) 2001-06-11
NO20005450D0 (no) 2000-10-27
EP1073656A1 (en) 2001-02-07
BR9909996B1 (pt) 2010-08-24
NO20005451L (no) 2000-12-27
UA67769C2 (uk) 2004-07-15
NO20005451D0 (no) 2000-10-27
PL195000B1 (pl) 2007-07-31
IL139200A0 (en) 2001-11-25
KR100595806B1 (ko) 2006-07-03
ES2252975T3 (es) 2006-05-16
ZA200005796B (en) 2002-01-18
NZ507638A (en) 2003-10-31
EP1491542A2 (en) 2004-12-29
EP1073657A1 (en) 2001-02-07
TR200102612T2 (tr) 2002-06-21
CZ292567B6 (cs) 2003-10-15
NZ507639A (en) 2004-01-30
NO20005450L (no) 2000-12-22
AR015769A1 (es) 2001-05-16
HUP0102425A3 (en) 2002-12-28
BR9909995B1 (pt) 2010-07-13
DE69937076D1 (de) 2007-10-18
WO1999055706A9 (en) 2000-03-16
CN1307577A (zh) 2001-08-08
US6313136B1 (en) 2001-11-06
KR100595805B1 (ko) 2006-07-03
RU2235725C2 (ru) 2004-09-10
EE200000664A (et) 2002-04-15
EP1491542B1 (en) 2007-09-05
IL139297A0 (en) 2001-11-25
SK14922000A3 (sk) 2001-06-11
JP2002513024A (ja) 2002-05-08
US6313137B1 (en) 2001-11-06
IL139297A (en) 2007-06-03
CN1174980C (zh) 2004-11-10
ATE307130T1 (de) 2005-11-15
SK285768B6 (sk) 2007-07-06
HK1033457A1 (en) 2001-08-31
JP2002513025A (ja) 2002-05-08
NO318203B1 (no) 2005-02-14
AU769190B2 (en) 2004-01-22
KR100650472B1 (ko) 2006-11-28
CA2329921A1 (en) 1999-11-04
DK1073657T3 (da) 2006-03-13
SA99200065A (ar) 2005-12-03
HK1036984A1 (en) 2002-01-25
BR9909995A (pt) 2000-12-26
SI1073656T1 (sl) 2006-02-28
WO1999055706A1 (en) 1999-11-04
ATE372339T1 (de) 2007-09-15
WO1999055705A1 (en) 1999-11-04
DE69937076T2 (de) 2008-05-29
KR20050121760A (ko) 2005-12-27
JP3692034B2 (ja) 2005-09-07
PL343797A1 (en) 2001-09-10
ZA200005797B (en) 2002-01-18
TR200003176T2 (tr) 2001-03-21
PL343801A1 (en) 2001-09-10
SE9801526D0 (sv) 1998-04-29
ATE372340T1 (de) 2007-09-15
AU4300699A (en) 1999-11-16
BR9909996A (pt) 2000-12-26
SA99200065B1 (ar) 2006-11-07
HUP0102313A2 (hu) 2001-12-28
TW490466B (en) 2002-06-11
IS5684A (is) 2000-10-25
CZ20003982A3 (cs) 2001-02-14
MY121389A (en) 2006-01-28
ID26819A (id) 2001-02-15
IL139200A (en) 2010-04-29
DE69928792D1 (de) 2006-01-12
AU769108B2 (en) 2004-01-15
TR200003149T2 (tr) 2001-03-21
MY121379A (en) 2006-01-28
DE69928792T2 (de) 2006-07-20
EP1491543B1 (en) 2007-09-05
SA99200064B1 (ar) 2006-10-11
DK1073656T3 (da) 2006-01-16
DE69937077D1 (de) 2007-10-18
TWI250159B (en) 2006-03-01
EE200000626A (et) 2002-04-15
CN1165535C (zh) 2004-09-08
EP1073657B1 (en) 2005-12-07
CZ20003981A3 (cs) 2001-03-14
DE69927803T2 (de) 2006-07-06
EE04916B1 (et) 2007-10-15
CN1306533A (zh) 2001-08-01
CZ293977B6 (cs) 2004-09-15
TR200102728T2 (tr) 2002-06-21
AU4300799A (en) 1999-11-16
NO317262B1 (no) 2004-09-27
CA2329922A1 (en) 1999-11-04
HUP0102425A2 (hu) 2001-11-28
JP3883383B2 (ja) 2007-02-21
EP1073656B1 (en) 2005-10-19
ID27530A (id) 2001-04-12
RU2238271C2 (ru) 2004-10-20
ES2249913T3 (es) 2006-04-01
CA2329922C (en) 2006-04-11
HK1071139A1 (en) 2005-07-08
IS5683A (is) 2000-10-25
HUP0102313A3 (en) 2002-10-28
EP1491542A3 (en) 2005-01-05
HK1033317A1 (en) 2001-08-24
DE69937077T2 (de) 2008-05-29
KR20010043134A (ko) 2001-05-25

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