SK280295B6 - Farmaceutický prostriedok s riadeným uvoľňovaním o - Google Patents
Farmaceutický prostriedok s riadeným uvoľňovaním o Download PDFInfo
- Publication number
- SK280295B6 SK280295B6 SK922-93A SK92293A SK280295B6 SK 280295 B6 SK280295 B6 SK 280295B6 SK 92293 A SK92293 A SK 92293A SK 280295 B6 SK280295 B6 SK 280295B6
- Authority
- SK
- Slovakia
- Prior art keywords
- oxycodone
- oxy
- hours
- tablets
- controlled release
- Prior art date
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- BRUQQQPBMZOVGD-XFKAJCMBSA-N Oxycodone Chemical compound O=C([C@@H]1O2)CC[C@@]3(O)[C@H]4CC5=CC=C(OC)C2=C5[C@@]13CCN4C BRUQQQPBMZOVGD-XFKAJCMBSA-N 0.000 title claims abstract description 147
- 229960002085 oxycodone Drugs 0.000 title claims abstract description 130
- 239000008194 pharmaceutical composition Substances 0.000 title claims abstract description 35
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- QCQCHGYLTSGIGX-GHXANHINSA-N 4-[[(3ar,5ar,5br,7ar,9s,11ar,11br,13as)-5a,5b,8,8,11a-pentamethyl-3a-[(5-methylpyridine-3-carbonyl)amino]-2-oxo-1-propan-2-yl-4,5,6,7,7a,9,10,11,11b,12,13,13a-dodecahydro-3h-cyclopenta[a]chrysen-9-yl]oxy]-2,2-dimethyl-4-oxobutanoic acid Chemical compound N([C@@]12CC[C@@]3(C)[C@]4(C)CC[C@H]5C(C)(C)[C@@H](OC(=O)CC(C)(C)C(O)=O)CC[C@]5(C)[C@H]4CC[C@@H]3C1=C(C(C2)=O)C(C)C)C(=O)C1=CN=CC(C)=C1 QCQCHGYLTSGIGX-GHXANHINSA-N 0.000 claims description 2
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5015—Organic compounds, e.g. fats, sugars
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Emergency Medicine (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
- Measuring Fluid Pressure (AREA)
- Polyethers (AREA)
- Saccharide Compounds (AREA)
- Polysaccharides And Polysaccharide Derivatives (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Plant Substances (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/800,549 US5266331A (en) | 1991-11-27 | 1991-11-27 | Controlled release oxycodone compositions |
| PCT/US1992/010146 WO1993010765A1 (en) | 1991-11-27 | 1992-11-25 | Controlled release oxycodone compositions |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| SK92293A3 SK92293A3 (en) | 1994-04-06 |
| SK280295B6 true SK280295B6 (sk) | 1999-11-08 |
Family
ID=25178688
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK922-93A SK280295B6 (sk) | 1991-11-27 | 1992-11-25 | Farmaceutický prostriedok s riadeným uvoľňovaním o |
Country Status (31)
| Country | Link |
|---|---|
| US (13) | US5266331A (pt) |
| EP (15) | EP0576643B1 (pt) |
| JP (2) | JP3375960B2 (pt) |
| KR (1) | KR100280973B1 (pt) |
| CN (2) | CN1245958C (pt) |
| AT (9) | ATE261726T1 (pt) |
| AU (1) | AU657027B2 (pt) |
| BG (1) | BG61753B1 (pt) |
| BR (1) | BR9205498A (pt) |
| CA (1) | CA2098738C (pt) |
| CZ (4) | CZ286913B6 (pt) |
| DE (10) | DE69232837T3 (pt) |
| DK (10) | DK1327446T4 (pt) |
| ES (9) | ES2096781T3 (pt) |
| FI (5) | FI113152B (pt) |
| GR (1) | GR3022273T3 (pt) |
| HK (6) | HK1068004A1 (pt) |
| HU (10) | HU227517B1 (pt) |
| IL (1) | IL103909A (pt) |
| MX (1) | MX9302968A (pt) |
| NO (6) | NO307028B3 (pt) |
| PH (1) | PH31679A (pt) |
| PL (2) | PL172236B1 (pt) |
| PT (8) | PT722730E (pt) |
| RO (1) | RO115112B1 (pt) |
| RS (3) | RS50056B (pt) |
| RU (1) | RU2122411C1 (pt) |
| SK (1) | SK280295B6 (pt) |
| WO (1) | WO1993010765A1 (pt) |
| YU (1) | YU49495B (pt) |
| ZA (1) | ZA929227B (pt) |
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| PC4A | Assignment and transfer of rights |
Owner name: MUNDIPHARMA MEDICAL GMBH, BASEL, CH Free format text: FORMER OWNER: PURDUE PHARMA L.P., STAMFORD, CONNECTICUT, US Effective date: 20091119 Owner name: PURDUE PHARMA L.P., STAMFORD, CONNECTICUT, US Free format text: FORMER OWNER: EURO-CELTIQUE, S. A., LUXEMBOURG, LU Effective date: 20091119 |
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| MK4A | Patent expired |
Expiry date: 20121125 |