SI9500293A - Synthesis of 3-/4-(2-aminoethoxy)-benzoyl/-2- aryl-6-hydroxybenzo/b/ thyophenes - Google Patents

Synthesis of 3-/4-(2-aminoethoxy)-benzoyl/-2- aryl-6-hydroxybenzo/b/ thyophenes Download PDF

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Publication number
SI9500293A
SI9500293A SI9500293A SI9500293A SI9500293A SI 9500293 A SI9500293 A SI 9500293A SI 9500293 A SI9500293 A SI 9500293A SI 9500293 A SI9500293 A SI 9500293A SI 9500293 A SI9500293 A SI 9500293A
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SI
Slovenia
Prior art keywords
group
formula
crystalline
chlorine
benzoyl
Prior art date
Application number
SI9500293A
Other languages
English (en)
Slovenian (sl)
Inventor
Smith Elizabeth Labell
Douglas Wayne Luke
Mcneill John Mcgill Iii
Scot Randal Miller
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26976194&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI9500293(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US08/308,325 external-priority patent/US5629425A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of SI9500293A publication Critical patent/SI9500293A/sl

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56—Radicals substituted by oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
SI9500293A 1994-09-19 1995-09-18 Synthesis of 3-/4-(2-aminoethoxy)-benzoyl/-2- aryl-6-hydroxybenzo/b/ thyophenes SI9500293A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/308,325 US5629425A (en) 1994-09-19 1994-09-19 Haloalkyl hemisolvates of 6-hydroxy-2-(4-hydroxyphenyl)-3-[4-piperidinoethoxy)-benzoyl]benzo[b]thiophene
US42791495A 1995-04-26 1995-04-26

Publications (1)

Publication Number Publication Date
SI9500293A true SI9500293A (en) 1996-06-30

Family

ID=26976194

Family Applications (2)

Application Number Title Priority Date Filing Date
SI9500292A SI9500292A (en) 1994-09-19 1995-09-18 Novel pharmaceutical product on bases of new non-solvated crystalline form of a 2-aryl-6-hydroxy-3-/4-(2-aminoethoxy)benzoyl/ benzo /b/ thiophene
SI9500293A SI9500293A (en) 1994-09-19 1995-09-18 Synthesis of 3-/4-(2-aminoethoxy)-benzoyl/-2- aryl-6-hydroxybenzo/b/ thyophenes

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SI9500292A SI9500292A (en) 1994-09-19 1995-09-18 Novel pharmaceutical product on bases of new non-solvated crystalline form of a 2-aryl-6-hydroxy-3-/4-(2-aminoethoxy)benzoyl/ benzo /b/ thiophene

Country Status (51)

Country Link
US (4) US6472531B1 (fi)
JP (2) JP2860071B2 (fi)
KR (2) KR100367376B1 (fi)
CN (2) CN1075069C (fi)
AP (1) AP754A (fi)
AT (2) AT502957A1 (fi)
AU (3) AU691955B2 (fi)
BE (2) BE1009625A3 (fi)
BG (1) BG62793B1 (fi)
BR (2) BR9504059A (fi)
CA (2) CA2158400C (fi)
CH (3) CH691478A5 (fi)
CO (2) CO4410191A1 (fi)
CZ (2) CZ292007B6 (fi)
DE (3) DE19549755B4 (fi)
DK (4) DK175897B1 (fi)
EE (1) EE03386B1 (fi)
EG (1) EG23763A (fi)
ES (2) ES2129293B1 (fi)
FI (2) FI112226B (fi)
FR (2) FR2724655B1 (fi)
GB (2) GB2293602B (fi)
GE (1) GEP19991821B (fi)
GR (2) GR1002709B (fi)
HK (1) HK1019009A1 (fi)
HR (2) HRP950482B1 (fi)
HU (2) HU225417B1 (fi)
IE (2) IE80883B1 (fi)
IL (3) IL115314A (fi)
IS (1) IS1788B (fi)
IT (2) IT1277601B1 (fi)
LU (2) LU88660A1 (fi)
LV (2) LV11177B (fi)
MY (1) MY116371A (fi)
NL (2) NL1001194C2 (fi)
NO (2) NO308107B1 (fi)
NZ (2) NZ280028A (fi)
OA (1) OA10406A (fi)
PE (2) PE14796A1 (fi)
PL (2) PL187686B1 (fi)
PT (2) PT101771B (fi)
RO (2) RO115259B1 (fi)
RS (2) RS49513B (fi)
SE (2) SE520721C2 (fi)
SI (2) SI9500292A (fi)
SK (1) SK283502B6 (fi)
TR (1) TR199501136A2 (fi)
TW (1) TW412534B (fi)
UA (2) UA42716C2 (fi)
UY (1) UY24040A1 (fi)
WO (1) WO1996009045A1 (fi)

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HU227683B1 (en) 2011-11-28
NZ280027A (en) 1997-05-26
BG62793B1 (bg) 2000-08-31
AU3718695A (en) 1996-04-09
CA2158399C (en) 2001-03-20
RO115260B1 (ro) 1999-12-30
US5731327A (en) 1998-03-24
ES2109882B1 (es) 1998-08-16
HRP950483B1 (en) 2003-02-28
IS1788B (is) 2001-11-28
CO4410191A1 (es) 1997-01-09
GB2293602A (en) 1996-04-03
EG23763A (en) 2007-08-08
FR2724655A1 (fr) 1996-03-22
AP754A (en) 1999-07-22
AU692907B2 (en) 1998-06-18
CZ240395A3 (en) 1996-04-17
FR2732020A1 (fr) 1996-09-27
LV11177A (lv) 1996-04-20
IE950721A1 (en) 1996-03-20
US6472531B1 (en) 2002-10-29
US6399778B1 (en) 2002-06-04
HU225417B1 (en) 2006-11-28
FI954403A (fi) 1996-03-20
FR2732020B1 (fr) 1997-11-14
FI954402A (fi) 1996-03-20
UA44240C2 (uk) 2002-02-15
DE19534744A1 (de) 1996-03-21
CN1075069C (zh) 2001-11-21
HUT74178A (en) 1996-11-28
NL1001194A1 (nl) 1996-03-19
DK175887B1 (da) 2005-05-23
RS49578B (sr) 2007-04-10
IL115315A (en) 1999-09-22
GR1002709B (el) 1997-06-04
ES2129293A1 (es) 1999-06-01
NO953657D0 (no) 1995-09-15
IL115314A0 (en) 1996-05-14
PT101771A (pt) 1996-04-30
SE9503213L (sv) 1996-03-20
NL1001194C2 (nl) 1997-04-04
BE1009625A3 (fr) 1997-06-03
GB9519028D0 (en) 1995-11-15
HRP950482B1 (en) 2007-04-30
AU691955B2 (en) 1998-05-28
JPH08193081A (ja) 1996-07-30
PL310517A1 (en) 1996-04-01
CZ240295A3 (en) 1996-04-17
YU61495A (sh) 1998-05-15
IS4446A (is) 1997-03-18
PE14796A1 (es) 1996-05-19
SK23397A3 (en) 1997-08-06
HUT75033A (en) 1997-03-28
ITMI951935A0 (it) 1995-09-15
CZ290343B6 (cs) 2002-07-17
EE9700055A (et) 1997-08-15
PT101770B (pt) 1997-04-30
LV11178A (lv) 1996-04-20
FI121424B (fi) 2010-11-15
ITMI951936A0 (it) 1995-09-15
LU88660A1 (fr) 1996-07-15
PL187686B1 (pl) 2004-09-30
CA2158400C (en) 2006-10-24
CH691478A5 (de) 2001-07-31
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