AU2002230409A1 - Process for preparing 3-aryl-benzo(b)thiophenes - Google Patents
Process for preparing 3-aryl-benzo(b)thiophenesInfo
- Publication number
- AU2002230409A1 AU2002230409A1 AU2002230409A AU3040902A AU2002230409A1 AU 2002230409 A1 AU2002230409 A1 AU 2002230409A1 AU 2002230409 A AU2002230409 A AU 2002230409A AU 3040902 A AU3040902 A AU 3040902A AU 2002230409 A1 AU2002230409 A1 AU 2002230409A1
- Authority
- AU
- Australia
- Prior art keywords
- thiophenes
- benzo
- aryl
- preparing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/64—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/56—Radicals substituted by oxygen atoms
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US25321200P | 2000-11-27 | 2000-11-27 | |
US60/253,212 | 2000-11-27 | ||
PCT/US2001/042940 WO2002042289A2 (en) | 2000-11-27 | 2001-11-14 | Process for preparing 3-aryl-benzo[b]thiophenes |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2002230409A1 true AU2002230409A1 (en) | 2002-06-03 |
Family
ID=22959343
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2002230409A Abandoned AU2002230409A1 (en) | 2000-11-27 | 2001-11-14 | Process for preparing 3-aryl-benzo(b)thiophenes |
Country Status (3)
Country | Link |
---|---|
US (1) | US6921827B2 (en) |
AU (1) | AU2002230409A1 (en) |
WO (1) | WO2002042289A2 (en) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1826205A1 (en) | 2002-09-30 | 2007-08-29 | A/S GEA Farmaceutisk Fabrik | Novel raloxifene succinic acid addition salts and/or solvates thereof, and pharmaceutical compositions comprising these |
AU2002953533A0 (en) | 2002-12-24 | 2003-01-16 | Arthron Limited | Fc receptor modulating compounds and compositions |
Family Cites Families (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4133814A (en) * | 1975-10-28 | 1979-01-09 | Eli Lilly And Company | 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents |
AU509682B2 (en) * | 1975-10-28 | 1980-05-22 | Eli Lilly And Company | 2-Aroyl-3-Phenylbenzothiophene Derivatives |
US4380635A (en) * | 1981-04-03 | 1983-04-19 | Eli Lilly And Company | Synthesis of acylated benzothiophenes |
US4358593A (en) * | 1981-04-03 | 1982-11-09 | Eli Lilly And Company | Process for preparing 3-(4-aminoethoxybenzoyl)benzo[b]thiophenes |
US4418068A (en) * | 1981-04-03 | 1983-11-29 | Eli Lilly And Company | Antiestrogenic and antiandrugenic benzothiophenes |
US5523416A (en) * | 1994-07-22 | 1996-06-04 | Eli Lilly And Company | Process for preparing 3-(4-aminoethoxy-benzoyl) benzo (B)-thiophenes |
US5629425A (en) * | 1994-09-19 | 1997-05-13 | Eli Lilly And Company | Haloalkyl hemisolvates of 6-hydroxy-2-(4-hydroxyphenyl)-3-[4-piperidinoethoxy)-benzoyl]benzo[b]thiophene |
CO4410191A1 (en) * | 1994-09-19 | 1997-01-09 | Lilly Co Eli | SYNTHESIS OF 3- [4- (2-AMINOETOXI) BENZOIL] -2-ARYL-6- HYDROXYBENZO [b] THIOPHENES |
US5510357A (en) * | 1995-02-28 | 1996-04-23 | Eli Lilly And Company | Benzothiophene compounds as anti-estrogenic agents |
US5552401A (en) * | 1995-02-28 | 1996-09-03 | Eli Lilly And Company | 2-benzyl-3-arylbenzothiophenes |
IN183239B (en) * | 1996-09-25 | 1999-10-09 | Lilly Co Eli | |
ZA9710262B (en) * | 1996-11-19 | 1999-05-13 | Lilly Co Eli | Process for the synthesis of benzothiophenes |
RU2186065C1 (en) * | 1998-03-31 | 2002-07-27 | Сионоги Энд Ко., Лтд. | Method of synthesis of derivatives of 5-hydroxy-benzo[b]thiophene-3- carboxylic acid (variants) and thiophenic acid derivatives |
DE19913349A1 (en) * | 1999-03-24 | 2000-09-28 | Clariant Gmbh | Use of benzothiophene derivatives as components of liquid crystal mixtures, especially for use in ferroelectric switching and display devices |
WO2001009115A2 (en) | 1999-07-29 | 2001-02-08 | Eli Lilly And Company | A NOVEL CRYSTALLINE FORM OF 6-HYDROXY-3- (4-[2-(PIPERIDIN-1- YL)ETHOXY] PHENOXY)-2- (4-METHOXYPHENYL) BENZO[b]THIOPHENE HYDROCHLORIDE |
EP1204656A2 (en) | 1999-07-29 | 2002-05-15 | Eli Lilly And Company | A crystalline form of 6-hydroxy-3-(4-[2-(piperidin-1-yl) ethoxy] phenoxy)-2-(4-methoxyphenyl) benzo[b]thiophene hydrochloride |
ES2258431T3 (en) * | 1999-08-02 | 2006-09-01 | F. Hoffmann-La Roche Ag | PROCESS FOR THE PREPARATION OF BENZOTIOFEN DERIVATIVES. |
AU1033101A (en) * | 1999-10-21 | 2001-04-30 | Rhodia Chimie | Method for preparing a benzofuran or benzothiophene compound |
WO2002042261A2 (en) | 2000-11-27 | 2002-05-30 | Eli Lilly And Company | PROCESS FOR PREPARING α-(3-ARYLTHIO)-ACETOPHENONES |
US6388105B1 (en) * | 2001-09-27 | 2002-05-14 | Allergan Sales, Inc. | Benzofuran, indole or benzothiophene 2,4-pentadienoic acid derivatives having selective activity for retinoid X (RXR) receptors |
-
2001
- 2001-11-14 AU AU2002230409A patent/AU2002230409A1/en not_active Abandoned
- 2001-11-14 US US10/415,569 patent/US6921827B2/en not_active Expired - Fee Related
- 2001-11-14 WO PCT/US2001/042940 patent/WO2002042289A2/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO2002042289A8 (en) | 2004-02-12 |
WO2002042289A3 (en) | 2002-09-06 |
WO2002042289A2 (en) | 2002-05-30 |
US6921827B2 (en) | 2005-07-26 |
US20040132775A1 (en) | 2004-07-08 |
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