NO20055591L - Antivirale fosfonatanaloger - Google Patents
Antivirale fosfonatanalogerInfo
- Publication number
- NO20055591L NO20055591L NO20055591A NO20055591A NO20055591L NO 20055591 L NO20055591 L NO 20055591L NO 20055591 A NO20055591 A NO 20055591A NO 20055591 A NO20055591 A NO 20055591A NO 20055591 L NO20055591 L NO 20055591L
- Authority
- NO
- Norway
- Prior art keywords
- compounds
- phosphonate analogues
- antiviral phosphonate
- antiviral
- analogues
- Prior art date
Links
- 230000000840 anti-viral effect Effects 0.000 title abstract 2
- ABLZXFCXXLZCGV-UHFFFAOYSA-N Phosphorous acid Chemical class OP(O)=O ABLZXFCXXLZCGV-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 4
- OAICVXFJPJFONN-UHFFFAOYSA-N Phosphorus Chemical group [P] OAICVXFJPJFONN-UHFFFAOYSA-N 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 229910052698 phosphorus Inorganic materials 0.000 abstract 1
- 239000011574 phosphorus Substances 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
Classifications
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- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
- C07F9/65616—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings containing the ring system having three or more than three double bonds between ring members or between ring members and non-ring members, e.g. purine or analogs
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- A61K31/662—Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
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- A61K31/7068—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
- A61K31/7072—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid having two oxo groups directly attached to the pyrimidine ring, e.g. uridine, uridylic acid, thymidine, zidovudine
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Abstract
Oppfinnelsen angår fosforsubstituerte forbindelser med antiviral aktivitet, preparater som inneholder slike forbindelser og terapeutiske fremgangsmåter som innbefatter administrasjon av slike forbindelser, samt fremgangsmåter og mellomprodukter som er anvendelige ved fremstilling av slike forbindelser.
Applications Claiming Priority (92)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US46532203P | 2003-04-25 | 2003-04-25 | |
US46560803P | 2003-04-25 | 2003-04-25 | |
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- 2004-04-26 DK DK04750807.2T patent/DK1628685T3/da active
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- 2004-04-26 NZ NZ542342A patent/NZ542342A/en unknown
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2005
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2006
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2008
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-
2013
- 2013-03-21 US US13/848,593 patent/US8871785B2/en not_active Expired - Lifetime
-
2014
- 2014-06-19 US US14/309,790 patent/US9139604B2/en not_active Expired - Lifetime
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NO342571B1 (no) * | 2004-07-27 | 2018-06-18 | Gilead Sciences Inc | Fosfonatanaloger til HIV-inhibitorsammensetninger |
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