MY137619A - 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions - Google Patents

8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

Info

Publication number
MY137619A
MY137619A MYPI20033150A MYPI20033150A MY137619A MY 137619 A MY137619 A MY 137619A MY PI20033150 A MYPI20033150 A MY PI20033150A MY PI20033150 A MYPI20033150 A MY PI20033150A MY 137619 A MY137619 A MY 137619A
Authority
MY
Malaysia
Prior art keywords
xanthines
piperidin
amino
preparation
pharmaceutical compositions
Prior art date
Application number
MYPI20033150A
Other languages
English (en)
Inventor
Frank Dr Himmelsbach
Matthias Dr Eckhardt
Elke Dr Langkopf
Michael Dr Mark
Roland Dr Maier
Ralf R H Dr Lotz
Mohammad Dr Tadayyon
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31947613&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MY137619(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE10238243A external-priority patent/DE10238243A1/de
Priority claimed from DE10312353A external-priority patent/DE10312353A1/de
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of MY137619A publication Critical patent/MY137619A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
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    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
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    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C07D473/12Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1, 3, and 7, e.g. caffeine

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MYPI20033150A 2002-08-21 2003-08-19 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions MY137619A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10238243A DE10238243A1 (de) 2002-08-21 2002-08-21 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
DE10312353A DE10312353A1 (de) 2003-03-20 2003-03-20 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel

Publications (1)

Publication Number Publication Date
MY137619A true MY137619A (en) 2009-02-27

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ID=31947613

Family Applications (2)

Application Number Title Priority Date Filing Date
MYPI20033150A MY137619A (en) 2002-08-21 2003-08-19 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
MYPI20083230A MY165643A (en) 2002-08-21 2003-08-19 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

Family Applications After (1)

Application Number Title Priority Date Filing Date
MYPI20083230A MY165643A (en) 2002-08-21 2003-08-19 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

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JP (6) JP4233524B2 (bs)
KR (2) KR101111101B1 (bs)
CN (4) CN107674077A (bs)
AR (3) AR041025A1 (bs)
AT (1) ATE453644T1 (bs)
AU (2) AU2003253418B2 (bs)
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EC (2) ECSP055617A (bs)
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ES (1) ES2339112T3 (bs)
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HK (6) HK1081552A1 (bs)
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IL (1) IL166964A (bs)
IN (2) IN2015DN01133A (bs)
LU (2) LU91889I2 (bs)
ME (1) ME00396B (bs)
MX (1) MXPA05001684A (bs)
MY (2) MY137619A (bs)
NO (4) NO333970B1 (bs)
PE (1) PE20040897A1 (bs)
PL (2) PL403104A1 (bs)
PT (1) PT1532149E (bs)
RS (2) RS20120139A3 (bs)
SA (1) SA03240448B1 (bs)
SI (1) SI1532149T1 (bs)
TW (3) TWI319320B (bs)
UA (1) UA84275C2 (bs)
UY (1) UY27946A1 (bs)
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Families Citing this family (175)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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