MX364937B - Composiciones farmaceuticas de acido 3-(6-(1-(2,2-difluorobenzo [d][1,3]dioxol-5-il)ciclopropancarboxamido)-3-metilpiridin-2-il) benzoico y su administracion. - Google Patents
Composiciones farmaceuticas de acido 3-(6-(1-(2,2-difluorobenzo [d][1,3]dioxol-5-il)ciclopropancarboxamido)-3-metilpiridin-2-il) benzoico y su administracion.Info
- Publication number
- MX364937B MX364937B MX2012011656A MX2012011656A MX364937B MX 364937 B MX364937 B MX 364937B MX 2012011656 A MX2012011656 A MX 2012011656A MX 2012011656 A MX2012011656 A MX 2012011656A MX 364937 B MX364937 B MX 364937B
- Authority
- MX
- Mexico
- Prior art keywords
- cyclopropanecarboxamido
- difluorobenzo
- dioxol
- administration
- methylpyriodin
- Prior art date
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Abstract
Una composición farmacéutica que comprende el Compuesto 1, ácido (3-(6-(1-(2, 2-difluorobenzo[d] [1, 3] dioxol-5-il)ciclopropancarb oxamido)-3-metilpiridin-2-il)benzoico), y al menos un excipiente seleccionado de: un relleno, un diluyente, un disgregante, un agente tensioactivo, un aglutinante, un deslizante y un lubricante, la composición siendo adecuada para administración oral a una paciente en la necesidad de esto para tratar una enfermedad mediada por CFTR tal como Fibrosis Cística. Métodos para tratar un paciente en a necesidad de esto incluyen la administración de una formulación farmacéutica oral del Compuesto 1 al paciente.
Applications Claiming Priority (4)
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US36656210P | 2010-07-22 | 2010-07-22 | |
PCT/US2011/031519 WO2011127241A2 (en) | 2010-04-07 | 2011-04-07 | Pharmaceutical compositions of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyriodin-2-yl)benzoic acid and administration thereof |
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MX2012011656A MX2012011656A (es) | 2012-11-23 |
MX364937B true MX364937B (es) | 2019-05-15 |
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MX2012011656A MX364937B (es) | 2010-04-07 | 2011-04-07 | Composiciones farmaceuticas de acido 3-(6-(1-(2,2-difluorobenzo [d][1,3]dioxol-5-il)ciclopropancarboxamido)-3-metilpiridin-2-il) benzoico y su administracion. |
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US (8) | US8552034B2 (es) |
EP (3) | EP3150198B1 (es) |
JP (3) | JP2013523833A (es) |
CN (3) | CN106943403A (es) |
AR (1) | AR081760A1 (es) |
AU (1) | AU2011237601B2 (es) |
BR (1) | BR112012026255A2 (es) |
CA (1) | CA2795804C (es) |
CY (1) | CY1124852T1 (es) |
DK (1) | DK3150198T3 (es) |
ES (2) | ES2900353T3 (es) |
HR (1) | HRP20211752T1 (es) |
HU (1) | HUE056525T2 (es) |
IL (2) | IL222314A (es) |
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MX (1) | MX364937B (es) |
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PT (1) | PT3150198T (es) |
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RU (1) | RU2592368C2 (es) |
SI (1) | SI3150198T1 (es) |
WO (1) | WO2011127241A2 (es) |
ZA (1) | ZA201208225B (es) |
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