KR101925620B1 - Glp-1 아고니스트 및 n-(8-(2-히드록시벤조일)아미노)카프릴산의 염을 포함하는 고체 조성물 - Google Patents
Glp-1 아고니스트 및 n-(8-(2-히드록시벤조일)아미노)카프릴산의 염을 포함하는 고체 조성물 Download PDFInfo
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- KR101925620B1 KR101925620B1 KR1020137017719A KR20137017719A KR101925620B1 KR 101925620 B1 KR101925620 B1 KR 101925620B1 KR 1020137017719 A KR1020137017719 A KR 1020137017719A KR 20137017719 A KR20137017719 A KR 20137017719A KR 101925620 B1 KR101925620 B1 KR 101925620B1
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| UA116217C2 (uk) | 2012-10-09 | 2018-02-26 | Санофі | Пептидна сполука як подвійний агоніст рецепторів glp1-1 та глюкагону |
| HRP20181300T1 (hr) | 2012-12-21 | 2018-10-05 | Sanofi | Derivati eksendina-4 kao dvostruki glp1/gip- ili trostruki glp1/gip/glukagon agonisti |
| CN105101950B (zh) | 2013-03-05 | 2019-10-11 | 安特里斯生物制药公司 | 口服递送的药物 |
| CN104055735B (zh) * | 2013-03-22 | 2016-08-03 | 深圳翰宇药业股份有限公司 | 一种萨摩鲁泰的脂质体及其制备方法 |
| KR20210086717A (ko) | 2013-05-02 | 2021-07-08 | 노보 노르디스크 에이/에스 | Glp-1 화합물의 경구 투여 |
| EP3080154B1 (en) | 2013-12-13 | 2018-02-07 | Sanofi | Dual glp-1/gip receptor agonists |
| TW201609796A (zh) | 2013-12-13 | 2016-03-16 | 賽諾菲公司 | 非醯化之艾塞那肽-4(exendin-4)胜肽類似物 |
| EP3080149A1 (en) | 2013-12-13 | 2016-10-19 | Sanofi | Dual glp-1/glucagon receptor agonists |
| WO2015086728A1 (en) | 2013-12-13 | 2015-06-18 | Sanofi | Exendin-4 peptide analogues as dual glp-1/gip receptor agonists |
| TW201625670A (zh) | 2014-04-07 | 2016-07-16 | 賽諾菲公司 | 衍生自exendin-4之雙重glp-1/升糖素受體促效劑 |
| TW201625669A (zh) | 2014-04-07 | 2016-07-16 | 賽諾菲公司 | 衍生自艾塞那肽-4(Exendin-4)之肽類雙重GLP-1/升糖素受體促效劑 |
| TW201625668A (zh) | 2014-04-07 | 2016-07-16 | 賽諾菲公司 | 作為胜肽性雙重glp-1/昇糖素受體激動劑之艾塞那肽-4衍生物 |
| US9932381B2 (en) | 2014-06-18 | 2018-04-03 | Sanofi | Exendin-4 derivatives as selective glucagon receptor agonists |
| DK3006045T3 (en) * | 2014-10-07 | 2017-07-17 | Cyprumed Gmbh | Pharmaceutical formulations for oral administration of peptide or protein drugs |
| CN105777872B (zh) * | 2014-12-16 | 2019-06-07 | 深圳翰宇药业股份有限公司 | 一种萨摩鲁肽的纯化方法 |
| JP6910950B2 (ja) | 2015-01-12 | 2021-07-28 | エンテリス・バイオファーマ・インコーポレイテッドEnteris Biopharma,Inc. | 固形経口剤形 |
| EP3250191B1 (en) * | 2015-01-29 | 2024-01-17 | Novo Nordisk A/S | Tablets comprising glp-1 agonist and enteric coating |
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| WO2016168388A2 (en) | 2015-04-14 | 2016-10-20 | Palatin Technologies, Inc. | Therapies for obesity, diabetes and related indications |
| AR105319A1 (es) | 2015-06-05 | 2017-09-27 | Sanofi Sa | Profármacos que comprenden un conjugado agonista dual de glp-1 / glucagón conector ácido hialurónico |
| AR105284A1 (es) | 2015-07-10 | 2017-09-20 | Sanofi Sa | Derivados de exendina-4 como agonistas peptídicos duales específicos de los receptores de glp-1 / glucagón |
| JP7053480B2 (ja) | 2016-03-03 | 2022-04-12 | ノヴォ ノルディスク アー/エス | Glp-1誘導体及びその使用 |
| ES2928007T3 (es) | 2016-04-28 | 2022-11-14 | Novo Nordisk As | Semaglutida en afecciones cardiovasculares |
| WO2018033927A1 (en) | 2016-08-17 | 2018-02-22 | Entera Bio Ltd. | Formulations for oral administration of active agents |
| JOP20190060A1 (ar) | 2016-09-26 | 2019-03-26 | Chugai Pharmaceutical Co Ltd | مشتق بيرازولو بيريدين له تأثير مساعد لمستقبل glp-1 |
| TWI789391B (zh) * | 2017-04-25 | 2023-01-11 | 日商大塚製藥股份有限公司 | 具有可攝取事件標記的利欣諾普組成物 |
| AR112015A1 (es) * | 2017-06-09 | 2019-09-11 | Novo Nordisk As | Composiciones sólidas para administración oral |
| US11291629B2 (en) | 2017-06-27 | 2022-04-05 | Bioserentach Co., Ltd. | Mucoadhesive oral preparation |
| MX2020001525A (es) | 2017-08-24 | 2020-03-20 | Novo Nordisk As | Composiciones de peptido similar al glucagon tipo 1 (glp-1) y sus usos. |
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| CN111683676B (zh) * | 2018-02-02 | 2024-06-18 | 诺和诺德股份有限公司 | 包含glp-1激动剂、n-(8-(2-羟基苯甲酰基)氨基)辛酸的盐和润滑剂的固体组合物 |
| TWI829687B (zh) | 2018-05-07 | 2024-01-21 | 丹麥商諾佛 儂迪克股份有限公司 | 包含glp-1促效劑與n-(8-(2-羥基苯甲醯基)胺基)辛酸之鹽的固體組成物 |
| CN120617158A (zh) | 2018-10-26 | 2025-09-12 | 诺和诺德股份有限公司 | 稳定的司美鲁肽组合物及其用途 |
| US20220072493A1 (en) | 2019-01-24 | 2022-03-10 | Novo Nordisk A/S | Roller compactor and method of dry granulation using a roller compactor |
| US12458612B2 (en) | 2019-04-10 | 2025-11-04 | Genfit | Combination therapy comprising compounds of formula (I) and GLP-1 receptor agonists |
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