JP2019516795A5 - - Google Patents

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JP2019516795A5
JP2019516795A5 JP2019512951A JP2019512951A JP2019516795A5 JP 2019516795 A5 JP2019516795 A5 JP 2019516795A5 JP 2019512951 A JP2019512951 A JP 2019512951A JP 2019512951 A JP2019512951 A JP 2019512951A JP 2019516795 A5 JP2019516795 A5 JP 2019516795A5
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salt
alkoxy
halogen
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JP2019512951A 2016-05-18 2017-05-18 （Ｓ）－Ｎ－（５－（（Ｒ）－２－（２，５－ジフルオロフェニル）ピロリジン－１－イル）－ピラゾロ［１，５－ａ］ピリミジン－３－イル）－３－ヒドロキシピロリジン－１－カルボキサミドの調製 Active JP7443057B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662338359P 2016-05-18 2016-05-18
US62/338,359 2016-05-18
PCT/US2017/033257 WO2017201241A1 (en) 2016-05-18 2017-05-18 Preparation of (s)-n-(5-((r)-2-(2,5-difluorophenyl)pyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidin-3-y l)-3-hydroxypyrrolidine-1-carboxamide

Publications (3)

Publication Number Publication Date
JP2019516795A JP2019516795A (ja) 2019-06-20
JP2019516795A5 true JP2019516795A5 (enExample) 2020-07-02
JP7443057B2 JP7443057B2 (ja) 2024-03-05

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JP2019512951A Active JP7443057B2 (ja) 2016-05-18 2017-05-18 （Ｓ）－Ｎ－（５－（（Ｒ）－２－（２，５－ジフルオロフェニル）ピロリジン－１－イル）－ピラゾロ［１，５－ａ］ピリミジン－３－イル）－３－ヒドロキシピロリジン－１－カルボキサミドの調製

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US (1) US11214571B2 (enExample)
EP (2) EP3458456B1 (enExample)
JP (1) JP7443057B2 (enExample)
KR (1) KR102566858B1 (enExample)
CN (1) CN110049987B (enExample)
AU (1) AU2017268371B2 (enExample)
CA (1) CA3024603A1 (enExample)
CL (1) CL2018003264A1 (enExample)
CO (1) CO2018013015A2 (enExample)
DK (2) DK3458456T3 (enExample)
ES (2) ES2952056T3 (enExample)
FI (1) FI3800189T3 (enExample)
HR (2) HRP20230704T1 (enExample)
HU (2) HUE063877T2 (enExample)
IL (1) IL262964B (enExample)
LT (2) LT3458456T (enExample)
MX (1) MX392604B (enExample)
PE (1) PE20190437A1 (enExample)
PL (2) PL3800189T3 (enExample)
PT (2) PT3800189T (enExample)
RS (2) RS61463B1 (enExample)
RU (1) RU2745953C2 (enExample)
SG (1) SG11201810245WA (enExample)
SI (2) SI3458456T1 (enExample)
UA (1) UA127826C2 (enExample)
WO (1) WO2017201241A1 (enExample)
ZA (1) ZA201808534B (enExample)

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CN115872905B (zh) * 2021-09-29 2024-08-09 凯特立斯（深圳）科技有限公司 一种拉罗替尼中间体的制备方法
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