BR9812644A - Quinolonas antimicrobianas, suas composições eaplicações - Google Patents

Quinolonas antimicrobianas, suas composições eaplicações

Info

Publication number
BR9812644A
BR9812644A BR9812644-0A BR9812644A BR9812644A BR 9812644 A BR9812644 A BR 9812644A BR 9812644 A BR9812644 A BR 9812644A BR 9812644 A BR9812644 A BR 9812644A
Authority
BR
Brazil
Prior art keywords
applications
antimicrobial
compounds
compositions
quinolones
Prior art date
Application number
BR9812644-0A
Other languages
English (en)
Other versions
BR9812644B1 (pt
Inventor
Benoit Ledoussal
Ji-In Kim Almstead
Jeffrey Lyle Gray
Xiufeng Eric Hu
Original Assignee
Procter & Gamble
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Procter & Gamble filed Critical Procter & Gamble
Publication of BR9812644A publication Critical patent/BR9812644A/pt
Publication of BR9812644B1 publication Critical patent/BR9812644B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Abstract

Patente de Invenção: "QUINOLONAS ANTIMICROBIANAS,SUAS COMPOSIçõES E APLICAçõES". A presente invençãorefere-se a novos compostos antimicrobianos de fórmula (1) em queX, R~ 1~, R~ 3~, R~ 5~, R~ 6~ e R~ 8~ são definidos nasreivindicações, e a seus isómeros óticos, diastereómeros ouenantiómeros, bem como sais, hidratos e ésteres bioidrolisáveis,amidas e imidas dos mesmos farmaceuticamente aceitáveis, e acomposições e aplicações dos compostos referidos. A invençãotambém se refere a compostos derivados destes compostos tendoaplicações antimicrobianas.
BRPI9812644-0A 1997-09-15 1998-09-15 quinolonas antimicrobianas, composição farmacêutica e uso das mesmas. BR9812644B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5889197P 1997-09-15 1997-09-15
US13985998A 1998-08-25 1998-08-25
PCT/US1998/019138 WO1999014214A1 (en) 1997-09-15 1998-09-15 Antimicrobial quinolones, their compositions and uses

Publications (2)

Publication Number Publication Date
BR9812644A true BR9812644A (pt) 2001-12-18
BR9812644B1 BR9812644B1 (pt) 2010-07-13

Family

ID=26738133

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI9812644-0A BR9812644B1 (pt) 1997-09-15 1998-09-15 quinolonas antimicrobianas, composição farmacêutica e uso das mesmas.

Country Status (31)

Country Link
US (3) US6329391B1 (pt)
EP (1) EP1015445B1 (pt)
JP (1) JP4669607B2 (pt)
KR (1) KR100423778B1 (pt)
CN (1) CN1264837C (pt)
AR (1) AR013493A1 (pt)
AT (1) ATE423776T1 (pt)
AU (1) AU735186B2 (pt)
BR (1) BR9812644B1 (pt)
CA (1) CA2303389C (pt)
CO (1) CO4970702A1 (pt)
CY (1) CY1110255T1 (pt)
CZ (1) CZ299554B6 (pt)
DE (1) DE69840599D1 (pt)
DK (1) DK1015445T3 (pt)
ES (1) ES2321042T3 (pt)
HK (1) HK1030415A1 (pt)
HU (1) HUP0100051A3 (pt)
ID (1) ID24703A (pt)
IL (2) IL135036A0 (pt)
MY (1) MY138335A (pt)
NO (1) NO323563B1 (pt)
NZ (1) NZ503740A (pt)
PE (1) PE128799A1 (pt)
PL (1) PL339408A1 (pt)
PT (1) PT1015445E (pt)
RU (1) RU2193558C2 (pt)
SA (1) SA99191136B1 (pt)
SK (1) SK286420B6 (pt)
TR (2) TR200001435T2 (pt)
WO (1) WO1999014214A1 (pt)

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BR112012009583A2 (pt) * 2009-10-23 2015-09-29 Vertex Pharma processo para preparação de moduladores de regulador de condutância de transmembrana de fibrose cística
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CN102746223B (zh) * 2012-07-30 2013-10-23 浙江新东港药业股份有限公司 一种氟哌酸与氯哌酸的分离方法
CN103819401B (zh) * 2012-11-19 2016-04-13 浙江中欣氟材股份有限公司 1-环丙基-4-氧代-7-氟-8-甲氧基-1,4-二氢喹啉-3-羧酸的合成方法
US20160326165A1 (en) 2013-12-26 2016-11-10 Kinki University Alkoxycarbonyl hemiacetal-type ester prodrug of pyridone carboxylic acid antibacterial drug
RU2636751C1 (ru) 2016-11-02 2017-12-01 федеральное государственное автономное образовательное учреждение высшего образования "Казанский (Приволжский) федеральный университет" (ФГАОУ ВО КФУ) Антибактериальные средства на основе производных ципрофлоксацина
CN114008031A (zh) 2019-10-23 2022-02-01 太景生物科技股份有限公司 喹诺酮羧酸衍生物

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ATE423776T1 (de) 2009-03-15
EP1015445B1 (en) 2009-02-25
CA2303389C (en) 2007-07-17
ES2321042T3 (es) 2009-06-01
US7868021B2 (en) 2011-01-11
US6329391B1 (en) 2001-12-11
NZ503740A (en) 2002-09-27
JP4669607B2 (ja) 2011-04-13
IL135036A0 (en) 2001-05-20
TR200001435T2 (tr) 2000-08-21
NO20001340D0 (no) 2000-03-15
US20090111851A1 (en) 2009-04-30
SK286420B6 (sk) 2008-09-05
EP1015445A1 (en) 2000-07-05
WO1999014214A1 (en) 1999-03-25
CN1278813A (zh) 2001-01-03
NO20001340L (no) 2000-05-15
HUP0100051A3 (en) 2002-08-28
TR200505120T2 (tr) 2006-08-21
AR013493A1 (es) 2000-12-27
CZ299554B6 (cs) 2008-09-03
MY138335A (en) 2009-05-29
SA99191136B1 (ar) 2006-07-30
AU735186B2 (en) 2001-07-05
SK3812000A3 (en) 2000-09-12
KR20010024007A (ko) 2001-03-26
DK1015445T3 (da) 2009-05-11
ID24703A (id) 2000-08-03
NO323563B1 (no) 2007-06-11
PT1015445E (pt) 2009-05-14
CO4970702A1 (es) 2000-11-07
RU2193558C2 (ru) 2002-11-27
CN1264837C (zh) 2006-07-19
JP2001516756A (ja) 2001-10-02
BR9812644B1 (pt) 2010-07-13
US7482454B2 (en) 2009-01-27
US20060100436A1 (en) 2006-05-11
HUP0100051A2 (hu) 2001-10-28
CZ2000931A3 (cs) 2000-08-16
CY1110255T1 (el) 2015-01-14
HK1030415A1 (en) 2001-05-04
DE69840599D1 (de) 2009-04-09
IL135036A (en) 2007-12-03
PE128799A1 (es) 2000-02-17
CA2303389A1 (en) 1999-03-25
KR100423778B1 (ko) 2004-03-24
AU9482998A (en) 1999-04-05
PL339408A1 (en) 2000-12-18

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