BR9812644A - Quinolonas antimicrobianas, suas composições eaplicações - Google Patents
Quinolonas antimicrobianas, suas composições eaplicaçõesInfo
- Publication number
- BR9812644A BR9812644A BR9812644-0A BR9812644A BR9812644A BR 9812644 A BR9812644 A BR 9812644A BR 9812644 A BR9812644 A BR 9812644A BR 9812644 A BR9812644 A BR 9812644A
- Authority
- BR
- Brazil
- Prior art keywords
- applications
- antimicrobial
- compounds
- compositions
- quinolones
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Quinoline Compounds (AREA)
Abstract
Patente de Invenção: "QUINOLONAS ANTIMICROBIANAS,SUAS COMPOSIçõES E APLICAçõES". A presente invençãorefere-se a novos compostos antimicrobianos de fórmula (1) em queX, R~ 1~, R~ 3~, R~ 5~, R~ 6~ e R~ 8~ são definidos nasreivindicações, e a seus isómeros óticos, diastereómeros ouenantiómeros, bem como sais, hidratos e ésteres bioidrolisáveis,amidas e imidas dos mesmos farmaceuticamente aceitáveis, e acomposições e aplicações dos compostos referidos. A invençãotambém se refere a compostos derivados destes compostos tendoaplicações antimicrobianas.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US5889197P | 1997-09-15 | 1997-09-15 | |
US13985998A | 1998-08-25 | 1998-08-25 | |
PCT/US1998/019138 WO1999014214A1 (en) | 1997-09-15 | 1998-09-15 | Antimicrobial quinolones, their compositions and uses |
Publications (2)
Publication Number | Publication Date |
---|---|
BR9812644A true BR9812644A (pt) | 2001-12-18 |
BR9812644B1 BR9812644B1 (pt) | 2010-07-13 |
Family
ID=26738133
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI9812644-0A BR9812644B1 (pt) | 1997-09-15 | 1998-09-15 | quinolonas antimicrobianas, composição farmacêutica e uso das mesmas. |
Country Status (31)
Country | Link |
---|---|
US (3) | US6329391B1 (pt) |
EP (1) | EP1015445B1 (pt) |
JP (1) | JP4669607B2 (pt) |
KR (1) | KR100423778B1 (pt) |
CN (1) | CN1264837C (pt) |
AR (1) | AR013493A1 (pt) |
AT (1) | ATE423776T1 (pt) |
AU (1) | AU735186B2 (pt) |
BR (1) | BR9812644B1 (pt) |
CA (1) | CA2303389C (pt) |
CO (1) | CO4970702A1 (pt) |
CY (1) | CY1110255T1 (pt) |
CZ (1) | CZ299554B6 (pt) |
DE (1) | DE69840599D1 (pt) |
DK (1) | DK1015445T3 (pt) |
ES (1) | ES2321042T3 (pt) |
HK (1) | HK1030415A1 (pt) |
HU (1) | HUP0100051A3 (pt) |
ID (1) | ID24703A (pt) |
IL (2) | IL135036A0 (pt) |
MY (1) | MY138335A (pt) |
NO (1) | NO323563B1 (pt) |
NZ (1) | NZ503740A (pt) |
PE (1) | PE128799A1 (pt) |
PL (1) | PL339408A1 (pt) |
PT (1) | PT1015445E (pt) |
RU (1) | RU2193558C2 (pt) |
SA (1) | SA99191136B1 (pt) |
SK (1) | SK286420B6 (pt) |
TR (2) | TR200505120T2 (pt) |
WO (1) | WO1999014214A1 (pt) |
Families Citing this family (48)
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EP1015445B1 (en) * | 1997-09-15 | 2009-02-25 | The Procter & Gamble Company | Antimicrobial quinolones, their compositions and uses |
US6387928B1 (en) | 1997-09-15 | 2002-05-14 | The Procter & Gamble Co. | Antimicrobial quinolones, their compositions and uses |
ES2244248T3 (es) * | 1998-11-24 | 2005-12-01 | Daiichi Pharmaceutical Co., Ltd. | Derivados de aminometilpirrolidina sustituidos por cicloalquilos. |
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US6750224B1 (en) | 1999-05-07 | 2004-06-15 | Wockhardt Limited | Antibacterial optically pure benzoquinolizine carboxylic acids, processes, compositions and methods of treatment |
US6514986B2 (en) | 2000-11-22 | 2003-02-04 | Wockhardt Limited | Chiral fluoroquinolone arginine salt forms |
US6608078B2 (en) | 2000-05-08 | 2003-08-19 | Wockhardt Limited | Antibacterial chiral 8-(substituted piperidino)-benzo [i,j] quinolizines, processes, compositions and methods of treatment |
US7098219B2 (en) | 2000-08-01 | 2006-08-29 | Wockhart Limited | Inhibitors of cellular efflux pumps of microbes |
KR100777149B1 (ko) | 2000-11-20 | 2007-11-19 | 다이이찌 세이야꾸 가부시기가이샤 | 데할로게노 화합물 |
AU3089102A (en) * | 2000-12-14 | 2002-06-24 | Procter & Gamble | Antimicrobial quinolones |
US6878713B2 (en) | 2001-04-25 | 2005-04-12 | Wockhardt Limited | Generation triple-targeting, chiral, broad-spectrum antimicrobial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation, compositions and use as medicaments |
US6964966B2 (en) | 2001-04-25 | 2005-11-15 | Wockhardt Limited | Generation triple-targeting, chiral, broad-spectrum antimicrobial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation, compositions and use as medicaments |
WO2003099815A1 (en) | 2002-05-28 | 2003-12-04 | Wockhardt Limited | Crystalline fluoroquinolone arginine salt form |
US6900224B2 (en) * | 2002-07-31 | 2005-05-31 | The Procter & Gamble Company | Antimicrobial quinolones, their compositions and uses |
KR100742012B1 (ko) | 2002-11-21 | 2007-07-23 | 화이자 프로덕츠 인코포레이티드 | 3-아미노-피페리딘 유도체 및 그의 제조 방법 |
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RU2553989C2 (ru) * | 2009-10-23 | 2015-06-20 | Вертекс Фармасьютикалз Инкорпорейтед | Способ получения модуляторов регулятора трансмембранной проводимости кистозного фиброза |
JP5766278B2 (ja) * | 2010-05-11 | 2015-08-19 | サノフイ | 置換されたn−アルキルおよびn−アシルテトラヒドロ−イソキノリン誘導体、それらの製造および治療上の使用 |
CN102746223B (zh) * | 2012-07-30 | 2013-10-23 | 浙江新东港药业股份有限公司 | 一种氟哌酸与氯哌酸的分离方法 |
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