SK286420B6 - Zlúčenina so štruktúrou chinolónu, farmaceutický prostriedok s jej obsahom a jej použitie - Google Patents

Zlúčenina so štruktúrou chinolónu, farmaceutický prostriedok s jej obsahom a jej použitie Download PDF

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Publication number
SK286420B6
SK286420B6 SK381-2000A SK3812000A SK286420B6 SK 286420 B6 SK286420 B6 SK 286420B6 SK 3812000 A SK3812000 A SK 3812000A SK 286420 B6 SK286420 B6 SK 286420B6
Authority
SK
Slovakia
Prior art keywords
methoxy
cyclopropyl
dihydro
oxo
ethyl
Prior art date
Application number
SK381-2000A
Other languages
English (en)
Slovak (sk)
Other versions
SK3812000A3 (en
Inventor
Benoir Ledoussal
Ji-In Kim Almstead
Jeffrey Lyle Gray
Xiufeng Eric Hu
Original Assignee
The Procter & Gamble Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by The Procter & Gamble Company filed Critical The Procter & Gamble Company
Publication of SK3812000A3 publication Critical patent/SK3812000A3/sk
Publication of SK286420B6 publication Critical patent/SK286420B6/sk

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Quinoline Compounds (AREA)
SK381-2000A 1997-09-15 1998-09-15 Zlúčenina so štruktúrou chinolónu, farmaceutický prostriedok s jej obsahom a jej použitie SK286420B6 (sk)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5889197P 1997-09-15 1997-09-15
US13985998A 1998-08-25 1998-08-25
PCT/US1998/019138 WO1999014214A1 (en) 1997-09-15 1998-09-15 Antimicrobial quinolones, their compositions and uses

Publications (2)

Publication Number Publication Date
SK3812000A3 SK3812000A3 (en) 2000-09-12
SK286420B6 true SK286420B6 (sk) 2008-09-05

Family

ID=26738133

Family Applications (1)

Application Number Title Priority Date Filing Date
SK381-2000A SK286420B6 (sk) 1997-09-15 1998-09-15 Zlúčenina so štruktúrou chinolónu, farmaceutický prostriedok s jej obsahom a jej použitie

Country Status (31)

Country Link
US (3) US6329391B1 (pt)
EP (1) EP1015445B1 (pt)
JP (1) JP4669607B2 (pt)
KR (1) KR100423778B1 (pt)
CN (1) CN1264837C (pt)
AR (1) AR013493A1 (pt)
AT (1) ATE423776T1 (pt)
AU (1) AU735186B2 (pt)
BR (1) BR9812644B1 (pt)
CA (1) CA2303389C (pt)
CO (1) CO4970702A1 (pt)
CY (1) CY1110255T1 (pt)
CZ (1) CZ299554B6 (pt)
DE (1) DE69840599D1 (pt)
DK (1) DK1015445T3 (pt)
ES (1) ES2321042T3 (pt)
HK (1) HK1030415A1 (pt)
HU (1) HUP0100051A3 (pt)
ID (1) ID24703A (pt)
IL (2) IL135036A0 (pt)
MY (1) MY138335A (pt)
NO (1) NO323563B1 (pt)
NZ (1) NZ503740A (pt)
PE (1) PE128799A1 (pt)
PL (1) PL339408A1 (pt)
PT (1) PT1015445E (pt)
RU (1) RU2193558C2 (pt)
SA (1) SA99191136B1 (pt)
SK (1) SK286420B6 (pt)
TR (2) TR200505120T2 (pt)
WO (1) WO1999014214A1 (pt)

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US6514986B2 (en) 2000-11-22 2003-02-04 Wockhardt Limited Chiral fluoroquinolone arginine salt forms
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FR2937034B1 (fr) * 2008-10-10 2012-11-23 Novexel Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens
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JP2012512172A (ja) * 2008-12-15 2012-05-31 タイゲン バイオテクノロジー カンパニー，リミテッド ピペリジン誘導体の立体選択的合成
CN102648182A (zh) * 2009-10-23 2012-08-22 沃泰克斯药物股份有限公司 用于制备囊性纤维化跨膜传导调节因子的调节剂的方法
EP2569303A1 (en) * 2010-05-11 2013-03-20 Sanofi Substituted n-alkyl and n-acyl tetrahydro-isoquinoline derivatives, preparation and therapeutic use thereof
CN102746223B (zh) * 2012-07-30 2013-10-23 浙江新东港药业股份有限公司 一种氟哌酸与氯哌酸的分离方法
CN103819401B (zh) * 2012-11-19 2016-04-13 浙江中欣氟材股份有限公司 1-环丙基-4-氧代-7-氟-8-甲氧基-1,4-二氢喹啉-3-羧酸的合成方法
JP2015143209A (ja) 2013-12-26 2015-08-06 学校法人近畿大学 ピリドンカルボン酸系抗菌薬のアルコキシカルボニルヘミアセタール型エステルプロドラッグ
RU2636751C1 (ru) 2016-11-02 2017-12-01 федеральное государственное автономное образовательное учреждение высшего образования "Казанский (Приволжский) федеральный университет" (ФГАОУ ВО КФУ) Антибактериальные средства на основе производных ципрофлоксацина
TW202128645A (zh) * 2019-10-23 2021-08-01 太景生物科技股份有限公司 喹諾酮羧酸衍生物
CA3170415A1 (en) * 2020-03-03 2021-09-10 Anna M. Ericsson Compounds targeting rna-binding proteins or rna-modifying proteins

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