SK280295B6 - Farmaceutický prostriedok s riadeným uvoľňovaním o - Google Patents
Farmaceutický prostriedok s riadeným uvoľňovaním o Download PDFInfo
- Publication number
- SK280295B6 SK280295B6 SK922-93A SK92293A SK280295B6 SK 280295 B6 SK280295 B6 SK 280295B6 SK 92293 A SK92293 A SK 92293A SK 280295 B6 SK280295 B6 SK 280295B6
- Authority
- SK
- Slovakia
- Prior art keywords
- oxycodone
- oxy
- hours
- tablets
- controlled release
- Prior art date
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- BRUQQQPBMZOVGD-XFKAJCMBSA-N Oxycodone Chemical compound O=C([C@@H]1O2)CC[C@@]3(O)[C@H]4CC5=CC=C(OC)C2=C5[C@@]13CCN4C BRUQQQPBMZOVGD-XFKAJCMBSA-N 0.000 title claims abstract description 147
- 229960002085 oxycodone Drugs 0.000 title claims abstract description 130
- 239000008194 pharmaceutical composition Substances 0.000 title claims abstract description 35
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- QCQCHGYLTSGIGX-GHXANHINSA-N 4-[[(3ar,5ar,5br,7ar,9s,11ar,11br,13as)-5a,5b,8,8,11a-pentamethyl-3a-[(5-methylpyridine-3-carbonyl)amino]-2-oxo-1-propan-2-yl-4,5,6,7,7a,9,10,11,11b,12,13,13a-dodecahydro-3h-cyclopenta[a]chrysen-9-yl]oxy]-2,2-dimethyl-4-oxobutanoic acid Chemical compound N([C@@]12CC[C@@]3(C)[C@]4(C)CC[C@H]5C(C)(C)[C@@H](OC(=O)CC(C)(C)C(O)=O)CC[C@]5(C)[C@H]4CC[C@@H]3C1=C(C(C2)=O)C(C)C)C(=O)C1=CN=CC(C)=C1 QCQCHGYLTSGIGX-GHXANHINSA-N 0.000 claims description 2
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5015—Organic compounds, e.g. fats, sugars
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/800,549 US5266331A (en) | 1991-11-27 | 1991-11-27 | Controlled release oxycodone compositions |
| PCT/US1992/010146 WO1993010765A1 (en) | 1991-11-27 | 1992-11-25 | Controlled release oxycodone compositions |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| SK92293A3 SK92293A3 (en) | 1994-04-06 |
| SK280295B6 true SK280295B6 (sk) | 1999-11-08 |
Family
ID=25178688
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK922-93A SK280295B6 (sk) | 1991-11-27 | 1992-11-25 | Farmaceutický prostriedok s riadeným uvoľňovaním o |
Country Status (31)
| Country | Link |
|---|---|
| US (13) | US5266331A (pl) |
| EP (15) | EP2243484A3 (pl) |
| JP (2) | JP3375960B2 (pl) |
| KR (1) | KR100280973B1 (pl) |
| CN (2) | CN1165307C (pl) |
| AT (9) | ATE454150T1 (pl) |
| AU (1) | AU657027B2 (pl) |
| BG (1) | BG61753B1 (pl) |
| BR (1) | BR9205498A (pl) |
| CA (1) | CA2098738C (pl) |
| CZ (4) | CZ300183B6 (pl) |
| DE (10) | DE69233691T2 (pl) |
| DK (10) | DK1438959T3 (pl) |
| ES (9) | ES2339392T3 (pl) |
| FI (5) | FI113152B (pl) |
| GR (1) | GR3022273T3 (pl) |
| HK (6) | HK1068004A1 (pl) |
| HU (10) | HU227515B1 (pl) |
| IL (1) | IL103909A (pl) |
| MX (1) | MX9302968A (pl) |
| NO (6) | NO307028B3 (pl) |
| PH (1) | PH31679A (pl) |
| PL (2) | PL173574B1 (pl) |
| PT (8) | PT1327445E (pl) |
| RO (1) | RO115112B1 (pl) |
| RS (3) | RS50056B (pl) |
| RU (1) | RU2122411C1 (pl) |
| SK (1) | SK280295B6 (pl) |
| WO (1) | WO1993010765A1 (pl) |
| YU (1) | YU49495B (pl) |
| ZA (1) | ZA929227B (pl) |
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- 1992-11-25 BR BR9205498A patent/BR9205498A/pt not_active Application Discontinuation
- 1992-11-25 PL PL92300145A patent/PL172236B1/pl unknown
- 1992-11-27 ZA ZA929227A patent/ZA929227B/xx unknown
- 1992-11-27 IL IL10390992A patent/IL103909A/en not_active IP Right Cessation
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1993
- 1993-05-21 RS YUP-2005/0410A patent/RS50056B/sr unknown
- 1993-05-21 RS YUP-2005/0409A patent/RS50055B/sr unknown
- 1993-05-21 RS YUP-2005/0408A patent/RS50054B/sr unknown
- 1993-05-21 PH PH46222A patent/PH31679A/en unknown
- 1993-05-21 YU YU35893A patent/YU49495B/sh unknown
- 1993-05-25 CN CNB931063787A patent/CN1165307C/zh not_active Expired - Lifetime
- 1993-05-25 CN CNB011354526A patent/CN1245958C/zh not_active Expired - Lifetime
- 1993-07-20 BG BG97973A patent/BG61753B1/bg unknown
- 1993-07-23 FI FI933330A patent/FI113152B/fi not_active IP Right Cessation
- 1993-07-23 NO NO19932661A patent/NO307028B3/no not_active IP Right Cessation
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1995
- 1995-06-06 US US08/467,584 patent/US5508042A/en not_active Expired - Lifetime
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1997
- 1997-01-14 GR GR970400044T patent/GR3022273T3/el unknown
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1999
- 1999-04-01 CZ CZ19991153A patent/CZ292849B6/cs not_active IP Right Cessation
- 1999-12-23 NO NO19996447A patent/NO318890B1/no not_active IP Right Cessation
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2000
- 2000-12-08 DK DK200000364U patent/DK200000364U3/da active
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2001
- 2001-02-16 US US09/784,888 patent/US20010008639A1/en not_active Abandoned
- 2001-08-20 US US09/933,411 patent/US20020018810A1/en not_active Abandoned
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2002
- 2002-06-05 US US10/163,484 patent/US20030099704A1/en not_active Abandoned
- 2002-06-11 JP JP2002169981A patent/JP4016074B2/ja not_active Expired - Lifetime
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2003
- 2003-04-09 HK HK05100220A patent/HK1068004A1/xx not_active IP Right Cessation
- 2003-04-09 HK HK05105981A patent/HK1073255A1/xx not_active IP Right Cessation
- 2003-04-09 HK HK04100077A patent/HK1059210A1/xx not_active IP Right Cessation
- 2003-04-09 HK HK03102581A patent/HK1051803A1/xx not_active IP Right Cessation
- 2003-04-09 HK HK04100076A patent/HK1059209A1/xx not_active IP Right Cessation
- 2003-04-09 HK HK04100081A patent/HK1058474A1/xx not_active IP Right Cessation
- 2003-11-12 US US10/706,371 patent/US20040096500A1/en not_active Abandoned
- 2003-11-12 US US10/706,496 patent/US20040105887A1/en not_active Abandoned
- 2003-12-22 FI FI20031889A patent/FI116658B/fi not_active IP Right Cessation
- 2003-12-22 FI FI20031890A patent/FI118251B/fi not_active IP Right Cessation
- 2003-12-22 FI FI20031891A patent/FI118252B/fi not_active IP Right Cessation
- 2003-12-22 FI FI20031888A patent/FI118250B/fi not_active IP Right Cessation
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2004
- 2004-03-24 US US10/809,766 patent/US20040185098A1/en not_active Abandoned
- 2004-04-22 NO NO20041939A patent/NO325483B1/no not_active IP Right Cessation
- 2004-04-22 NO NO20041667A patent/NO322378B1/no unknown
- 2004-04-22 NO NO20041662A patent/NO323334B1/no unknown
- 2004-08-04 NO NO20043264A patent/NO20043264L/no not_active Application Discontinuation
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2005
- 2005-08-17 US US11/207,144 patent/US20060057210A1/en not_active Abandoned
- 2005-12-16 US US11/303,553 patent/US20060099255A1/en not_active Abandoned
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2006
- 2006-01-12 US US11/332,644 patent/US20060165792A1/en not_active Abandoned
- 2006-01-12 US US11/332,632 patent/US20060165791A1/en not_active Abandoned
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| PC4A | Assignment and transfer of rights |
Owner name: MUNDIPHARMA MEDICAL GMBH, BASEL, CH Free format text: FORMER OWNER: PURDUE PHARMA L.P., STAMFORD, CONNECTICUT, US Effective date: 20091119 Owner name: PURDUE PHARMA L.P., STAMFORD, CONNECTICUT, US Free format text: FORMER OWNER: EURO-CELTIQUE, S. A., LUXEMBOURG, LU Effective date: 20091119 |
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| MK4A | Patent expired |
Expiry date: 20121125 |