SG10201801069QA - Sustained release dosage forms for a jak1 inhibitor - Google Patents

Sustained release dosage forms for a jak1 inhibitor

Info

Publication number
SG10201801069QA
SG10201801069QA SG10201801069QA SG10201801069QA SG10201801069QA SG 10201801069Q A SG10201801069Q A SG 10201801069QA SG 10201801069Q A SG10201801069Q A SG 10201801069QA SG 10201801069Q A SG10201801069Q A SG 10201801069QA SG 10201801069Q A SG10201801069Q A SG 10201801069QA
Authority
SG
Singapore
Prior art keywords
dosage forms
sustained release
release dosage
jak1 inhibitor
jak1
Prior art date
Application number
SG10201801069QA
Other languages
English (en)
Inventor
Krishnaswamy Yeleswaram
Bhavnish Parikh
Dilip P Modi
Trupti Sheth
Original Assignee
Incyte Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Incyte Corp filed Critical Incyte Corp
Publication of SG10201801069QA publication Critical patent/SG10201801069QA/en

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
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    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
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    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
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    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
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    • A61K9/20—Pills, tablets, discs, rods
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    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
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  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Neurology (AREA)
  • Dermatology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Inorganic Chemistry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Transplantation (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
SG10201801069QA 2013-08-07 2014-08-06 Sustained release dosage forms for a jak1 inhibitor SG10201801069QA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361863325P 2013-08-07 2013-08-07
US201361913066P 2013-12-06 2013-12-06

Publications (1)

Publication Number Publication Date
SG10201801069QA true SG10201801069QA (en) 2018-03-28

Family

ID=51383933

Family Applications (3)

Application Number Title Priority Date Filing Date
SG10201801069QA SG10201801069QA (en) 2013-08-07 2014-08-06 Sustained release dosage forms for a jak1 inhibitor
SG10201912203XA SG10201912203XA (en) 2013-08-07 2014-08-06 Sustained release dosage forms for a jak1 inhibitor
SG11201600815WA SG11201600815WA (en) 2013-08-07 2014-08-06 Sustained release dosage forms for a jak1 inhibitor

Family Applications After (2)

Application Number Title Priority Date Filing Date
SG10201912203XA SG10201912203XA (en) 2013-08-07 2014-08-06 Sustained release dosage forms for a jak1 inhibitor
SG11201600815WA SG11201600815WA (en) 2013-08-07 2014-08-06 Sustained release dosage forms for a jak1 inhibitor

Country Status (30)

Country Link
US (4) US9655854B2 (de)
EP (2) EP3030227B1 (de)
JP (5) JP6334700B2 (de)
KR (3) KR20160045081A (de)
CN (3) CN105579032A (de)
AU (3) AU2014305989B2 (de)
BR (1) BR122020001831A8 (de)
CA (2) CA2920108C (de)
CL (1) CL2016000292A1 (de)
CR (3) CR20190343A (de)
CY (1) CY1123314T1 (de)
DK (1) DK3030227T3 (de)
EA (1) EA201690357A1 (de)
ES (1) ES2792549T3 (de)
HR (1) HRP20200955T1 (de)
HU (1) HUE049345T2 (de)
IL (2) IL277554B2 (de)
LT (1) LT3030227T (de)
MX (2) MX2016001639A (de)
MY (1) MY195091A (de)
PE (2) PE20220579A1 (de)
PH (3) PH12016500243A1 (de)
PL (1) PL3030227T3 (de)
PT (1) PT3030227T (de)
RS (1) RS60469B1 (de)
SG (3) SG10201801069QA (de)
SI (1) SI3030227T1 (de)
TW (3) TWI789516B (de)
UA (1) UA120499C2 (de)
WO (1) WO2015021153A1 (de)

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