NO328651B1 - Syreaddisjonssalter av et hydropyridinderivat, medikamenter som inneholder disse, anvendelse av saltene til fremstilling av medikamenter og fremgangsmate for fremstilling av syreaddisjonssaltene av hydropyridinderivatet - Google Patents
Syreaddisjonssalter av et hydropyridinderivat, medikamenter som inneholder disse, anvendelse av saltene til fremstilling av medikamenter og fremgangsmate for fremstilling av syreaddisjonssaltene av hydropyridinderivatet Download PDFInfo
- Publication number
- NO328651B1 NO328651B1 NO20030022A NO20030022A NO328651B1 NO 328651 B1 NO328651 B1 NO 328651B1 NO 20030022 A NO20030022 A NO 20030022A NO 20030022 A NO20030022 A NO 20030022A NO 328651 B1 NO328651 B1 NO 328651B1
- Authority
- NO
- Norway
- Prior art keywords
- fluorobenzyl
- acetoxy
- tetrahydrothieno
- pyridine
- cyclopropylcarbonyl
- Prior art date
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- IUVKMZGDUIUOCP-BTNSXGMBSA-N quinbolone Chemical compound O([C@H]1CC[C@H]2[C@H]3[C@@H]([C@]4(C=CC(=O)C=C4CC3)C)CC[C@@]21C)C1=CCCC1 IUVKMZGDUIUOCP-BTNSXGMBSA-N 0.000 description 1
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pyridine Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2000205396 | 2000-07-06 | ||
| JP2000266780 | 2000-09-04 | ||
| PCT/JP2001/005764 WO2002004461A1 (fr) | 2000-07-06 | 2001-07-03 | Sels d'addition acides de dérivés hydropyridine |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20030022D0 NO20030022D0 (no) | 2003-01-03 |
| NO20030022L NO20030022L (no) | 2003-03-05 |
| NO328651B1 true NO328651B1 (no) | 2010-04-19 |
Family
ID=26595526
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20030022A NO328651B1 (no) | 2000-07-06 | 2003-01-03 | Syreaddisjonssalter av et hydropyridinderivat, medikamenter som inneholder disse, anvendelse av saltene til fremstilling av medikamenter og fremgangsmate for fremstilling av syreaddisjonssaltene av hydropyridinderivatet |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US6693115B2 (ja) |
| EP (2) | EP1728794B1 (ja) |
| KR (6) | KR20080021152A (ja) |
| CN (1) | CN1214031C (ja) |
| AT (2) | ATE398624T1 (ja) |
| AU (2) | AU2001267916B2 (ja) |
| BR (1) | BR0112168A (ja) |
| CA (2) | CA2415558C (ja) |
| CY (3) | CY1107554T1 (ja) |
| CZ (1) | CZ302990B6 (ja) |
| DE (2) | DE60124712T2 (ja) |
| DK (2) | DK1728794T3 (ja) |
| ES (2) | ES2276801T3 (ja) |
| HK (2) | HK1051362A1 (ja) |
| HU (2) | HU230762B1 (ja) |
| IL (2) | IL153546A0 (ja) |
| MX (1) | MXPA03000031A (ja) |
| NO (1) | NO328651B1 (ja) |
| NZ (1) | NZ523416A (ja) |
| PL (1) | PL208386B1 (ja) |
| PT (2) | PT1728794E (ja) |
| RU (1) | RU2238275C1 (ja) |
| TW (1) | TWI290927B (ja) |
| WO (1) | WO2002004461A1 (ja) |
Families Citing this family (100)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100692934B1 (ko) * | 2000-12-25 | 2007-03-12 | 상꾜 가부시키가이샤 | 아스피린을 함유하는 의약 조성물 |
| RU2005104432A (ru) * | 2002-07-18 | 2005-08-10 | Санкио Компани, Лимитед (Jp) | Лекарственная композиция для лечения артериосклероза |
| EP1660183A2 (en) * | 2003-05-05 | 2006-05-31 | Eli Lilly and Company | Treating cardiovascular diseases with a compound of formula 1 (cs 747 - prasugrel; rn 150322-43-4) |
| US20060099262A1 (en) * | 2004-11-08 | 2006-05-11 | Biokey, Inc. | Methods and formulations for making controlled release oral dosage form |
| US8586085B2 (en) * | 2004-11-08 | 2013-11-19 | Biokey, Inc. | Methods and formulations for making pharmaceutical compositions containing bupropion |
| US20060099261A1 (en) * | 2004-11-08 | 2006-05-11 | Biokey, Inc. | Methods and formulations for making controlled release oral dosage form |
| CN1318428C (zh) * | 2005-02-23 | 2007-05-30 | 天津药物研究院 | 噻吩并吡啶取代的乙酰肼衍生物 |
| TWI318571B (en) * | 2005-06-10 | 2009-12-21 | Lilly Co Eli | Formulation of a thienopyridine platelet aggregation inhibitor |
| CA2612315A1 (en) * | 2005-06-17 | 2006-12-28 | Eli Lilly And Company | Dosage regimen for prasugrel |
| US20080214599A1 (en) * | 2005-08-19 | 2008-09-04 | John Thomas Brandt | Use of Par-1/Par-4 Inhibitors for Treating or Preventing Vascular Diseases |
| US8056072B2 (en) | 2005-10-31 | 2011-11-08 | Microsoft Corporation | Rebootless display driver upgrades |
| KR20150105419A (ko) | 2006-04-04 | 2015-09-16 | 케이지 액퀴지션 엘엘씨 | 항혈소판제와 산 억제제를 포함하는 경구 투여 형태 |
| TWI392681B (zh) | 2006-04-06 | 2013-04-11 | Daiichi Sankyo Co Ltd | 高純度普拉格雷及其酸加成鹽之製法 |
| EP2032521B1 (en) * | 2006-06-27 | 2009-10-28 | Sandoz AG | New method for salt preparation |
| US20100062066A1 (en) * | 2006-11-14 | 2010-03-11 | Acusphere, Inc | Formulations of Tetrahydropyridine Antiplatelet Agents for Parenteral or Oral Administration |
| JP5433235B2 (ja) * | 2006-12-07 | 2014-03-05 | 第一三共株式会社 | 固形製剤の製造方法 |
| JPWO2008069262A1 (ja) * | 2006-12-07 | 2010-03-25 | 第一三共株式会社 | 安定性が改善されたフィルムコーティング製剤 |
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