MX391408B - Inhibidores de biaril meta-pirimidina de cinasas. - Google Patents

Inhibidores de biaril meta-pirimidina de cinasas.

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Publication number
MX391408B
MX391408B MX2018008723A MX2018008723A MX391408B MX 391408 B MX391408 B MX 391408B MX 2018008723 A MX2018008723 A MX 2018008723A MX 2018008723 A MX2018008723 A MX 2018008723A MX 391408 B MX391408 B MX 391408B
Authority
MX
Mexico
Prior art keywords
meta
biaryl
kinase inhibitors
pyrimidine
pyrimidine kinase
Prior art date
Application number
MX2018008723A
Other languages
English (en)
Spanish (es)
Inventor
Jon Jianguo Cao
John Hood
Dan Lohse
Chi Ching Mak
Pherson Andrew Mc
Glenn Noronha
Ved PATHAK
Joel Renick
Richard M Soll
Binqi Zeng
Original Assignee
Impact Biomedicines Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Impact Biomedicines Inc filed Critical Impact Biomedicines Inc
Publication of MX391408B publication Critical patent/MX391408B/es

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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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