NZ592990A - Bi-aryl meta-pyrimidine inhibitors of kinases - Google Patents
Bi-aryl meta-pyrimidine inhibitors of kinasesInfo
- Publication number
- NZ592990A NZ592990A NZ592990A NZ59299006A NZ592990A NZ 592990 A NZ592990 A NZ 592990A NZ 592990 A NZ592990 A NZ 592990A NZ 59299006 A NZ59299006 A NZ 59299006A NZ 592990 A NZ592990 A NZ 592990A
- Authority
- NZ
- New Zealand
- Prior art keywords
- kinases
- pyrimidine inhibitors
- aryl meta
- meta
- aryl
- Prior art date
Links
Classifications
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- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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- C07D207/06—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with radicals, containing only hydrogen and carbon atoms, attached to ring carbon atoms
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- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
- C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US73262905P | 2005-11-01 | 2005-11-01 | |
| US83800306P | 2006-08-15 | 2006-08-15 | |
| PCT/US2006/042044 WO2007053452A1 (en) | 2005-11-01 | 2006-10-26 | Bi-aryl meta-pyrimidine inhibitors of kinases |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NZ592990A true NZ592990A (en) | 2013-01-25 |
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ID=38006192
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NZ592990A NZ592990A (en) | 2005-11-01 | 2006-10-26 | Bi-aryl meta-pyrimidine inhibitors of kinases |
| NZ567851A NZ567851A (en) | 2005-11-01 | 2006-10-26 | Bi-aryl meta-pyrimidine inhibitors of kinases |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NZ567851A NZ567851A (en) | 2005-11-01 | 2006-10-26 | Bi-aryl meta-pyrimidine inhibitors of kinases |
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