PT1951684T - Inibidores de cinases de tipo biaril-meta-pirimidina - Google Patents

Inibidores de cinases de tipo biaril-meta-pirimidina

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Publication number
PT1951684T
PT1951684T PT68365832T PT06836583T PT1951684T PT 1951684 T PT1951684 T PT 1951684T PT 68365832 T PT68365832 T PT 68365832T PT 06836583 T PT06836583 T PT 06836583T PT 1951684 T PT1951684 T PT 1951684T
Authority
PT
Portugal
Prior art keywords
kinases
pyrimidine inhibitors
aryl meta
meta
aryl
Prior art date
Application number
PT68365832T
Other languages
English (en)
Portuguese (pt)
Inventor
Hood John
Cao Jianguo
Lohse* Daniel
Ching Mak Chi
Mc Pherson Andrew
Pathak* Ved
Renick Joel
M Soll Richard
Zeng Binqi
Original Assignee
Targegen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Targegen Inc filed Critical Targegen Inc
Publication of PT1951684T publication Critical patent/PT1951684T/pt

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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