JP2006522746A - 置換されたアミドの薬学的使用 - Google Patents

置換されたアミドの薬学的使用 Download PDF

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Publication number
JP2006522746A
JP2006522746A JP2006504353A JP2006504353A JP2006522746A JP 2006522746 A JP2006522746 A JP 2006522746A JP 2006504353 A JP2006504353 A JP 2006504353A JP 2006504353 A JP2006504353 A JP 2006504353A JP 2006522746 A JP2006522746 A JP 2006522746A
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Japan
Prior art keywords
alkyl
aryl
phenyl
hetaryl
methyl
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JP2006504353A
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Japanese (ja)
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JP2006522746A5 (https=
Inventor
アンデルセン、ヘンリク・スネ
カムペン、ギタ・カミラ・テイルガルト
クリステンセン、インゲ・ソガー
モゲンセン、ジョン・パトリック
ラルセン、アネット・ロセンダル
キルバーン、ジョン・ポール
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Novo Nordisk AS
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Novo Nordisk AS
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Publication of JP2006522746A publication Critical patent/JP2006522746A/ja
Publication of JP2006522746A5 publication Critical patent/JP2006522746A5/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
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    • A61K31/16—Amides, e.g. hydroxamic acids
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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