DD153374A5 - Verfahren zur herstellung von beta-lactamen - Google Patents

Verfahren zur herstellung von beta-lactamen Download PDF

Info

Publication number
DD153374A5
DD153374A5 DD80218818A DD21881880A DD153374A5 DD 153374 A5 DD153374 A5 DD 153374A5 DD 80218818 A DD80218818 A DD 80218818A DD 21881880 A DD21881880 A DD 21881880A DD 153374 A5 DD153374 A5 DD 153374A5
Authority
DD
German Democratic Republic
Prior art keywords
general formula
chlorine
protected
item
hydroxy
Prior art date
Application number
DD80218818A
Other languages
German (de)
English (en)
Inventor
Lowell D Hatfield
Larry C Blaszczak
Jack W Fisher
Charles A Bunnell
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27358615&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DD153374(A5) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US06/008,645 external-priority patent/US4223133A/en
Priority claimed from US06/008,647 external-priority patent/US4226986A/en
Priority claimed from US06/008,470 external-priority patent/US4211702A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of DD153374A5 publication Critical patent/DD153374A5/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04—Preparation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/02—Preparation
    • C07D501/04—Preparation from compounds already containing the ring or condensed ring systems, e.g. by dehydrogenation of the ring, by introduction, elimination or modification of substituents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DD80218818A 1979-02-01 1980-02-01 Verfahren zur herstellung von beta-lactamen DD153374A5 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US06/008,645 US4223133A (en) 1979-02-01 1979-02-01 Cephalosporin reduction process
US06/008,647 US4226986A (en) 1979-02-01 1979-02-01 Process for halogenation of β-lactam compounds
US06/008,470 US4211702A (en) 1979-02-01 1979-02-01 Process for preparation of penicillin and cephalosporin imino halides

Publications (1)

Publication Number Publication Date
DD153374A5 true DD153374A5 (de) 1982-01-06

Family

ID=27358615

Family Applications (1)

Application Number Title Priority Date Filing Date
DD80218818A DD153374A5 (de) 1979-02-01 1980-02-01 Verfahren zur herstellung von beta-lactamen

Country Status (32)

Country Link
EP (1) EP0014567B1 (ja)
JP (12) JPS55113789A (ja)
KR (1) KR830001901B1 (ja)
AT (1) AT372684B (ja)
AU (1) AU538175B2 (ja)
BE (1) BE881425A (ja)
BG (1) BG35899A3 (ja)
CA (1) CA1133468A (ja)
CH (3) CH656385A5 (ja)
DD (1) DD153374A5 (ja)
DE (1) DE3066119D1 (ja)
DK (2) DK163513C (ja)
ES (1) ES8101603A1 (ja)
FI (1) FI74968C (ja)
FR (1) FR2447924A1 (ja)
GB (1) GB2044256B (ja)
GR (1) GR72278B (ja)
IE (1) IE49377B1 (ja)
IL (1) IL59269A (ja)
IT (1) IT1193908B (ja)
LU (1) LU82120A1 (ja)
MA (1) MA18715A1 (ja)
MW (1) MW880A1 (ja)
MY (1) MY8500598A (ja)
NL (1) NL191791C (ja)
NO (1) NO160660C (ja)
NZ (1) NZ192749A (ja)
OA (1) OA06451A (ja)
PH (1) PH15158A (ja)
PL (4) PL128595B1 (ja)
PT (1) PT70744A (ja)
YU (4) YU22580A (ja)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2063129T3 (es) * 1988-06-22 1995-01-01 Lilly Co Eli Intermedio de la 1-carba(detia)cefalosporina.
EP1961636B1 (en) 2007-02-20 2013-04-24 Yamaha Hatsudoki Kabushiki Kaisha Hydraulic master cylinder and vehicle provided with the same
EP2823864B1 (en) 2012-03-09 2017-06-28 Tani, Shinichiro Training ladder
EP2906661B1 (de) 2012-10-11 2016-10-26 Merck Patent GmbH Materialien für organische elektrolumineszenzvorrichtungen
JP6202969B2 (ja) * 2013-10-01 2017-09-27 富士電機株式会社 情報処理装置、暗号化方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK118506B (da) * 1963-02-18 1970-08-31 Ciba Geigy Fremgangsmåde til fremstilling af 7-aminocephalosporansyre eller estere deraf.
US3641014A (en) * 1968-10-03 1972-02-08 Lilly Co Eli Reduction of delta**3-cephalosporin sulfoxides
US3925372A (en) * 1973-02-23 1975-12-09 Lilly Co Eli Alpha-aminoacyl-3-halo cephalosporins

Also Published As

Publication number Publication date
IL59269A0 (en) 1980-05-30
IL59269A (en) 1984-04-30
ATA50280A (de) 1983-03-15
JPH0372632B2 (ja) 1991-11-19
JPH0334983A (ja) 1991-02-14
JPH0334985A (ja) 1991-02-14
YU16383A (en) 1984-02-29
JPH0372634B2 (ja) 1991-11-19
AU5502980A (en) 1980-08-07
DK163667B (da) 1992-03-23
GR72278B (ja) 1983-10-11
JPH089629B2 (ja) 1996-01-31
NO160660B (no) 1989-02-06
JPH0517483A (ja) 1993-01-26
CH652405A5 (fr) 1985-11-15
EP0014567B1 (en) 1984-01-18
DK163513C (da) 1992-07-27
IT8019609A0 (it) 1980-01-31
DK179991D0 (da) 1991-10-30
EP0014567A1 (en) 1980-08-20
YU16483A (en) 1984-02-29
YU18283A (en) 1984-02-29
IT1193908B (it) 1988-08-31
JPH0532669A (ja) 1993-02-09
JPH0372631B2 (ja) 1991-11-19
AU538175B2 (en) 1984-08-02
MW880A1 (en) 1981-09-09
JPH054990A (ja) 1993-01-14
CH656385A5 (fr) 1986-06-30
NL191791C (nl) 1996-08-02
CA1133468A (en) 1982-10-12
PL129399B1 (en) 1984-05-31
PL221744A1 (ja) 1980-12-01
NO160660C (no) 1989-05-16
LU82120A1 (fr) 1980-04-23
GB2044256A (en) 1980-10-15
JPH0565513B2 (ja) 1993-09-17
DE3066119D1 (en) 1984-02-23
JPH0372633B2 (ja) 1991-11-19
PL128595B1 (en) 1984-02-29
PL129604B1 (en) 1984-05-31
YU44734B (en) 1991-02-28
JPH0334984A (ja) 1991-02-14
BG35899A3 (en) 1984-07-16
DK163513B (da) 1992-03-09
OA06451A (fr) 1981-07-31
DK163667C (da) 1992-08-17
JPH0371435B2 (ja) 1991-11-13
DK41480A (da) 1980-08-02
JPH0334982A (ja) 1991-02-14
FR2447924B1 (ja) 1983-10-21
IE49377B1 (en) 1985-10-02
PT70744A (en) 1980-02-01
JPH0334981A (ja) 1991-02-14
NL191791B (nl) 1996-04-01
NL8000545A (nl) 1980-08-05
ES488231A0 (es) 1980-12-16
DK179991A (da) 1991-10-30
KR830001943A (ko) 1983-05-19
JPH0649706B2 (ja) 1994-06-29
JPH0649705B2 (ja) 1994-06-29
FI74968C (fi) 1988-04-11
NO800251L (no) 1980-08-04
JPH0565514B2 (ja) 1993-09-17
FR2447924A1 (fr) 1980-08-29
JPH04356490A (ja) 1992-12-10
JPS55113789A (en) 1980-09-02
CH648318A5 (fr) 1985-03-15
JPH054991A (ja) 1993-01-14
GB2044256B (en) 1983-05-05
FI800303A (fi) 1980-08-02
ES8101603A1 (es) 1980-12-16
MY8500598A (en) 1985-12-31
JPH07121950B2 (ja) 1995-12-25
BE881425A (fr) 1980-07-30
JPH04364187A (ja) 1992-12-16
AT372684B (de) 1983-11-10
FI74968B (fi) 1987-12-31
JPH0372231B2 (ja) 1991-11-18
YU22580A (en) 1983-06-30
PL126947B1 (en) 1983-09-30
IE800190L (en) 1980-08-01
MA18715A1 (fr) 1980-10-01
PH15158A (en) 1982-08-24
KR830001901B1 (ko) 1983-09-19
NZ192749A (en) 1983-06-17

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