FR2447924A1 - Procede de preparation de composes b-lactame - Google Patents

Procede de preparation de composes b-lactame

Info

Publication number
FR2447924A1
FR2447924A1 FR8001968A FR8001968A FR2447924A1 FR 2447924 A1 FR2447924 A1 FR 2447924A1 FR 8001968 A FR8001968 A FR 8001968A FR 8001968 A FR8001968 A FR 8001968A FR 2447924 A1 FR2447924 A1 FR 2447924A1
Authority
FR
France
Prior art keywords
preparation
various
interesting
antibiotics
cephalosporins
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR8001968A
Other languages
English (en)
Other versions
FR2447924B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27358615&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FR2447924(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US06/008,645 external-priority patent/US4223133A/en
Priority claimed from US06/008,647 external-priority patent/US4226986A/en
Priority claimed from US06/008,470 external-priority patent/US4211702A/en
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of FR2447924A1 publication Critical patent/FR2447924A1/fr
Application granted granted Critical
Publication of FR2447924B1 publication Critical patent/FR2447924B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04—Preparation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/02—Preparation
    • C07D501/04—Preparation from compounds already containing the ring or condensed ring systems, e.g. by dehydrogenation of the ring, by introduction, elimination or modification of substituents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'INVENTION CONCERNE LA PREPARATION DE DIFFERENTS DERIVES DE B-LACTAME PAR UTILISATION D'AGENTS D'HALOGENATION DE TYPE COMPLEXE CINETIQUE PHOSPHITE DE TRIARYLEHALOGENE. L'UTILISATION DE QUANTITES VARIABLES DE CES DIFFERENTS REACTIFS SUR DIVERSES CEPHALOSPORINES ET PENICILLINES PERMET D'OBTENIR EN PARTICULIER LES IMINO-HALOGENURES, LES DERIVES HALOGENES EN POSITION C-3 DES CEPHALOSPORINES, LES FORMES SULFURES DES CEPHALOSPORINES A PARTIR DES FORMES SULFOXYDES, ETC. LES COMPOSES OBTENUS DANS CES PROCEDES SONT DES ANTIBIOTIQUES INTERESSANTS OU DES INTERMEDIAIRES PERMETTANT DE PREPARER DES ANTIBIOTIQUES INTERESSANTS.
FR8001968A 1979-02-01 1980-01-30 Procede de preparation de composes b-lactame Granted FR2447924A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US06/008,645 US4223133A (en) 1979-02-01 1979-02-01 Cephalosporin reduction process
US06/008,647 US4226986A (en) 1979-02-01 1979-02-01 Process for halogenation of β-lactam compounds
US06/008,470 US4211702A (en) 1979-02-01 1979-02-01 Process for preparation of penicillin and cephalosporin imino halides

Publications (2)

Publication Number Publication Date
FR2447924A1 true FR2447924A1 (fr) 1980-08-29
FR2447924B1 FR2447924B1 (fr) 1983-10-21

Family

ID=27358615

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8001968A Granted FR2447924A1 (fr) 1979-02-01 1980-01-30 Procede de preparation de composes b-lactame

Country Status (32)

Country Link
EP (1) EP0014567B1 (fr)
JP (12) JPS55113789A (fr)
KR (1) KR830001901B1 (fr)
AT (1) AT372684B (fr)
AU (1) AU538175B2 (fr)
BE (1) BE881425A (fr)
BG (1) BG35899A3 (fr)
CA (1) CA1133468A (fr)
CH (3) CH648318A5 (fr)
DD (1) DD153374A5 (fr)
DE (1) DE3066119D1 (fr)
DK (2) DK163513C (fr)
ES (1) ES8101603A1 (fr)
FI (1) FI74968C (fr)
FR (1) FR2447924A1 (fr)
GB (1) GB2044256B (fr)
GR (1) GR72278B (fr)
IE (1) IE49377B1 (fr)
IL (1) IL59269A (fr)
IT (1) IT1193908B (fr)
LU (1) LU82120A1 (fr)
MA (1) MA18715A1 (fr)
MW (1) MW880A1 (fr)
MY (1) MY8500598A (fr)
NL (1) NL191791C (fr)
NO (1) NO160660C (fr)
NZ (1) NZ192749A (fr)
OA (1) OA06451A (fr)
PH (1) PH15158A (fr)
PL (4) PL128595B1 (fr)
PT (1) PT70744A (fr)
YU (4) YU22580A (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2809711B2 (ja) * 1988-06-22 1998-10-15 イーライ・リリー・アンド・カンパニー １―カルバ（デチア）セファロスポリンの中間体
EP1961636B1 (fr) 2007-02-20 2013-04-24 Yamaha Hatsudoki Kabushiki Kaisha Cylindre maître hydraulique et véhicule doté de celui-ci
KR101466783B1 (ko) 2012-03-09 2014-11-28 신이치로 다니 트레이닝 래더
US9741942B2 (en) 2012-10-11 2017-08-22 Merck Patent Gmbh Materials for organic electroluminescent devices
JP6202969B2 (ja) * 2013-10-01 2017-09-27 富士電機株式会社 情報処理装置、暗号化方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK118506B (da) * 1963-02-18 1970-08-31 Ciba Geigy Fremgangsmåde til fremstilling af 7-aminocephalosporansyre eller estere deraf.
US3641014A (en) * 1968-10-03 1972-02-08 Lilly Co Eli Reduction of delta**3-cephalosporin sulfoxides
US3925372A (en) * 1973-02-23 1975-12-09 Lilly Co Eli Alpha-aminoacyl-3-halo cephalosporins

Also Published As

Publication number Publication date
CH652405A5 (fr) 1985-11-15
DE3066119D1 (en) 1984-02-23
NO160660C (no) 1989-05-16
MY8500598A (en) 1985-12-31
DK163667B (da) 1992-03-23
DK163513C (da) 1992-07-27
FI800303A (fi) 1980-08-02
EP0014567A1 (fr) 1980-08-20
JPH04364187A (ja) 1992-12-16
CH656385A5 (fr) 1986-06-30
BE881425A (fr) 1980-07-30
GB2044256A (en) 1980-10-15
IE800190L (en) 1980-08-01
EP0014567B1 (fr) 1984-01-18
JPH054991A (ja) 1993-01-14
PL128595B1 (en) 1984-02-29
AU5502980A (en) 1980-08-07
DK179991A (da) 1991-10-30
MW880A1 (en) 1981-09-09
JPH0372632B2 (fr) 1991-11-19
LU82120A1 (fr) 1980-04-23
YU16483A (en) 1984-02-29
JPH054990A (ja) 1993-01-14
IT1193908B (it) 1988-08-31
NL191791B (nl) 1996-04-01
GR72278B (fr) 1983-10-11
IT8019609A0 (it) 1980-01-31
AU538175B2 (en) 1984-08-02
KR830001901B1 (ko) 1983-09-19
DD153374A5 (de) 1982-01-06
JPH0334982A (ja) 1991-02-14
JPH0334983A (ja) 1991-02-14
FI74968C (fi) 1988-04-11
IL59269A0 (en) 1980-05-30
ES488231A0 (es) 1980-12-16
JPS55113789A (en) 1980-09-02
IE49377B1 (en) 1985-10-02
NZ192749A (en) 1983-06-17
PL126947B1 (en) 1983-09-30
CH648318A5 (fr) 1985-03-15
JPH0334984A (ja) 1991-02-14
YU22580A (en) 1983-06-30
MA18715A1 (fr) 1980-10-01
PH15158A (en) 1982-08-24
JPH0532669A (ja) 1993-02-09
PT70744A (en) 1980-02-01
JPH0334981A (ja) 1991-02-14
DK163513B (da) 1992-03-09
JPH089629B2 (ja) 1996-01-31
PL221744A1 (fr) 1980-12-01
JPH0565513B2 (fr) 1993-09-17
JPH0517483A (ja) 1993-01-26
JPH0372231B2 (fr) 1991-11-18
ATA50280A (de) 1983-03-15
DK179991D0 (da) 1991-10-30
JPH0371435B2 (fr) 1991-11-13
JPH0372631B2 (fr) 1991-11-19
JPH0649706B2 (ja) 1994-06-29
DK41480A (da) 1980-08-02
JPH0649705B2 (ja) 1994-06-29
IL59269A (en) 1984-04-30
ES8101603A1 (es) 1980-12-16
JPH04356490A (ja) 1992-12-10
PL129604B1 (en) 1984-05-31
GB2044256B (en) 1983-05-05
AT372684B (de) 1983-11-10
YU44734B (en) 1991-02-28
NL8000545A (nl) 1980-08-05
OA06451A (fr) 1981-07-31
NO160660B (no) 1989-02-06
YU16383A (en) 1984-02-29
NO800251L (no) 1980-08-04
NL191791C (nl) 1996-08-02
CA1133468A (fr) 1982-10-12
DK163667C (da) 1992-08-17
JPH0372634B2 (fr) 1991-11-19
FR2447924B1 (fr) 1983-10-21
KR830001943A (ko) 1983-05-19
BG35899A3 (en) 1984-07-16
JPH0565514B2 (fr) 1993-09-17
JPH0334985A (ja) 1991-02-14
FI74968B (fi) 1987-12-31
JPH0372633B2 (fr) 1991-11-19
PL129399B1 (en) 1984-05-31
JPH07121950B2 (ja) 1995-12-25
YU18283A (en) 1984-02-29

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