BG63992B1 - Амидно съединение и приложение му като rho киназен инхибитор - Google Patents
Амидно съединение и приложение му като rho киназен инхибитор Download PDFInfo
- Publication number
- BG63992B1 BG63992B1 BG107195/2002A BG10719502A BG63992B1 BG 63992 B1 BG63992 B1 BG 63992B1 BG 107195/2002 A BG107195/2002 A BG 107195/2002A BG 10719502 A BG10719502 A BG 10719502A BG 63992 B1 BG63992 B1 BG 63992B1
- Authority
- BG
- Bulgaria
- Prior art keywords
- pharmaceutically acceptable
- isomer
- kinase inhibitor
- hydrogen
- salt
- Prior art date
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Cardiology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Heart & Thoracic Surgery (AREA)
- Virology (AREA)
- AIDS & HIV (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Molecular Biology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Ophthalmology & Optometry (AREA)
- Transplantation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Materials Applied To Surfaces To Minimize Adherence Of Mist Or Water (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Enzymes And Modification Thereof (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP21240996 | 1996-08-12 | ||
| PCT/JP1997/002793 WO1998006433A1 (fr) | 1996-08-12 | 1997-08-08 | MEDICAMENTS COMPRENANT UN INHIBITEUR DE LA Rho KINASE |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG63992B1 true BG63992B1 (bg) | 2003-09-30 |
Family
ID=16622116
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG107195/2002A BG107195A (en) | 1996-08-12 | 1999-03-12 | AMIDE COMPOUND AND ITS APPLICATION AS Rho KINASE INHIBITOR |
| BG103246A BG63991B1 (bg) | 1996-08-12 | 1999-03-12 | Фармацевтично средство, съдържащо rно киназен инхибитор |
| BG107195/2002A BG63992B1 (bg) | 1996-08-12 | 1999-03-12 | Амидно съединение и приложение му като rho киназен инхибитор |
| BG107645/2003A BG107645A (en) | 1996-08-12 | 2003-03-19 | MEDICINES COMPRISING Rho KINASE INHIBITOR |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG107195/2002A BG107195A (en) | 1996-08-12 | 1999-03-12 | AMIDE COMPOUND AND ITS APPLICATION AS Rho KINASE INHIBITOR |
| BG103246A BG63991B1 (bg) | 1996-08-12 | 1999-03-12 | Фармацевтично средство, съдържащо rно киназен инхибитор |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG107645/2003A BG107645A (en) | 1996-08-12 | 2003-03-19 | MEDICINES COMPRISING Rho KINASE INHIBITOR |
Country Status (26)
| Country | Link |
|---|---|
| US (3) | US6218410B1 (es) |
| EP (1) | EP0956865B2 (es) |
| JP (1) | JP3669711B2 (es) |
| KR (2) | KR100576148B1 (es) |
| CN (1) | CN100389828C (es) |
| AT (1) | ATE359822T1 (es) |
| AU (1) | AU738620B2 (es) |
| BG (4) | BG107195A (es) |
| BR (1) | BR9711154A (es) |
| CA (1) | CA2263425C (es) |
| CZ (1) | CZ301044B6 (es) |
| DE (1) | DE69737631T3 (es) |
| DK (1) | DK0956865T4 (es) |
| EE (1) | EE9900050A (es) |
| ES (1) | ES2286834T5 (es) |
| HK (1) | HK1022436A1 (es) |
| HU (1) | HU229864B1 (es) |
| IL (1) | IL128456A0 (es) |
| IS (1) | IS4973A (es) |
| NO (1) | NO990622L (es) |
| NZ (2) | NZ513800A (es) |
| PL (1) | PL331561A1 (es) |
| PT (1) | PT956865E (es) |
| RU (3) | RU2206321C2 (es) |
| SI (1) | SI0956865T2 (es) |
| WO (1) | WO1998006433A1 (es) |
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