TWI372624B - Azaindoles useful as inhibitors of jak and other protein kinases - Google Patents

Azaindoles useful as inhibitors of jak and other protein kinases

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Publication number
TWI372624B
TWI372624B TW094110160A TW94110160A TWI372624B TW I372624 B TWI372624 B TW I372624B TW 094110160 A TW094110160 A TW 094110160A TW 94110160 A TW94110160 A TW 94110160A TW I372624 B TWI372624 B TW I372624B
Authority
TW
Taiwan
Prior art keywords
jak
inhibitors
protein kinases
azaindoles useful
azaindoles
Prior art date
Application number
TW094110160A
Other languages
English (en)
Chinese (zh)
Other versions
TW200602052A (en
Inventor
Francesco G Salituro
Luc Farmer
Randy S Bethiel
Edmund M Harrington
Jeremy Green
John J Court
Jon H Come
David J Lauffer
Alex Aronov
Hayley Binch
Dean Boyall
Jean-Damien Charrier
Simon Everitt
Damien Fraysse
Michael Mortimore
Francoise Pierard
Daniel Robinson
Albert Pierce
Jian Wang
Joanne Pinder
Tiansheng Wang
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34971569&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TWI372624(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of TW200602052A publication Critical patent/TW200602052A/zh
Application granted granted Critical
Publication of TWI372624B publication Critical patent/TWI372624B/zh

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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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